FI841679A - 17-(isocyano-sulfonylmetylen)- steroider, 17-(formamido-sulfonylmetylen)- steroider och deras framstaellning. - Google Patents

17-(isocyano-sulfonylmetylen)- steroider, 17-(formamido-sulfonylmetylen)- steroider och deras framstaellning. Download PDF

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Publication number
FI841679A
FI841679A FI841679A FI841679A FI841679A FI 841679 A FI841679 A FI 841679A FI 841679 A FI841679 A FI 841679A FI 841679 A FI841679 A FI 841679A FI 841679 A FI841679 A FI 841679A
Authority
FI
Finland
Prior art keywords
sulphonylmethylene
steroider
formamido
isocyano
deras framstaellning
Prior art date
Application number
FI841679A
Other languages
English (en)
Other versions
FI841679A0 (fi
FI82061B (fi
FI82061C (fi
Inventor
Leusen Albert Mattheus Van
Leusen Adriaan Marinus Van
Original Assignee
Gist Brocades Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades Nv filed Critical Gist Brocades Nv
Publication of FI841679A0 publication Critical patent/FI841679A0/fi
Publication of FI841679A publication Critical patent/FI841679A/fi
Publication of FI82061B publication Critical patent/FI82061B/fi
Application granted granted Critical
Publication of FI82061C publication Critical patent/FI82061C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/005—3 membered carbocyclic rings in position 12
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI841679A 1983-04-29 1984-04-27 17-(isocyano-sulfonylmetylen)- steroider och foerfarande foer deras framstaellning samt 17-(formamido- ylen)taellning. FI82061C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP83200616 1983-04-29
EP83200616A EP0123734A1 (en) 1983-04-29 1983-04-29 17-(Isocyano-sulfonylmethylene)-steroids, 17-(formamido-sulfonylmethylene)-steroids and their preparation

Publications (4)

Publication Number Publication Date
FI841679A0 FI841679A0 (fi) 1984-04-27
FI841679A true FI841679A (fi) 1984-10-30
FI82061B FI82061B (fi) 1990-09-28
FI82061C FI82061C (fi) 1991-01-10

Family

ID=8190949

Family Applications (1)

Application Number Title Priority Date Filing Date
FI841679A FI82061C (fi) 1983-04-29 1984-04-27 17-(isocyano-sulfonylmetylen)- steroider och foerfarande foer deras framstaellning samt 17-(formamido- ylen)taellning.

Country Status (17)

Country Link
US (1) US4647410A (fi)
EP (2) EP0123734A1 (fi)
JP (2) JPS59206399A (fi)
KR (1) KR860001469B1 (fi)
AU (1) AU568643B2 (fi)
CA (1) CA1257249A (fi)
DE (1) DE3461381D1 (fi)
DK (2) DK166545B1 (fi)
ES (2) ES8608537A1 (fi)
FI (1) FI82061C (fi)
GR (1) GR81997B (fi)
HU (2) HU193207B (fi)
IE (1) IE57328B1 (fi)
IL (1) IL71658A (fi)
NO (1) NO167093C (fi)
NZ (1) NZ207985A (fi)
PT (1) PT78503B (fi)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0123735A1 (en) * 1983-04-29 1984-11-07 Gist-Brocades N.V. New process for the preparation of 20-keto-delta-16-steroids and new intermediate compounds formed in this process
WO1989009781A1 (en) * 1988-04-08 1989-10-19 Gist-Brocades N.V. 9-alpha-hydroxy-17-methylene steroids, their preparation and utilization
HU226413B1 (en) * 1991-06-25 2008-11-28 Aventis Pharma Sa Novel 16-(nitro-substituted methyl)pregna-1,4-dien-3,20-dion derivatives and process for producing them
FR2681069B1 (fr) * 1991-09-06 1995-04-28 Roussel Uclaf Nouveau procede de preparation de l'hydrocortisone et nouveaux intermediaires.
ATE365171T1 (de) * 1995-12-11 2007-07-15 Searle Llc Verfahren zur herstellung einer epoxyverbindung
US6887991B1 (en) 1996-12-11 2005-05-03 G. D. Searle & Company Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein
NZ336004A (en) 1996-12-11 2001-04-27 G Process for preparation of 3-keto-7-alpha-alkoxycarbonyl substituted delta-4,5-steroid by reacting 4,5-dihydro-5,7-lactone steroid substrate in the presence of a base
AU4093799A (en) 1998-05-22 1999-12-13 Board Of Trustees Of The Leland Stanford Junior University Bifunctional molecules and therapies based thereon
EP2287721A3 (en) 1999-11-02 2011-04-06 Canon Kabushiki Kaisha Print control method and apparatus
US7235655B2 (en) 2002-03-22 2007-06-26 Pharmacia & Upjohn Company Processes to prepare eplerenone
PT1889198E (pt) 2005-04-28 2015-03-06 Proteus Digital Health Inc Sistema fármaco-informático
JP2009508494A (ja) 2005-09-16 2009-03-05 ラプトール ファーマシューティカル インコーポレイテッド Ｃｒを含むタンパク質に対して特異的な受容体−結合タンパク質（ｒａｐ）変異体を含む組成物およびその使用
PT2398500T (pt) 2009-02-20 2019-06-14 2 Bbb Medicines B V Sistema de entrega de medicamentos à base de glutationas
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
CN105481924B (zh) * 2015-11-24 2017-08-15 浙江省诸暨合力化学对外贸易有限公司 一种***的制备方法
EP4392036A1 (en) * 2021-08-26 2024-07-03 Brandeis University Selective isonitrile inhibitors of cytochrome p450 subtypes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7807631A (nl) * 1978-07-17 1980-01-21 Gist Brocades Nv Isocyanoderivaten en hun bereiding.
FR2462445A1 (fr) * 1979-07-31 1981-02-13 Roussel Uclaf Nouveaux derives 17-/(hydroxymethyl) (formamido) methylene/steroides, leur procede de preparation et leur application a l'introduction de la chaine laterale hydroxyacetyle
FR2486947A1 (fr) * 1980-07-15 1982-01-22 Roussel Uclaf Nouveaux derives steroides 20-isonitriles 17(20) insatures, leur procede de preparation et leur application a la preparation des steroides 17a-hydroxy 20-ceto

Also Published As

Publication number Publication date
PT78503B (en) 1986-05-20
EP0123734A1 (en) 1984-11-07
AU2713384A (en) 1984-11-01
ES553609A0 (es) 1987-11-01
DK166545B1 (da) 1993-06-07
JPH0559097A (ja) 1993-03-09
DK22192D0 (da) 1992-02-21
NO167093C (no) 1991-10-02
DK22192A (da) 1992-02-21
KR840008461A (ko) 1984-12-15
NZ207985A (en) 1986-11-12
JPS59206399A (ja) 1984-11-22
ES8800263A1 (es) 1987-11-01
HU193207B (en) 1987-08-28
JPH053478B2 (fi) 1993-01-14
IL71658A (en) 1988-03-31
DK166831B1 (da) 1993-07-19
JPH0717673B2 (ja) 1995-03-01
IL71658A0 (en) 1984-07-31
EP0124934A1 (en) 1984-11-14
IE841038L (en) 1984-10-29
NO841700L (no) 1984-10-30
CA1257249A (en) 1989-07-11
DE3461381D1 (en) 1987-01-08
HUT34220A (en) 1985-02-28
ES8608537A1 (es) 1986-07-16
ES532029A0 (es) 1986-07-16
FI841679A0 (fi) 1984-04-27
HU194277B (en) 1988-01-28
FI82061B (fi) 1990-09-28
DK212184D0 (da) 1984-04-27
FI82061C (fi) 1991-01-10
DK212184A (da) 1984-10-30
GR81997B (fi) 1984-12-12
US4647410A (en) 1987-03-03
EP0124934B1 (en) 1986-11-20
KR860001469B1 (ko) 1986-09-26
AU568643B2 (en) 1988-01-07
IE57328B1 (en) 1992-07-29
NO167093B (no) 1991-06-24
PT78503A (en) 1984-05-01

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PC Transfer of assignment of patent

Owner name: ROUSSEL-UCLAF

MM Patent lapsed

Owner name: ROUSSEL UCLAF SOCIETE ANONYME