EA200601552A1 - Замещенные конденсированные гетероциклические с-гликозиды - Google Patents

Замещенные конденсированные гетероциклические с-гликозиды

Info

Publication number
EA200601552A1
EA200601552A1 EA200601552A EA200601552A EA200601552A1 EA 200601552 A1 EA200601552 A1 EA 200601552A1 EA 200601552 A EA200601552 A EA 200601552A EA 200601552 A EA200601552 A EA 200601552A EA 200601552 A1 EA200601552 A1 EA 200601552A1
Authority
EA
Eurasian Patent Office
Prior art keywords
glycosides
condensed heterocyclic
substituted condensed
substituted
diabetes
Prior art date
Application number
EA200601552A
Other languages
English (en)
Other versions
EA009768B1 (ru
Inventor
Филип Рибжински
Мод Урбански
Сяоянь Чжан
Original Assignee
Янссен Фармацевтика Н. В.
Танабе Сейяку Ко., Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Н. В., Танабе Сейяку Ко., Лтд. filed Critical Янссен Фармацевтика Н. В.
Publication of EA200601552A1 publication Critical patent/EA200601552A1/ru
Publication of EA009768B1 publication Critical patent/EA009768B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/06—Heterocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

В заявке описаны замещенные конденсированные гетероциклические С-гликозиды, композиции, содержащие их, и способы их применения, например, для лечения или профилактики диабета или синдрома X.
EA200601552A 2003-08-01 2004-07-30 Замещенные конденсированные гетероциклические с-гликозиды EA009768B1 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US49152303P 2003-08-01 2003-08-01
US49153403P 2003-08-01 2003-08-01
US51921003P 2003-11-12 2003-11-12
US57973004P 2004-06-15 2004-06-15
PCT/US2004/024625 WO2005012318A2 (en) 2003-08-01 2004-07-30 Substituted fused heterocyclic c-glycosides

Publications (2)

Publication Number Publication Date
EA200601552A1 true EA200601552A1 (ru) 2007-02-27
EA009768B1 EA009768B1 (ru) 2008-04-28

Family

ID=34120044

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200601552A EA009768B1 (ru) 2003-08-01 2004-07-30 Замещенные конденсированные гетероциклические с-гликозиды

Country Status (9)

Country Link
US (4) US7094763B2 (ru)
EP (1) EP1679965A4 (ru)
AR (1) AR048376A1 (ru)
AU (1) AU2004261660A1 (ru)
CA (1) CA2549015A1 (ru)
EA (1) EA009768B1 (ru)
IL (1) IL175489A0 (ru)
TW (1) TW200521131A (ru)
WO (1) WO2005012318A2 (ru)

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AU2002246317A1 (en) 2002-04-08 2003-10-27 Council Of Scientific And Industrial Research Novel glucopyranoside, process for isolation thereof, pharmaceutical composition containing same and use thereof
PL1980560T3 (pl) 2003-03-14 2011-11-30 Astellas Pharma Inc Pochodne C-glikozydowe do leczenia cukrzycy
JP2004300102A (ja) 2003-03-31 2004-10-28 Kissei Pharmaceut Co Ltd 縮合複素環誘導体、それを含有する医薬組成物およびその医薬用途
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US7816328B2 (en) 2010-10-19
CA2549015A1 (en) 2005-02-10
EA009768B1 (ru) 2008-04-28
US20090105162A1 (en) 2009-04-23
EP1679965A4 (en) 2009-05-27
EP1679965A2 (en) 2006-07-19
WO2005012318A2 (en) 2005-02-10
TW200521131A (en) 2005-07-01
US7482330B2 (en) 2009-01-27
AR048376A1 (es) 2006-04-26
US20050037980A1 (en) 2005-02-17
US20060229260A1 (en) 2006-10-12
IL175489A0 (en) 2009-02-11
US20100004160A1 (en) 2010-01-07

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