DK7483A - Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf - Google Patents

Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf Download PDF

Info

Publication number: DK7483A
Authority: DK; Denmark
Prior art keywords: sublicencillanic; aminoal; dioxides; derivatives; preparation
Prior art date: 1982-01-11

Application number

DK7483A

Other languages

English (en)

Other versions

DK7483D0 (da

DK166883B1 (da

Inventor

Wayne Ernest Barth

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-01-11

Filing date

1983-01-10

Publication date

1983-07-12

1982-06-14 Priority claimed from US06/388,323 external-priority patent/US4427678A/en

1982-10-21 Priority claimed from US06/434,371 external-priority patent/US4452796A/en

1983-01-10 Application filed by Pfizer filed Critical Pfizer

1983-01-10 Publication of DK7483D0 publication Critical patent/DK7483D0/da

1983-07-12 Publication of DK7483A publication Critical patent/DK7483A/da

1993-07-26 Application granted granted Critical

1993-07-26 Publication of DK166883B1 publication Critical patent/DK166883B1/da

Links

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Medicinal Preparation (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

DK007483A 1982-01-11 1983-01-10 Analogifremgangsmaade til fremstilling af 6-aminoalkylpenicillansyre-1,1-dioxider samt derivater eller salte deraf DK166883B1 (da)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
US33879782A	1982-01-11	1982-01-11
US33879782		1982-01-11
US38832482A	1982-06-14	1982-06-14
US38832382		1982-06-14
US06/388,323 US4427678A (en)	1982-01-11	1982-06-14	6-Aminomethylpenicillanic acid 1,1-dioxide derivatives as beta-lactamase inhibitors
US38832482		1982-06-14
US43437182		1982-10-21
US06/434,371 US4452796A (en)	1982-06-14	1982-10-21	6-Aminoalkylpenicillanic acid 1,1-dioxides as beta-lactamase inhibitors

Publications (3)

Publication Number	Publication Date
DK7483D0 DK7483D0 (da)	1983-01-10
DK7483A true DK7483A (da)	1983-07-12
DK166883B1 DK166883B1 (da)	1993-07-26

Family

ID=27502592

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK007483A DK166883B1 (da)	1982-01-11	1983-01-10	Analogifremgangsmaade til fremstilling af 6-aminoalkylpenicillansyre-1,1-dioxider samt derivater eller salte deraf

Country Status (20)

Country	Link
EP (1)	EP0084925B1 (da)
JP (1)	JPH0689005B2 (da)
AU (1)	AU538468B2 (da)
BG (1)	BG42676A3 (da)
CA (1)	CA1190921A (da)
DD (2)	DD209462A5 (da)
DE (1)	DE3362826D1 (da)
DK (1)	DK166883B1 (da)
ES (2)	ES8403489A1 (da)
FI (1)	FI79112C (da)
GR (1)	GR77152B (da)
HU (1)	HU189211B (da)
IE (1)	IE54390B1 (da)
IL (1)	IL67647A (da)
NO (6)	NO830046L (da)
NZ (1)	NZ202982A (da)
PL (1)	PL142315B1 (da)
PT (1)	PT76077B (da)
RO (2)	RO84910B (da)
YU (1)	YU43646B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4502990A (en) *	1983-06-06	1985-03-05	Pfizer Inc.	Process for 6-(aminomethyl)penicillanic acid 1,1-dioxide and derivatives thereof
US4499017A (en) *	1983-06-06	1985-02-12	Pfizer Inc.	Beta-lactamase inhibiting 6-(alkoxyamino-methyl) penicillanic acid 1,1-dioxide and derivatives
JPS60239489A (ja) *	1984-05-15	1985-11-28	Meiji Seika Kaisha Ltd	６−エピペニシリンスルホン化合物及びその製造方法
GB2206579B (en) *	1987-07-10	1991-05-29	Erba Farmitalia	6a and 6b-(substituted methyl)-penicillanic acid derivatives
ES2428167T3 (es) *	2007-05-21	2013-11-06	Hans Rudolf Pfaendler	Composición farmacéutica bactericida activa anti-MRSA conteniendo carbapenemos

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4237051A (en) *	1979-04-19	1980-12-02	Schering Corporation	Stereospecific production of 6- or 7-carbon-substituted-β-lactams
DE2927004A1 (de) *	1979-07-04	1981-05-27	Bayer Ag, 5090 Leverkusen	Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) *	1979-10-22	1981-09-01	Pfizer Inc.	Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

1983
- 1983-01-04 RO RO109609A patent/RO84910B/ro unknown
- 1983-01-04 RO RO83113375A patent/RO87705A/ro unknown
- 1983-01-05 DE DE8383300042T patent/DE3362826D1/de not_active Expired
- 1983-01-05 EP EP83300042A patent/EP0084925B1/en not_active Expired
- 1983-01-07 NO NO830046A patent/NO830046L/no unknown
- 1983-01-07 GR GR70215A patent/GR77152B/el unknown
- 1983-01-10 HU HU8370A patent/HU189211B/hu not_active IP Right Cessation
- 1983-01-10 BG BG8359284A patent/BG42676A3/xx unknown
- 1983-01-10 AU AU10232/83A patent/AU538468B2/en not_active Ceased
- 1983-01-10 NZ NZ202982A patent/NZ202982A/en unknown
- 1983-01-10 CA CA000419181A patent/CA1190921A/en not_active Expired
- 1983-01-10 IL IL67647A patent/IL67647A/xx not_active IP Right Cessation
- 1983-01-10 PT PT76077A patent/PT76077B/pt not_active IP Right Cessation
- 1983-01-10 IE IE42/83A patent/IE54390B1/en not_active IP Right Cessation
- 1983-01-10 YU YU44/83A patent/YU43646B/xx unknown
- 1983-01-10 DK DK007483A patent/DK166883B1/da active
- 1983-01-10 FI FI830081A patent/FI79112C/fi not_active IP Right Cessation
- 1983-01-11 PL PL1983240108A patent/PL142315B1/pl unknown
- 1983-01-11 ES ES518912A patent/ES8403489A1/es not_active Expired
- 1983-01-11 DD DD83247166A patent/DD209462A5/de not_active IP Right Cessation
- 1983-01-11 JP JP58002768A patent/JPH0689005B2/ja not_active Expired - Lifetime
- 1983-01-11 DD DD83262053A patent/DD218365A5/de not_active IP Right Cessation
- 1983-08-30 ES ES525238A patent/ES8507147A1/es not_active Expired
- 1983-09-22 NO NO833416A patent/NO833416L/no unknown
- 1983-09-22 NO NO833415A patent/NO833415L/no unknown
1984
- 1984-03-20 NO NO841069A patent/NO841069L/no unknown
- 1984-03-20 NO NO841068A patent/NO841068L/no unknown
- 1984-03-20 NO NO841070A patent/NO841070L/no unknown

Also Published As

Publication number	Publication date
NO841068L (no)	1983-07-12
RO84910B (ro)	1984-09-30
YU4483A (en)	1986-02-28
ES525238A0 (es)	1985-08-16
RO87705A (ro)	1985-10-31
NO830046L (no)	1983-07-12
DD218365A5 (de)	1985-02-06
HU189211B (en)	1986-06-30
JPS58126889A (ja)	1983-07-28
FI79112C (fi)	1989-11-10
GR77152B (da)	1984-09-07
DK7483D0 (da)	1983-01-10
YU43646B (en)	1989-10-31
PL240108A1 (en)	1985-08-13
NO841070L (no)	1983-07-12
DD209462A5 (de)	1984-05-09
PT76077B (en)	1986-01-09
BG42676A3 (en)	1988-01-15
ES518912A0 (es)	1984-03-16
ES8507147A1 (es)	1985-08-16
AU538468B2 (en)	1984-08-16
FI830081L (fi)	1983-07-12
AU1023283A (en)	1983-07-21
FI830081A0 (fi)	1983-01-10
DK166883B1 (da)	1993-07-26
RO84910A (ro)	1984-08-17
IE54390B1 (en)	1989-09-13
IL67647A0 (en)	1983-05-15
RO87705B (ro)	1985-10-01
NO841069L (no)	1983-07-12
EP0084925A1 (en)	1983-08-03
NO833416L (no)	1983-07-12
IL67647A (en)	1986-08-31
EP0084925B1 (en)	1986-04-09
PL142315B1 (en)	1987-10-31
CA1190921A (en)	1985-07-23
NZ202982A (en)	1986-04-11
DE3362826D1 (en)	1986-05-15
NO833415L (no)	1983-07-12
ES8403489A1 (es)	1984-03-16
FI79112B (fi)	1989-07-31
JPH0689005B2 (ja)	1994-11-09
IE830042L (en)	1983-07-11
PT76077A (en)	1983-02-01

Publication	Publication Date	Title
NO821087L (no)	1982-10-07	Fremgangsmaate for fremstilling av cyklobutan-derivater.
DK112582A (da)	1982-09-17	Fremgangsmaade til fremstilling af triazolonderivater
DK307883D0 (da)	1983-07-04	Carbostyrilderivater samt fremgangsmade til fremstilling deraf
DK435181A (da)	1982-05-12	Fremgangsmaade til fremstilling af thiazol-derivater
DK66582A (da)	1982-08-18	Fremgangsmaade til fremstilling af carbostyrilderivater
DK106897A (da)	1997-09-17	Fremgangsmåde til fremstilling af urinstofderivater
DK158269C (da)	1990-10-08	Analogifremgangsmaade til fremstilling af morpholinyldaunorubicin- eller morpholinyldoxorubicinderivater
DK491582A (da)	1983-05-10	Fremgangsmaade til fremstilling af morphinanderivater
DK352082A (da)	1983-02-08	Fremgangsmaade til fremstilling af ergopeptinderivater
NO155693C (no)	1987-05-13	Fremgangsmaate for fremstilling av eburnamoninderivater.
ES522823A0 (es)	1984-08-16	Derivados de 6 -metilprednisolona.
DK116982A (da)	1982-09-18	Fremgangsmaade til fremstilling af alkylendioxybenzenderivater
DK7483A (da)	1983-07-12	Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf
DK113483D0 (da)	1983-03-08	Fremgangsmade til fremstilling af 3,4-diphenyl-5-methylpyrazolderivater
NO157143C (no)	1988-01-27	Fremgangsmaate for fremstilling av karbapen-2-em-derivater.
DK423284D0 (da)	1984-09-05	Naphthalenylimidazopyridin og derivater heraf samt fremgangsmaade til fremstilling af saadanne forbindelser
DK364483A (da)	1984-02-13	14-aminosteroid-derivater samt fremgangsmaade til fremstilling deraf
DK375882A (da)	1983-02-27	Fremgangsmaade til fremstilling af benzisoxazolderivater
DK570082A (da)	1983-06-26	4-cyan-2-azetidinoner samt fremgangsmaade til fremstilling af saadanne
ES517428A0 (es)	1983-08-16	Procedimiento de preparacion de derivados bencilidenicos.
DK70482A (da)	1982-08-20	Fremgangsmaade til fremstilling af diazolderivater
DK157036C (da)	1990-03-26	Endo-deoxyribonuklease a samt fremgangsmaade til fremstilling af samme
DK135081A (da)	1981-10-04	Fr&mgangsmaade til fremstilling af thiazoler
ES522652A0 (es)	1985-02-01	Procedimiento de preparacion de derivados de piperacina.
DK370982A (da)	1983-02-20	Fremgangsmaade til fremstilling af fluorerede alkandiaminderivater