FR2449682A1 - Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens - Google Patents
Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiensInfo
- Publication number
- FR2449682A1 FR2449682A1 FR8004168A FR8004168A FR2449682A1 FR 2449682 A1 FR2449682 A1 FR 2449682A1 FR 8004168 A FR8004168 A FR 8004168A FR 8004168 A FR8004168 A FR 8004168A FR 2449682 A1 FR2449682 A1 FR 2449682A1
- Authority
- FR
- France
- Prior art keywords
- carboxylic acid
- antimicrobial agents
- quinoleine
- acid derivatives
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
- A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Agronomy & Crop Science (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
LA PRESENTE INVENTION EST RELATIVE A DE NOUVEAUX DERIVES D'ACIDE QUINOLEINE-CARBOXYLIQUE. CES DERIVES REPONDENT A LA FORMULE GENERALE (1) CI-APRES: (CF DESSIN DANS BOPI) DANS LAQUELLE: R ET R SONT CHACUN UN GROUPE ALKYLE INFERIEUR; ET R EST UN ATOME D'HALOGENE OU UN GROUPE 1-PIPERAZINYLE, ET LEURS SELS. APPLICATION AUX AGENTS ANTIMICROBIENS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP54022162A JPS604820B2 (ja) | 1979-02-26 | 1979-02-26 | キノリンカルボン酸誘導体 |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2449682A1 true FR2449682A1 (fr) | 1980-09-19 |
FR2449682B1 FR2449682B1 (fr) | 1983-08-26 |
Family
ID=12075122
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8004168A Granted FR2449682A1 (fr) | 1979-02-26 | 1980-02-26 | Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens |
Country Status (6)
Country | Link |
---|---|
US (1) | US4544747A (fr) |
JP (1) | JPS604820B2 (fr) |
BR (1) | BR8001094A (fr) |
CA (1) | CA1141383A (fr) |
DE (1) | DE3007006C2 (fr) |
FR (1) | FR2449682A1 (fr) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0118854A1 (fr) * | 1983-03-12 | 1984-09-19 | Bayer Ag | Agent bactéricide contenant des acides quinolinonecarboxyliques |
EP0121727A1 (fr) * | 1983-03-12 | 1984-10-17 | Bayer Ag | Agent bactéricide basé en acides quinolinonecarboxyliques |
EP0230295A2 (fr) * | 1986-01-21 | 1987-07-29 | Kyorin Pharmaceutical Co., Ltd. | Acide 8-alkoxyquinoléine et ses sels avec une toxicité sélective excellente et un procédé pour leur préparation |
EP0237955A2 (fr) * | 1986-03-17 | 1987-09-23 | Kyorin Pharmaceutical Co., Ltd. | Dérivés de l'acide quinolonecarboxylique et leur préparation |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS604820B2 (ja) * | 1979-02-26 | 1985-02-06 | 大塚製薬株式会社 | キノリンカルボン酸誘導体 |
DE3248507A1 (de) * | 1982-12-29 | 1984-07-05 | Bayer Ag, 5090 Leverkusen | Mikrobizide mittel auf chinoloncarbonsaeure basis |
US4760057A (en) * | 1983-06-23 | 1988-07-26 | Merck & Co., Inc. | (Acyloxyalkoxy)carbonyl derivatives as bioreversible prodrug moieties for primary and secondary amine functions in drugs |
DE3441788A1 (de) * | 1984-11-15 | 1986-05-15 | Bayer Ag, 5090 Leverkusen | Alkyl-1-cyclopropyl-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
DE3705621C2 (de) * | 1986-02-25 | 1997-01-09 | Otsuka Pharma Co Ltd | Heterocyclisch substituierte Chinoloncarbonsäurederivate |
US5563138A (en) * | 1987-04-16 | 1996-10-08 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
US5157189A (en) * | 1987-10-19 | 1992-10-20 | Karra Sankaram B | Conversion of light hydrocarbons to higher hydrocarbons |
US4931446A (en) * | 1988-03-23 | 1990-06-05 | Abbott Laboratories | Antimicrobial for in-vitro diagnostic kits |
DE4301246A1 (de) * | 1993-01-19 | 1994-07-21 | Bayer Ag | Chinolon- und Naphthyridoncarbonsäurederivate |
US6387928B1 (en) * | 1997-09-15 | 2002-05-14 | The Procter & Gamble Co. | Antimicrobial quinolones, their compositions and uses |
EP1015445B1 (fr) | 1997-09-15 | 2009-02-25 | The Procter & Gamble Company | Quinolones antimicrobiennes, compositions et utilisations de celles-ci |
DE10108750A1 (de) * | 2001-02-23 | 2002-09-05 | Bayer Ag | Verbessertes Verfahren zur Herstellung von Fluorchinoloncarbonsäuren |
US7456279B2 (en) * | 2006-03-28 | 2008-11-25 | The Procter & Gamble Company | Coupling process for preparing quinolone intermediates |
SMP200800058B (it) * | 2006-03-28 | 2009-09-07 | Procter & Gamble | Sali e polimorfi malati di un acido (3s, 5s) -7- [3-ammino-5-metilpiperidinil]-1-ciclopropil-1,4-diidro-8-metossi-4-osso-3-chinolincarbossilico |
KR101030202B1 (ko) * | 2006-03-28 | 2011-04-22 | 워너 칠콧 컴퍼니 엘엘씨 | 퀴놀론 중간체의 제조를 위한 수소화물 환원 방법 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB830832A (en) * | 1957-02-15 | 1960-03-23 | Ici Ltd | New quinolones and therapeutic compositions containing them |
NL7101049A (fr) * | 1970-01-28 | 1971-07-30 | ||
DE2246503A1 (de) * | 1972-09-22 | 1974-04-04 | Boehringer Mannheim Gmbh | 7,8-dimethylchinolon-3-carbonsaeurederivate |
US4017622A (en) * | 1972-12-18 | 1977-04-12 | Dainippon Pharmaceutical Co., Ltd. | Piperazine derivatives |
US4156726A (en) * | 1974-12-07 | 1979-05-29 | Fisons Limited | 4-Oxo-2-carboxyl quinoline derivatives used as antiallergic compounds |
JPS5188973A (ja) * | 1975-01-29 | 1976-08-04 | Shinkinakinoronkarubonsanjudotainoseiho | |
JPS53141286A (en) * | 1977-05-16 | 1978-12-08 | Kyorin Seiyaku Kk | Novel substituted quinolinecarboxylic acid |
US4264604A (en) * | 1977-07-01 | 1981-04-28 | Ciba-Geigy Corporation | Quinolonecarboxylic acid derivatives as bactericides |
JPS5845426B2 (ja) * | 1978-09-29 | 1983-10-08 | 杏林製薬株式会社 | 置換キノリンカルボン酸誘導体 |
JPS604820B2 (ja) * | 1979-02-26 | 1985-02-06 | 大塚製薬株式会社 | キノリンカルボン酸誘導体 |
JPS56128703A (en) * | 1980-03-14 | 1981-10-08 | Otsuka Pharmaceut Co Ltd | Antimicrobial agent |
-
1979
- 1979-02-26 JP JP54022162A patent/JPS604820B2/ja not_active Expired
-
1980
- 1980-02-25 BR BR8001094A patent/BR8001094A/pt unknown
- 1980-02-25 DE DE3007006A patent/DE3007006C2/de not_active Expired
- 1980-02-25 CA CA000346373A patent/CA1141383A/fr not_active Expired
- 1980-02-26 FR FR8004168A patent/FR2449682A1/fr active Granted
-
1984
- 1984-04-27 US US06/604,574 patent/US4544747A/en not_active Expired - Fee Related
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0118854A1 (fr) * | 1983-03-12 | 1984-09-19 | Bayer Ag | Agent bactéricide contenant des acides quinolinonecarboxyliques |
EP0121727A1 (fr) * | 1983-03-12 | 1984-10-17 | Bayer Ag | Agent bactéricide basé en acides quinolinonecarboxyliques |
US4563448A (en) * | 1983-03-12 | 1986-01-07 | Bayer Aktiengesellschaft | Bactericidal agents |
EP0230295A2 (fr) * | 1986-01-21 | 1987-07-29 | Kyorin Pharmaceutical Co., Ltd. | Acide 8-alkoxyquinoléine et ses sels avec une toxicité sélective excellente et un procédé pour leur préparation |
EP0230295B1 (fr) * | 1986-01-21 | 1994-05-25 | Kyorin Pharmaceutical Co., Ltd. | Acide 8-alkoxyquinoléine et ses sels avec une toxicité sélective excellente et un procédé pour leur préparation |
EP0237955A2 (fr) * | 1986-03-17 | 1987-09-23 | Kyorin Pharmaceutical Co., Ltd. | Dérivés de l'acide quinolonecarboxylique et leur préparation |
EP0237955A3 (en) * | 1986-03-17 | 1987-11-25 | Kyorin Pharmaceutical Co., Ltd. | Quinolonecarboxylic acid derivatives and their preparation |
Also Published As
Publication number | Publication date |
---|---|
JPS55113765A (en) | 1980-09-02 |
CA1141383A (fr) | 1983-02-15 |
BR8001094A (pt) | 1980-10-29 |
DE3007006C2 (de) | 1982-12-09 |
FR2449682B1 (fr) | 1983-08-26 |
DE3007006A1 (de) | 1980-08-28 |
US4544747A (en) | 1985-10-01 |
JPS604820B2 (ja) | 1985-02-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |