HRP920923B1 - Dextrorotatory enantiomer of alpha-(4,5,6,7-tetrahydrothieno/3,2-c/pyrid-5-yl) (2-chlorophenyl)methyl acetate, its salts, and process for its preparation - Google Patents

Dextrorotatory enantiomer of alpha-(4,5,6,7-tetrahydrothieno/3,2-c/pyrid-5-yl) (2-chlorophenyl)methyl acetate, its salts, and process for its preparation

Info

Publication number
HRP920923B1
HRP920923B1 HR920923A HRP920923A HRP920923B1 HR P920923 B1 HRP920923 B1 HR P920923B1 HR 920923 A HR920923 A HR 920923A HR P920923 A HRP920923 A HR P920923A HR P920923 B1 HRP920923 B1 HR P920923B1
Authority
HR
Croatia
Prior art keywords
tetrahydrothieno
pyrid
chlorophenyl
alpha
salts
Prior art date
Application number
HR920923A
Other languages
English (en)
Inventor
Alain Badroc
Daniel Frehel
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26225786&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP920923(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from FR8702025A external-priority patent/FR2612929B1/fr
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of HRP920923A2 publication Critical patent/HRP920923A2/hr
Publication of HRP920923B1 publication Critical patent/HRP920923B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0055—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives
    • C07J41/0061—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives one of the carbon atoms being part of an amide group

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
HR920923A 1987-02-17 1992-10-02 Dextrorotatory enantiomer of alpha-(4,5,6,7-tetrahydrothieno/3,2-c/pyrid-5-yl) (2-chlorophenyl)methyl acetate, its salts, and process for its preparation HRP920923B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR8702025A FR2612929B1 (fr) 1987-02-17 1987-02-17 Enantiomere dextrogyre de 1a-(tetrahydro- 4,5,6,7 thieno (3,2-c) pyridyl-5) (chloro-2 phenyl)-acetate de methyle, son procede de preparation et les compositions pharmaceutiques le renfermant
FR878716516A FR2623810B2 (fr) 1987-02-17 1987-11-27 Sels de l'alpha-(tetrahydro-4,5,6,7 thieno(3,2-c) pyridyl-5) (chloro-2 phenyl) -acetate de methyle dextrogyre et compositions pharmaceutiques en contenant
YU23188A YU46748B (sh) 1987-02-17 1988-02-05 Dekstrogiri enantiomer metil alfa (4,5,6,7-tetrahidro-tien/,3,2-c/ pirid-5-il)-(2-hlorofenil)-acetata, njegove soli i postupak za dobijanje

Publications (2)

Publication Number Publication Date
HRP920923A2 HRP920923A2 (hr) 1994-04-30
HRP920923B1 true HRP920923B1 (en) 2001-12-31

Family

ID=26225786

Family Applications (1)

Application Number Title Priority Date Filing Date
HR920923A HRP920923B1 (en) 1987-02-17 1992-10-02 Dextrorotatory enantiomer of alpha-(4,5,6,7-tetrahydrothieno/3,2-c/pyrid-5-yl) (2-chlorophenyl)methyl acetate, its salts, and process for its preparation

Country Status (36)

Country Link
US (1) US4847265A (da)
EP (1) EP0281459B1 (da)
JP (1) JPH0645622B2 (da)
KR (1) KR960003615B1 (da)
AR (1) AR243891A1 (da)
AT (1) ATE121745T1 (da)
AU (1) AU597784B2 (da)
CA (1) CA1336777C (da)
CS (1) CS274420B2 (da)
CY (1) CY2087B1 (da)
DE (2) DE3853643T2 (da)
DK (1) DK173636B1 (da)
ES (1) ES2071621T4 (da)
FI (1) FI87216C (da)
FR (1) FR2623810B2 (da)
HK (1) HK1000093A1 (da)
HR (1) HRP920923B1 (da)
HU (2) HU197909B (da)
IE (1) IE66922B1 (da)
IL (1) IL85294A (da)
LU (1) LU90324I2 (da)
LV (1) LV5804B4 (da)
MA (1) MA21184A1 (da)
MX (1) MX9203026A (da)
MY (1) MY103198A (da)
NL (1) NL990002I1 (da)
NO (2) NO165924C (da)
NZ (1) NZ223475A (da)
OA (1) OA08808A (da)
PH (1) PH25960A (da)
PL (1) PL156689B1 (da)
PT (1) PT86726B (da)
RO (1) RO99191B1 (da)
SI (1) SI8810231A8 (da)
TN (1) TNSN88012A1 (da)
YU (1) YU46748B (da)

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CS96588A2 (en) 1990-09-12
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US4847265A (en) 1989-07-11
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