ES2006478A6 - Procedimiento de preparacion de esteres retinoicos de antibioticos. - Google Patents

Procedimiento de preparacion de esteres retinoicos de antibioticos.

Info

Publication number: ES2006478A6
Authority: ES; Spain
Prior art keywords: retinoic acid; antibiotics; acid esters; new retinoic; new
Prior art date: 1986-05-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES8701603A

Other languages

English (en)

Spanish (es)

Inventor

Michel Philippe

Henri Sebag

Didier Dupuis

Andre Rougier

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

LOreal SA

Original Assignee

LOreal SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-05-06

Filing date

1987-05-05

Publication date

1989-05-01

1987-05-05 Application filed by LOreal SA filed Critical LOreal SA

1989-05-01 Publication of ES2006478A6 publication Critical patent/ES2006478A6/es

Status Expired legal-status Critical Current

Links

SHGAZHPCJJPHSC-YCNIQYBTSA-N retinoic acid group Chemical class C\C(=C/C(=O)O)\C=C\C=C(\C=C\C1=C(CCCC1(C)C)C)/C SHGAZHPCJJPHSC-YCNIQYBTSA-N 0.000 title abstract 2
239000003242 anti bacterial agent Substances 0.000 title 1
229940088710 antibiotic agent Drugs 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 3
-1 13-cis-retinoic acid ester Chemical class 0.000 abstract 1
208000002874 Acne Vulgaris Diseases 0.000 abstract 1
201000004624 Dermatitis Diseases 0.000 abstract 1
ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical compound O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 abstract 1
229930006677 Erythromycin A Natural products 0.000 abstract 1
OJMMVQQUTAEWLP-UHFFFAOYSA-N Lincomycin Natural products CN1CC(CCC)CC1C(=O)NC(C(C)O)C1C(O)C(O)C(O)C(SC)O1 OJMMVQQUTAEWLP-UHFFFAOYSA-N 0.000 abstract 1
206010000496 acne Diseases 0.000 abstract 1
229960002227 clindamycin Drugs 0.000 abstract 1
KDLRVYVGXIQJDK-AWPVFWJPSA-N clindamycin Chemical compound CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@H](C)Cl)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 KDLRVYVGXIQJDK-AWPVFWJPSA-N 0.000 abstract 1
229960003276 erythromycin Drugs 0.000 abstract 1
229960005280 isotretinoin Drugs 0.000 abstract 1
OJMMVQQUTAEWLP-KIDUDLJLSA-N lincomycin Chemical compound CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@@H](C)O)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 OJMMVQQUTAEWLP-KIDUDLJLSA-N 0.000 abstract 1
229960005287 lincomycin Drugs 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/67—Vitamins
- A61K8/671—Vitamin A; Derivatives thereof, e.g. ester of vitamin A acid, ester of retinol, retinol, retinal
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
- C07H15/16—Lincomycin; Derivatives thereof

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Dermatology (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Communicable Diseases (AREA)
Epidemiology (AREA)
Birds (AREA)
Oncology (AREA)
Crystallography & Structural Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Cosmetics (AREA)

ES8701603A 1986-05-06 1987-05-05 Procedimiento de preparacion de esteres retinoicos de antibioticos. Expired ES2006478A6 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8606528A FR2598420B1 (fr)	1986-05-06	1986-05-06	Nouveaux esters retinoiques d'antibiotiques, leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant

Publications (1)

Publication Number	Publication Date
ES2006478A6 true ES2006478A6 (es)	1989-05-01

Family

ID=9334966

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ES8701603A Expired ES2006478A6 (es)	1986-05-06	1987-05-05	Procedimiento de preparacion de esteres retinoicos de antibioticos.

Country Status (13)

Country	Link
JP (1)	JP2504990B2 (fr)
BE (1)	BE1004152A4 (fr)
CA (1)	CA1300131C (fr)
CH (1)	CH674847A5 (fr)
DE (1)	DE3714937C2 (fr)
DK (1)	DK169345B1 (fr)
ES (1)	ES2006478A6 (fr)
FR (1)	FR2598420B1 (fr)
GB (1)	GB2191483B (fr)
IT (1)	IT1204556B (fr)
NL (1)	NL193946C (fr)
NO (1)	NO168041C (fr)
SE (1)	SE470379B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
LU87041A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters retinoiques de macrolides,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87039A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters biaromatiques d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87038A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters aromatiques d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87036A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters cycloaliphatiques insatures d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87037A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters polyaromatiques d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87040A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters aromatiques polycycliques d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87035A1 (fr) *	1987-11-04	1989-06-14	Oreal	Esters du type etretinique ou apparente d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
LU87070A1 (fr) *	1987-12-10	1989-07-07	Oreal	Association de derives de pyrimidine et d'agents pour induire et stimuler la croissance des cheveux et diminuer leur chute
FR2644460A1 (fr) *	1989-03-16	1990-09-21	Oreal	Esters retinoiques de d-desosamine, leur procede de preparation et leur utilisation en medecine humaine ou veterinaire et en cosmetique
GB2282596B (en) *	1993-10-06	1998-04-15	Ciba Geigy Ag	Water-soluble retinoids
FR2931662B1 (fr) *	2008-05-30	2010-07-30	Galderma Res & Dev	Nouvelles compositions depigmentantes sous forme d'une composition anhydre sans vaseline et sans elastomere comprenant un derive phenolique solubilise.
FR2931661B1 (fr) *	2008-05-30	2010-07-30	Galderma Res & Dev	Nouvelles compositions depigmentantes sous forme d'une composition anhydre sans vaseline et sans elastomere comprenant un derive phenolique solubilise et un retinoide.
AU2012272804B2 (en)	2011-06-22	2017-07-06	Vyome Therapeutics Limited	Conjugate-based antifungal and antibacterial prodrugs

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2862921A (en) *	1953-08-13	1958-12-02	Upjohn Co	Erythromycin esters
US3598806A (en) *	1969-04-15	1971-08-10	Upjohn Co	Process for preparing lincomycin-3-monoacylates
FR2378523A1 (fr) *	1977-01-26	1978-08-25	Grupper Charles	Medicament pour le traitement de l'acne
FR2582000B1 (fr) *	1985-05-14	1987-06-26	Oreal	Esters gras bi ou tri-eniques d'erythromycine a, leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant

1986
- 1986-05-06 FR FR8606528A patent/FR2598420B1/fr not_active Expired - Lifetime
1987
- 1987-05-02 JP JP62107980A patent/JP2504990B2/ja not_active Expired - Lifetime
- 1987-05-04 NL NL8701054A patent/NL193946C/nl not_active IP Right Cessation
- 1987-05-05 NO NO871870A patent/NO168041C/no unknown
- 1987-05-05 DK DK229387A patent/DK169345B1/da not_active IP Right Cessation
- 1987-05-05 CA CA000536348A patent/CA1300131C/fr not_active Expired - Lifetime
- 1987-05-05 SE SE8701845A patent/SE470379B/sv not_active IP Right Cessation
- 1987-05-05 CH CH1705/87A patent/CH674847A5/fr not_active IP Right Cessation
- 1987-05-05 DE DE3714937A patent/DE3714937C2/de not_active Expired - Lifetime
- 1987-05-05 IT IT20389/87A patent/IT1204556B/it active
- 1987-05-05 ES ES8701603A patent/ES2006478A6/es not_active Expired
- 1987-05-06 GB GB8710673A patent/GB2191483B/en not_active Expired - Lifetime
- 1987-05-06 BE BE8700486A patent/BE1004152A4/fr not_active IP Right Cessation

Also Published As

Publication number	Publication date
CH674847A5 (fr)	1990-07-31
SE8701845D0 (sv)	1987-05-05
SE470379B (sv)	1994-02-07
NL193946C (nl)	2001-03-02
DE3714937A1 (de)	1987-11-12
BE1004152A4 (fr)	1992-10-06
GB8710673D0 (en)	1987-06-10
GB2191483B (en)	1990-05-30
DE3714937C2 (de)	1998-02-26
DK229387D0 (da)	1987-05-05
NL193946B (nl)	2000-11-01
IT8720389A0 (it)	1987-05-05
CA1300131C (fr)	1992-05-05
DK229387A (da)	1987-11-07
NO168041B (no)	1991-09-30
FR2598420A1 (fr)	1987-11-13
NL8701054A (nl)	1987-12-01
JPS62289593A (ja)	1987-12-16
NO168041C (no)	1992-01-08
DK169345B1 (da)	1994-10-10
GB2191483A (en)	1987-12-16
IT1204556B (it)	1989-03-10
JP2504990B2 (ja)	1996-06-05
SE8701845L (sv)	1987-11-07
NO871870L (no)	1987-11-09
FR2598420B1 (fr)	1991-06-07
NO871870D0 (no)	1987-05-05

Legal Events

Date	Code	Title	Description
2008-06-16	FD1A	Patent lapsed	Effective date: 20070507

Publication	Publication Date	Title
ES2006478A6 (es)	1989-05-01	Procedimiento de preparacion de esteres retinoicos de antibioticos.
EP0326151A3 (fr)	1991-03-13	Formulations perfectionnées à libération contrôlée
MY103234A (en)	1993-05-29	Bleaching composition
AU598204B2 (en)	1990-06-21	Chemical derivatives of antibiotics S541
AU7611791A (en)	1991-10-03	Malonic acid derivative compounds
GR3005156T3 (fr)	1993-05-24
AU6999794A (en)	1995-01-03	Process for the preparation of n-acetylneuraminic acid
AU2830889A (en)	1990-08-09	Process for the production of an aromatic polycarboxylic acid
ES2029832T3 (es)	1992-10-01	Procedimiento para la produccion de compuestos de macrolida.
WO1995025091A3 (fr)	1995-10-12	Derives d'acide nipecotique utilises en tant que composes antithrombotiques
IE851204L (en)	1985-11-15	Beta-carbolines
UA8357A1 (uk)	1996-03-29	Спосіб оптичного поділу піранобензоксадіазольної сполуки
IE830664L (en)	1983-09-26	Treating acne
HUT59654A (en)	1992-06-29	Fungicide and insecticide composition containing substituted acrylic ester derivatives, and process for producing the active components and theyr intermediates
WO1988003922A3 (fr)	1988-06-30	Herbicides a base de thiophenesulfonamide
AU8162394A (en)	1995-06-29	Process for the preparation of 2,4,5-tribromopyrrole-3-carbonitrile
GR3022731T3 (en)	1997-06-30	Antibiotic a 40926 ester derivatives
IE862533L (en)	1987-03-26	Bicyclic catechol derivatives
ES2130392T3 (es)	1999-07-01	Procedimiento para la preparacion de acido clavulanico.
AU2891084A (en)	1984-12-06	Esters of 2-bromo-4-methylimidazole-5-carboxylic acid
AU542522B2 (en)	1985-02-21	Alpha-substituted ureidobenzylpenicillanic acid and process for producing the same
GB9305853D0 (en)	1993-05-05	Chemical compounds
IN170286B (fr)	1992-03-07
EP0307177A3 (fr)	1989-10-25	Dérivés d'érythromycine
EP0082656A3 (fr)	1984-09-12	Préparation de dérivés céphame