HK1049165A1 - 循環β-氨基酸衍生物作為質基金屬蛋白酶及TNF-α的抑制劑 - Google Patents

循環β-氨基酸衍生物作為質基金屬蛋白酶及TNF-α的抑制劑

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Publication number
HK1049165A1
HK1049165A1 HK03101351.8A HK03101351A HK1049165A1 HK 1049165 A1 HK1049165 A1 HK 1049165A1 HK 03101351 A HK03101351 A HK 03101351A HK 1049165 A1 HK1049165 A1 HK 1049165A1
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HK
Hong Kong
Prior art keywords
tnf
inhibitors
alpha
amino acid
acid derivatives
Prior art date
Application number
HK03101351.8A
Other languages
English (en)
Inventor
Duan Jingwu
Ott Gregory
Chen Linhua
Lu Zhonghui
P Maduskuie Thomas Jr
E Voss Matthew
Xue Chu-Biao
Decicco Carl
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Publication of HK1049165A1 publication Critical patent/HK1049165A1/zh

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HK03101351.8A 2000-03-17 2003-02-21 循環β-氨基酸衍生物作為質基金屬蛋白酶及TNF-α的抑制劑 HK1049165A1 (zh)

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US19018200P 2000-03-17 2000-03-17
US23337300P 2000-09-18 2000-09-18
US25553900P 2000-12-14 2000-12-14
PCT/US2001/008334 WO2001070673A2 (en) 2000-03-17 2001-03-15 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a)

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HK1049165A1 true HK1049165A1 (zh) 2003-05-02

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US (2) US6743807B2 (zh)
EP (1) EP1263755A2 (zh)
JP (1) JP2003528072A (zh)
KR (1) KR20030009391A (zh)
CN (1) CN1481377A (zh)
AR (1) AR035710A1 (zh)
AU (1) AU2001250849A1 (zh)
BR (1) BR0109467A (zh)
CA (1) CA2401870A1 (zh)
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US20020016336A1 (en) 2002-02-07
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IL151552A0 (en) 2003-04-10
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US6984648B2 (en) 2006-01-10
CA2401870A1 (en) 2001-09-27
PL360678A1 (en) 2004-09-20
US20040162426A1 (en) 2004-08-19
US6743807B2 (en) 2004-06-01
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EP1263755A2 (en) 2002-12-11
JP2003528072A (ja) 2003-09-24
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