HRP20020021B1 - Method for preparing 2-(2-arylmorpholin-2-yl)ethanol derivatives and intermediates - Google Patents
Method for preparing 2-(2-arylmorpholin-2-yl)ethanol derivatives and intermediatesInfo
- Publication number
- HRP20020021B1 HRP20020021B1 HR20020021A HRP20020021A HRP20020021B1 HR P20020021 B1 HRP20020021 B1 HR P20020021B1 HR 20020021 A HR20020021 A HR 20020021A HR P20020021 A HRP20020021 A HR P20020021A HR P20020021 B1 HRP20020021 B1 HR P20020021B1
- Authority
- HR
- Croatia
- Prior art keywords
- intermediates
- arylmorpholin
- preparing
- ethanol derivatives
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
- C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
- C07C215/30—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings containing hydroxy groups and carbon atoms of six-membered aromatic rings bound to the same carbon atom of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
- C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
- C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
- C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
- C07C33/40—Halogenated unsaturated alcohols
- C07C33/46—Halogenated unsaturated alcohols containing only six-membered aromatic rings as cyclic parts
- C07C33/48—Halogenated unsaturated alcohols containing only six-membered aromatic rings as cyclic parts with unsaturation outside the aromatic rings
- C07C33/483—Monocyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
- C07C45/46—Friedel-Crafts reactions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/56—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
- C07C45/562—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with nitrogen as the only hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/08—Compounds containing oxirane rings with hydrocarbon radicals, substituted by halogen atoms, nitro radicals or nitroso radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Epoxy Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9909061A FR2796069B3 (fr) | 1999-07-09 | 1999-07-09 | Nouveaux procedes de preparation de derives de 2-(2- arylmorpholin-2-yl)ethanol substitues, enantiomeriquement purs, et composes intermediaires utiles dans ces procedes |
PCT/FR2000/001966 WO2001004105A1 (fr) | 1999-07-09 | 2000-07-07 | Preparation de derives de 2-(2-arylmorpholin-2-yl)ethanol et intermediaires |
Publications (2)
Publication Number | Publication Date |
---|---|
HRP20020021A2 HRP20020021A2 (en) | 2003-08-31 |
HRP20020021B1 true HRP20020021B1 (en) | 2004-10-31 |
Family
ID=9548041
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20020021A HRP20020021B1 (en) | 1999-07-09 | 2002-01-09 | Method for preparing 2-(2-arylmorpholin-2-yl)ethanol derivatives and intermediates |
Country Status (19)
Country | Link |
---|---|
US (3) | US7038044B1 (ja) |
EP (1) | EP1200417B1 (ja) |
JP (1) | JP3891840B2 (ja) |
CN (2) | CN1183121C (ja) |
AT (1) | ATE252566T1 (ja) |
AU (1) | AU6295600A (ja) |
BR (1) | BR0012324A (ja) |
CA (1) | CA2378002C (ja) |
CZ (1) | CZ300744B6 (ja) |
DE (1) | DE60006125T2 (ja) |
ES (1) | ES2208381T3 (ja) |
FR (1) | FR2796069B3 (ja) |
HR (1) | HRP20020021B1 (ja) |
HU (1) | HUP0202383A3 (ja) |
MX (1) | MXPA02000307A (ja) |
PL (1) | PL203213B1 (ja) |
SI (1) | SI1200417T1 (ja) |
SK (1) | SK286671B6 (ja) |
WO (1) | WO2001004105A1 (ja) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2796069B3 (fr) * | 1999-07-09 | 2001-08-24 | Sanofi Synthelabo | Nouveaux procedes de preparation de derives de 2-(2- arylmorpholin-2-yl)ethanol substitues, enantiomeriquement purs, et composes intermediaires utiles dans ces procedes |
JP2008273841A (ja) * | 2005-07-14 | 2008-11-13 | Zeria Pharmaceut Co Ltd | エチレンジアミン誘導体及びその製造法 |
MX355697B (es) | 2010-04-12 | 2018-04-27 | Supernus Pharmaceuticals Inc | Métodos para producir sales de viloxazina y polimorfos novedosos de las mismas. |
CN115448816B (zh) * | 2022-09-16 | 2024-04-12 | 中国石油大学(华东) | 一种β-氟代烯基醇的合成方法 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH396942A (de) * | 1959-03-21 | 1965-08-15 | Thomae Gmbh Dr K | Verfahren zur Herstellung basisch substituierter Carbinole |
BE790604A (fr) * | 1971-10-28 | 1973-04-26 | Sandoz Sa | Nouveaux aminoalcanols, leur preparation et leur application comme medicaments |
GB9108629D0 (en) * | 1991-04-23 | 1991-06-12 | Wellcome Found | Heterocyclic pharmaceutical compounds,preparation and use |
US5780466A (en) | 1995-01-30 | 1998-07-14 | Sanofi | Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present |
FR2729954B1 (fr) * | 1995-01-30 | 1997-08-01 | Sanofi Sa | Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant |
US5616777A (en) * | 1995-04-19 | 1997-04-01 | Schering Corporation | Chiral hydrazine derivatives |
US5760466A (en) * | 1995-04-20 | 1998-06-02 | Kyocera Corporation | Semiconductor device having improved heat resistance |
RU2135494C1 (ru) * | 1995-12-01 | 1999-08-27 | Санкио Компани Лимитед | Гетероциклические соединения и композиция на их основе, проявляющая антагонистическое действие в отношении рецепторов тахикинина |
HUP0004321A3 (en) | 1997-12-04 | 2002-04-29 | Sankyo Co | Alicyclic acylated heterocyclic derivatives and pharmaceutical compositions containing the same |
KR100616029B1 (ko) | 1998-12-29 | 2006-08-28 | 파마시아 앤드 업존 캄파니 엘엘씨 | 아릴 에테르의 제조 방법 |
FR2796069B3 (fr) * | 1999-07-09 | 2001-08-24 | Sanofi Synthelabo | Nouveaux procedes de preparation de derives de 2-(2- arylmorpholin-2-yl)ethanol substitues, enantiomeriquement purs, et composes intermediaires utiles dans ces procedes |
-
1999
- 1999-07-09 FR FR9909061A patent/FR2796069B3/fr not_active Expired - Lifetime
-
2000
- 2000-07-07 MX MXPA02000307A patent/MXPA02000307A/es active IP Right Grant
- 2000-07-07 EP EP00949673A patent/EP1200417B1/fr not_active Expired - Lifetime
- 2000-07-07 CN CNB00811143XA patent/CN1183121C/zh not_active Expired - Fee Related
- 2000-07-07 CN CNB2004100322961A patent/CN1266115C/zh not_active Expired - Fee Related
- 2000-07-07 AT AT00949673T patent/ATE252566T1/de not_active IP Right Cessation
- 2000-07-07 SI SI200030283T patent/SI1200417T1/xx unknown
- 2000-07-07 CA CA002378002A patent/CA2378002C/en not_active Expired - Fee Related
- 2000-07-07 AU AU62956/00A patent/AU6295600A/en not_active Abandoned
- 2000-07-07 WO PCT/FR2000/001966 patent/WO2001004105A1/fr active IP Right Grant
- 2000-07-07 ES ES00949673T patent/ES2208381T3/es not_active Expired - Lifetime
- 2000-07-07 CZ CZ20020059A patent/CZ300744B6/cs not_active IP Right Cessation
- 2000-07-07 PL PL356064A patent/PL203213B1/pl not_active IP Right Cessation
- 2000-07-07 BR BR0012324-2A patent/BR0012324A/pt active Search and Examination
- 2000-07-07 DE DE60006125T patent/DE60006125T2/de not_active Expired - Lifetime
- 2000-07-07 JP JP2001509715A patent/JP3891840B2/ja not_active Expired - Fee Related
- 2000-07-07 US US10/030,600 patent/US7038044B1/en not_active Expired - Fee Related
- 2000-07-07 HU HU0202383A patent/HUP0202383A3/hu unknown
- 2000-07-07 SK SK18-2002A patent/SK286671B6/sk not_active IP Right Cessation
-
2002
- 2002-01-09 HR HR20020021A patent/HRP20020021B1/xx not_active IP Right Cessation
-
2006
- 2006-03-08 US US11/370,399 patent/US7223860B2/en not_active Expired - Fee Related
-
2007
- 2007-03-29 US US11/693,322 patent/US7378521B2/en not_active Expired - Fee Related
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Legal Events
Date | Code | Title | Description |
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ARAI | Request for the grant of a patent on the basis of the submitted results of a substantive examination of a patent application | ||
A1OB | Publication of a patent application | ||
B1PR | Patent granted | ||
PNAN | Change of the applicant name, address/residence |
Owner name: SANOFI-AVENTIS, FR |
|
ODRP | Renewal fee for the maintenance of a patent |
Payment date: 20100705 Year of fee payment: 11 |
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PBON | Lapse due to non-payment of renewal fee |
Effective date: 20110708 |