EA200501669A1 - Замещенные производные индолина и индола - Google Patents
Замещенные производные индолина и индолаInfo
- Publication number
- EA200501669A1 EA200501669A1 EA200501669A EA200501669A EA200501669A1 EA 200501669 A1 EA200501669 A1 EA 200501669A1 EA 200501669 A EA200501669 A EA 200501669A EA 200501669 A EA200501669 A EA 200501669A EA 200501669 A1 EA200501669 A1 EA 200501669A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- indoline
- indol
- substituted derivatives
- pharmaceutically acceptable
- general formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DKPA200300631 | 2003-04-25 | ||
PCT/DK2004/000283 WO2004096767A1 (fr) | 2003-04-25 | 2004-04-23 | Derives indole et indoline substitues |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200501669A1 true EA200501669A1 (ru) | 2006-04-28 |
Family
ID=58707218
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200501669A EA200501669A1 (ru) | 2003-04-25 | 2004-04-23 | Замещенные производные индолина и индола |
Country Status (10)
Country | Link |
---|---|
KR (1) | KR20060004957A (fr) |
CN (1) | CN1777582A (fr) |
AR (1) | AR044517A1 (fr) |
BR (1) | BRPI0409317A (fr) |
CA (1) | CA2523102A1 (fr) |
EA (1) | EA200501669A1 (fr) |
IS (1) | IS8002A (fr) |
NZ (1) | NZ541999A (fr) |
UA (1) | UA80190C2 (fr) |
ZA (1) | ZA200507186B (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103508960B (zh) * | 2012-06-29 | 2017-12-12 | 江苏先声药业有限公司 | 苯并杂环衍生物 |
CN108863893A (zh) * | 2018-07-09 | 2018-11-23 | 湖南博隽生物医药有限公司 | 二氢吲哚类衍生物及其在药物中的应用 |
CN112010808B (zh) * | 2019-05-31 | 2021-11-30 | 上海挚盟医药科技有限公司 | 作为钾通道调节剂的四氢-1h-苯氮杂卓类化合物及其制备和应用 |
-
2004
- 2004-04-23 BR BRPI0409317-8A patent/BRPI0409317A/pt not_active IP Right Cessation
- 2004-04-23 NZ NZ541999A patent/NZ541999A/en unknown
- 2004-04-23 EA EA200501669A patent/EA200501669A1/ru unknown
- 2004-04-23 CA CA002523102A patent/CA2523102A1/fr not_active Abandoned
- 2004-04-23 UA UAA200509297A patent/UA80190C2/uk unknown
- 2004-04-23 ZA ZA200507186A patent/ZA200507186B/en unknown
- 2004-04-23 AR ARP040101392A patent/AR044517A1/es not_active Application Discontinuation
- 2004-04-23 KR KR1020057020204A patent/KR20060004957A/ko not_active Application Discontinuation
- 2004-04-23 CN CNA2004800110190A patent/CN1777582A/zh active Pending
-
2005
- 2005-08-29 IS IS8002A patent/IS8002A/is unknown
Also Published As
Publication number | Publication date |
---|---|
CA2523102A1 (fr) | 2004-11-11 |
UA80190C2 (en) | 2007-08-27 |
ZA200507186B (en) | 2006-11-29 |
CN1777582A (zh) | 2006-05-24 |
AR044517A1 (es) | 2005-09-14 |
IS8002A (is) | 2005-08-29 |
KR20060004957A (ko) | 2006-01-16 |
BRPI0409317A (pt) | 2006-04-25 |
NZ541999A (en) | 2009-03-31 |
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