ES8401447A1 - Un procedimiento para preparar un tripeptido. - Google Patents

Un procedimiento para preparar un tripeptido.

Info

Publication number
ES8401447A1
ES8401447A1 ES517144A ES517144A ES8401447A1 ES 8401447 A1 ES8401447 A1 ES 8401447A1 ES 517144 A ES517144 A ES 517144A ES 517144 A ES517144 A ES 517144A ES 8401447 A1 ES8401447 A1 ES 8401447A1
Authority
ES
Spain
Prior art keywords
prolyl
prepared
carboxyalkylproline
containing tripeptides
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES517144A
Other languages
English (en)
Other versions
ES517144A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of ES517144A0 publication Critical patent/ES517144A0/es
Publication of ES8401447A1 publication Critical patent/ES8401447A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0823—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Cardiology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

UN PROCEDIMIENTO PARA PREPARAR UN TRIPEPTIDO.SE HACE REACCIONAR EL COMPUESTO (II) CON EL (III) DONDE R1 ES UN CARBOXI, SULFO O FOSFONO PROTEGIDO; R2 ES UN GRUPO PROTECTOR DE CARBOXI Y R3 ES EL GRUPO AMINO O N-METIL-AMINO; A CONTINUACION SE SEPARA ALGUNO DE LOS GRUPOS PROTECTORES PRESENTES Y OPCIONALMENTE SE FORMA LA SAL FARMACEUTICAMENTE ACEPTABLE. LA REACCION SE LLEVA A CABO EN PRESENCIA DE UNA CARBODIIMIDA, TAL COMO LA DICICLO-HEXILCARBODIIMID A. SE OBTIENE EL COMPUESTO (I) EN EL CUAL R ES CARBOXI, SULFO O FOSFONO.
ES517144A 1981-11-06 1982-11-05 Un procedimiento para preparar un tripeptido. Expired ES8401447A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US31872181A 1981-11-06 1981-11-06

Publications (2)

Publication Number Publication Date
ES517144A0 ES517144A0 (es) 1983-12-16
ES8401447A1 true ES8401447A1 (es) 1983-12-16

Family

ID=23239338

Family Applications (1)

Application Number Title Priority Date Filing Date
ES517144A Expired ES8401447A1 (es) 1981-11-06 1982-11-05 Un procedimiento para preparar un tripeptido.

Country Status (25)

Country Link
EP (1) EP0080283B1 (es)
JP (1) JPS5890537A (es)
KR (1) KR880002594B1 (es)
AT (1) ATE17736T1 (es)
AU (1) AU562011B2 (es)
CA (1) CA1247085A (es)
CS (1) CS235030B2 (es)
DD (1) DD206553A5 (es)
DE (1) DE3268884D1 (es)
DK (1) DK480682A (es)
ES (1) ES8401447A1 (es)
FI (1) FI75175C (es)
GR (1) GR77368B (es)
HU (1) HU187808B (es)
IE (1) IE53982B1 (es)
IL (1) IL67070A (es)
NO (1) NO160081C (es)
NZ (1) NZ202232A (es)
PH (1) PH18708A (es)
PL (1) PL136098B1 (es)
PT (1) PT75769B (es)
RO (1) RO84706B (es)
YU (1) YU245582A (es)
ZA (1) ZA827816B (es)
ZW (1) ZW23282A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE174343T1 (de) * 1991-02-27 1998-12-15 Lacer Sa Antihypertensive n-(alpha-substituiertes pyridyl)-carbonyldipeptide
JP3068200B2 (ja) 1995-06-06 2000-07-24 ファイザー・インコーポレーテッド グリコーゲンホスホリラーゼ阻害剤としての置換ｎ−（インドール−２−カルボニル−）アミドおよび誘導体
MY114711A (en) 1995-06-06 2002-12-31 Pfizer Substituted n-(indole-2-carbonyl)-b-alanmamides and derivatives as antidiabetic agents
CA2224062C (en) * 1995-06-06 2001-09-04 Pfizer Limited Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors
US6277877B1 (en) 2000-08-15 2001-08-21 Pfizer, Inc. Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors
KR20040013679A (ko) * 2002-08-08 2004-02-14 현대산업개발 주식회사 실내 공기 상태 표시장치

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2480747A1 (fr) * 1980-04-17 1981-10-23 Roques Bernard Derives d'acides amines et leur application therapeutique

Also Published As

Publication number Publication date
KR880002594B1 (ko) 1988-12-03
IL67070A0 (en) 1983-02-23
PL136098B1 (en) 1986-01-31
NO160081C (no) 1989-03-08
FI823798A0 (fi) 1982-11-05
PT75769A (en) 1982-11-01
EP0080283A1 (en) 1983-06-01
ATE17736T1 (de) 1986-02-15
NO160081B (no) 1988-11-28
JPS5890537A (ja) 1983-05-30
CS235030B2 (en) 1985-04-16
KR840002372A (ko) 1984-06-25
NO823693L (no) 1983-05-09
RO84706A (ro) 1984-07-17
PT75769B (en) 1985-07-26
NZ202232A (en) 1985-08-16
AU9017382A (en) 1983-05-12
CA1247085A (en) 1988-12-20
GR77368B (es) 1984-09-11
DE3268884D1 (en) 1986-03-13
IE822647L (en) 1983-05-06
PH18708A (en) 1985-09-05
IL67070A (en) 1986-01-31
ZW23282A1 (en) 1983-02-23
DK480682A (da) 1983-05-07
IE53982B1 (en) 1989-05-10
ZA827816B (en) 1983-08-31
RO84706B (ro) 1984-09-30
FI75175B (fi) 1988-01-29
AU562011B2 (en) 1987-05-28
ES517144A0 (es) 1983-12-16
HU187808B (en) 1986-02-28
EP0080283B1 (en) 1986-01-29
DD206553A5 (de) 1984-02-01
FI823798L (fi) 1983-05-07
YU245582A (en) 1985-03-20
FI75175C (fi) 1988-05-09
PL238893A1 (en) 1983-07-04

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