EA200601552A1 - Замещенные конденсированные гетероциклические с-гликозиды - Google Patents
Замещенные конденсированные гетероциклические с-гликозидыInfo
- Publication number
- EA200601552A1 EA200601552A1 EA200601552A EA200601552A EA200601552A1 EA 200601552 A1 EA200601552 A1 EA 200601552A1 EA 200601552 A EA200601552 A EA 200601552A EA 200601552 A EA200601552 A EA 200601552A EA 200601552 A1 EA200601552 A1 EA 200601552A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- glycosides
- condensed heterocyclic
- substituted condensed
- substituted
- diabetes
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
- C07H7/06—Heterocyclic radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biochemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
В заявке описаны замещенные конденсированные гетероциклические С-гликозиды, композиции, содержащие их, и способы их применения, например, для лечения или профилактики диабета или синдрома X.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49152303P | 2003-08-01 | 2003-08-01 | |
US49153403P | 2003-08-01 | 2003-08-01 | |
US51921003P | 2003-11-12 | 2003-11-12 | |
US57973004P | 2004-06-15 | 2004-06-15 | |
PCT/US2004/024625 WO2005012318A2 (en) | 2003-08-01 | 2004-07-30 | Substituted fused heterocyclic c-glycosides |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200601552A1 true EA200601552A1 (ru) | 2007-02-27 |
EA009768B1 EA009768B1 (ru) | 2008-04-28 |
Family
ID=34120044
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200601552A EA009768B1 (ru) | 2003-08-01 | 2004-07-30 | Замещенные конденсированные гетероциклические с-гликозиды |
Country Status (9)
Country | Link |
---|---|
US (4) | US7094763B2 (ru) |
EP (1) | EP1679965A4 (ru) |
AR (1) | AR048376A1 (ru) |
AU (1) | AU2004261660A1 (ru) |
CA (1) | CA2549015A1 (ru) |
EA (1) | EA009768B1 (ru) |
IL (1) | IL175489A0 (ru) |
TW (1) | TW200521131A (ru) |
WO (1) | WO2005012318A2 (ru) |
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CN100376592C (zh) | 2001-06-20 | 2008-03-26 | 橘生药品工业株式会社 | 含氮的杂环衍生物、含有该衍生物的药物组合物、其药物应用以及用于该衍生物制备的中间体 |
WO2003011880A1 (fr) | 2001-07-31 | 2003-02-13 | Kissei Pharmaceutical Co., Ltd. | Derive de glucopyranosyloxybenzylbenzene, composition medicinale contenant ce derive, usage medicinal de cette composition et produit intermediaire pour produire cette composition |
US20030087843A1 (en) | 2001-09-05 | 2003-05-08 | Washburn William N. | O-pyrazole glucoside SGLT2 inhibitors and method of use |
US6617313B1 (en) | 2002-03-13 | 2003-09-09 | Council Of Scientific And Industrial Research | Glucopyranoside and process of isolation thereof from pterocarpus marsupium pharmaceutical composition containing the same and use thereof |
US6562791B1 (en) * | 2002-03-29 | 2003-05-13 | Council Of Scientific And Industrial Research | Glucopyranoside, process for isolation thereof, pharmaceutical composition containing same and use thereof |
AU2002246317A1 (en) | 2002-04-08 | 2003-10-27 | Council Of Scientific And Industrial Research | Novel glucopyranoside, process for isolation thereof, pharmaceutical composition containing same and use thereof |
PL1980560T3 (pl) | 2003-03-14 | 2011-11-30 | Astellas Pharma Inc | Pochodne C-glikozydowe do leczenia cukrzycy |
JP2004300102A (ja) | 2003-03-31 | 2004-10-28 | Kissei Pharmaceut Co Ltd | 縮合複素環誘導体、それを含有する医薬組成物およびその医薬用途 |
EP1679965A4 (en) * | 2003-08-01 | 2009-05-27 | Janssen Pharmaceutica Nv | SUBSTITUTED FUSED HETEROCYCLIC C-GLYCOSIDES |
-
2004
- 2004-07-30 EP EP04779628A patent/EP1679965A4/en not_active Withdrawn
- 2004-07-30 US US10/903,136 patent/US7094763B2/en not_active Expired - Lifetime
- 2004-07-30 EA EA200601552A patent/EA009768B1/ru not_active IP Right Cessation
- 2004-07-30 AU AU2004261660A patent/AU2004261660A1/en not_active Abandoned
- 2004-07-30 AR ARP040102728A patent/AR048376A1/es not_active Application Discontinuation
- 2004-07-30 TW TW093122974A patent/TW200521131A/zh unknown
- 2004-07-30 WO PCT/US2004/024625 patent/WO2005012318A2/en active Application Filing
- 2004-07-30 CA CA002549015A patent/CA2549015A1/en not_active Abandoned
-
2006
- 2006-05-08 IL IL175489A patent/IL175489A0/en unknown
- 2006-06-15 US US11/453,728 patent/US7482330B2/en active Active
-
2008
- 2008-12-18 US US12/337,918 patent/US20090105162A1/en not_active Abandoned
-
2009
- 2009-09-11 US US12/557,728 patent/US7816328B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US7094763B2 (en) | 2006-08-22 |
WO2005012318A3 (en) | 2005-12-15 |
AU2004261660A1 (en) | 2005-02-10 |
US7816328B2 (en) | 2010-10-19 |
CA2549015A1 (en) | 2005-02-10 |
EA009768B1 (ru) | 2008-04-28 |
US20090105162A1 (en) | 2009-04-23 |
EP1679965A4 (en) | 2009-05-27 |
EP1679965A2 (en) | 2006-07-19 |
WO2005012318A2 (en) | 2005-02-10 |
TW200521131A (en) | 2005-07-01 |
US7482330B2 (en) | 2009-01-27 |
AR048376A1 (es) | 2006-04-26 |
US20050037980A1 (en) | 2005-02-17 |
US20060229260A1 (en) | 2006-10-12 |
IL175489A0 (en) | 2009-02-11 |
US20100004160A1 (en) | 2010-01-07 |
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MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |