FR2449682A1 - Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens - Google Patents

Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens

Info

Publication number
FR2449682A1
FR2449682A1 FR8004168A FR8004168A FR2449682A1 FR 2449682 A1 FR2449682 A1 FR 2449682A1 FR 8004168 A FR8004168 A FR 8004168A FR 8004168 A FR8004168 A FR 8004168A FR 2449682 A1 FR2449682 A1 FR 2449682A1
Authority
FR
France
Prior art keywords
carboxylic acid
antimicrobial agents
quinoleine
acid derivatives
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8004168A
Other languages
English (en)
Other versions
FR2449682B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Otsuka Pharmaceutical Co Ltd
Original Assignee
Otsuka Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharmaceutical Co Ltd filed Critical Otsuka Pharmaceutical Co Ltd
Publication of FR2449682A1 publication Critical patent/FR2449682A1/fr
Application granted granted Critical
Publication of FR2449682B1 publication Critical patent/FR2449682B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

LA PRESENTE INVENTION EST RELATIVE A DE NOUVEAUX DERIVES D'ACIDE QUINOLEINE-CARBOXYLIQUE. CES DERIVES REPONDENT A LA FORMULE GENERALE (1) CI-APRES: (CF DESSIN DANS BOPI) DANS LAQUELLE: R ET R SONT CHACUN UN GROUPE ALKYLE INFERIEUR; ET R EST UN ATOME D'HALOGENE OU UN GROUPE 1-PIPERAZINYLE, ET LEURS SELS. APPLICATION AUX AGENTS ANTIMICROBIENS.
FR8004168A 1979-02-26 1980-02-26 Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens Granted FR2449682A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP54022162A JPS604820B2 (ja) 1979-02-26 1979-02-26 キノリンカルボン酸誘導体

Publications (2)

Publication Number Publication Date
FR2449682A1 true FR2449682A1 (fr) 1980-09-19
FR2449682B1 FR2449682B1 (fr) 1983-08-26

Family

ID=12075122

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8004168A Granted FR2449682A1 (fr) 1979-02-26 1980-02-26 Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens

Country Status (6)

Country Link
US (1) US4544747A (fr)
JP (1) JPS604820B2 (fr)
BR (1) BR8001094A (fr)
CA (1) CA1141383A (fr)
DE (1) DE3007006C2 (fr)
FR (1) FR2449682A1 (fr)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0118854A1 (fr) * 1983-03-12 1984-09-19 Bayer Ag Agent bactéricide contenant des acides quinolinonecarboxyliques
EP0121727A1 (fr) * 1983-03-12 1984-10-17 Bayer Ag Agent bactéricide basé en acides quinolinonecarboxyliques
EP0230295A2 (fr) * 1986-01-21 1987-07-29 Kyorin Pharmaceutical Co., Ltd. Acide 8-alkoxyquinoléine et ses sels avec une toxicité sélective excellente et un procédé pour leur préparation
EP0237955A2 (fr) * 1986-03-17 1987-09-23 Kyorin Pharmaceutical Co., Ltd. Dérivés de l'acide quinolonecarboxylique et leur préparation

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS604820B2 (ja) * 1979-02-26 1985-02-06 大塚製薬株式会社 キノリンカルボン酸誘導体
DE3248507A1 (de) * 1982-12-29 1984-07-05 Bayer Ag, 5090 Leverkusen Mikrobizide mittel auf chinoloncarbonsaeure basis
US4760057A (en) * 1983-06-23 1988-07-26 Merck & Co., Inc. (Acyloxyalkoxy)carbonyl derivatives as bioreversible prodrug moieties for primary and secondary amine functions in drugs
DE3441788A1 (de) * 1984-11-15 1986-05-15 Bayer Ag, 5090 Leverkusen Alkyl-1-cyclopropyl-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3705621C2 (de) * 1986-02-25 1997-01-09 Otsuka Pharma Co Ltd Heterocyclisch substituierte Chinoloncarbonsäurederivate
US5563138A (en) * 1987-04-16 1996-10-08 Otsuka Pharmaceutical Company, Limited Benzoheterocyclic compounds
US5157189A (en) * 1987-10-19 1992-10-20 Karra Sankaram B Conversion of light hydrocarbons to higher hydrocarbons
US4931446A (en) * 1988-03-23 1990-06-05 Abbott Laboratories Antimicrobial for in-vitro diagnostic kits
DE4301246A1 (de) * 1993-01-19 1994-07-21 Bayer Ag Chinolon- und Naphthyridoncarbonsäurederivate
US6387928B1 (en) * 1997-09-15 2002-05-14 The Procter & Gamble Co. Antimicrobial quinolones, their compositions and uses
EP1015445B1 (fr) 1997-09-15 2009-02-25 The Procter & Gamble Company Quinolones antimicrobiennes, compositions et utilisations de celles-ci
DE10108750A1 (de) * 2001-02-23 2002-09-05 Bayer Ag Verbessertes Verfahren zur Herstellung von Fluorchinoloncarbonsäuren
US7456279B2 (en) * 2006-03-28 2008-11-25 The Procter & Gamble Company Coupling process for preparing quinolone intermediates
SMP200800058B (it) * 2006-03-28 2009-09-07 Procter & Gamble Sali e polimorfi malati di un acido (3s, 5s) -7- [3-ammino-5-metilpiperidinil]-1-ciclopropil-1,4-diidro-8-metossi-4-osso-3-chinolincarbossilico
KR101030202B1 (ko) * 2006-03-28 2011-04-22 워너 칠콧 컴퍼니 엘엘씨 퀴놀론 중간체의 제조를 위한 수소화물 환원 방법

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB830832A (en) * 1957-02-15 1960-03-23 Ici Ltd New quinolones and therapeutic compositions containing them
NL7101049A (fr) * 1970-01-28 1971-07-30
DE2246503A1 (de) * 1972-09-22 1974-04-04 Boehringer Mannheim Gmbh 7,8-dimethylchinolon-3-carbonsaeurederivate
US4017622A (en) * 1972-12-18 1977-04-12 Dainippon Pharmaceutical Co., Ltd. Piperazine derivatives
US4156726A (en) * 1974-12-07 1979-05-29 Fisons Limited 4-Oxo-2-carboxyl quinoline derivatives used as antiallergic compounds
JPS5188973A (ja) * 1975-01-29 1976-08-04 Shinkinakinoronkarubonsanjudotainoseiho
JPS53141286A (en) * 1977-05-16 1978-12-08 Kyorin Seiyaku Kk Novel substituted quinolinecarboxylic acid
US4264604A (en) * 1977-07-01 1981-04-28 Ciba-Geigy Corporation Quinolonecarboxylic acid derivatives as bactericides
JPS5845426B2 (ja) * 1978-09-29 1983-10-08 杏林製薬株式会社 置換キノリンカルボン酸誘導体
JPS604820B2 (ja) * 1979-02-26 1985-02-06 大塚製薬株式会社 キノリンカルボン酸誘導体
JPS56128703A (en) * 1980-03-14 1981-10-08 Otsuka Pharmaceut Co Ltd Antimicrobial agent

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0118854A1 (fr) * 1983-03-12 1984-09-19 Bayer Ag Agent bactéricide contenant des acides quinolinonecarboxyliques
EP0121727A1 (fr) * 1983-03-12 1984-10-17 Bayer Ag Agent bactéricide basé en acides quinolinonecarboxyliques
US4563448A (en) * 1983-03-12 1986-01-07 Bayer Aktiengesellschaft Bactericidal agents
EP0230295A2 (fr) * 1986-01-21 1987-07-29 Kyorin Pharmaceutical Co., Ltd. Acide 8-alkoxyquinoléine et ses sels avec une toxicité sélective excellente et un procédé pour leur préparation
EP0230295B1 (fr) * 1986-01-21 1994-05-25 Kyorin Pharmaceutical Co., Ltd. Acide 8-alkoxyquinoléine et ses sels avec une toxicité sélective excellente et un procédé pour leur préparation
EP0237955A2 (fr) * 1986-03-17 1987-09-23 Kyorin Pharmaceutical Co., Ltd. Dérivés de l'acide quinolonecarboxylique et leur préparation
EP0237955A3 (en) * 1986-03-17 1987-11-25 Kyorin Pharmaceutical Co., Ltd. Quinolonecarboxylic acid derivatives and their preparation

Also Published As

Publication number Publication date
JPS55113765A (en) 1980-09-02
CA1141383A (fr) 1983-02-15
BR8001094A (pt) 1980-10-29
DE3007006C2 (de) 1982-12-09
FR2449682B1 (fr) 1983-08-26
DE3007006A1 (de) 1980-08-28
US4544747A (en) 1985-10-01
JPS604820B2 (ja) 1985-02-06

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