DK199900554A - Paroxetinsalte, fremgangsmåde til fremstilling deraf, farmaceutiske præparater omfattende disse og anvendelser deraf - Google Patents

Paroxetinsalte, fremgangsmåde til fremstilling deraf, farmaceutiske præparater omfattende disse og anvendelser deraf

Info

Publication number
DK199900554A
DK199900554A DK199900554A DKPA199900554A DK199900554A DK 199900554 A DK199900554 A DK 199900554A DK 199900554 A DK199900554 A DK 199900554A DK PA199900554 A DKPA199900554 A DK PA199900554A DK 199900554 A DK199900554 A DK 199900554A
Authority
DK
Denmark
Prior art keywords
preparation
pharmaceutical compositions
paroxetine salts
paroxetine
salts
Prior art date
Application number
DK199900554A
Other languages
Danish (da)
English (en)
Inventor
Andrew Simon Craig
Jones Alan David
O'keeffe Deidre
Ward Neal
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269380&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK199900554(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9814316.7A external-priority patent/GB9814316D0/en
Priority claimed from GBGB9821732.6A external-priority patent/GB9821732D0/en
Priority claimed from GBGB9902935.7A external-priority patent/GB9902935D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of DK199900554A publication Critical patent/DK199900554A/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Inorganic Chemistry (AREA)
  • Psychology (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK199900554A 1998-07-02 1999-04-23 Paroxetinsalte, fremgangsmåde til fremstilling deraf, farmaceutiske præparater omfattende disse og anvendelser deraf DK199900554A (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9814316.7A GB9814316D0 (en) 1998-07-02 1998-07-02 Novel compounds
GBGB9821732.6A GB9821732D0 (en) 1998-10-06 1998-10-06 Novel compound
GBGB9902935.7A GB9902935D0 (en) 1999-02-10 1999-02-10 Novel compound

Publications (1)

Publication Number Publication Date
DK199900554A true DK199900554A (da) 2000-01-03

Family

ID=27269380

Family Applications (7)

Application Number Title Priority Date Filing Date
DK199900176U DK199900176U3 (da) 1998-07-02 1999-04-23 Paroxetinsalte, farmaceutisk præparat indeholdende disse og anvendelser deraf
DK199900554A DK199900554A (da) 1998-07-02 1999-04-23 Paroxetinsalte, fremgangsmåde til fremstilling deraf, farmaceutiske præparater omfattende disse og anvendelser deraf
DK99918159T DK1089996T3 (da) 1998-07-02 1999-04-23 Paroxetin-methansulfonat-acetonitril-solvat 1:1
DK99303151T DK0970955T3 (da) 1998-07-02 1999-04-23 Paroxetin-methansulfonat
DK199900234U DK199900234U4 (da) 1998-07-02 1999-06-15 Paroxetin-methansulfonat i krystallinsk form, farmaceutisk præparat indeholdende dette og andvendelse af forbindelsen til f
DK00201290T DK1020464T3 (da) 1998-07-02 2000-04-10 Paroxetin-methansulfonat
DK200000390U DK200000390U1 (da) 1998-07-02 2000-12-27 Farmaceutiske præparater til oral indgivelse, der omfatter paroxetin-methansulfonat.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK199900176U DK199900176U3 (da) 1998-07-02 1999-04-23 Paroxetinsalte, farmaceutisk præparat indeholdende disse og anvendelser deraf

Family Applications After (5)

Application Number Title Priority Date Filing Date
DK99918159T DK1089996T3 (da) 1998-07-02 1999-04-23 Paroxetin-methansulfonat-acetonitril-solvat 1:1
DK99303151T DK0970955T3 (da) 1998-07-02 1999-04-23 Paroxetin-methansulfonat
DK199900234U DK199900234U4 (da) 1998-07-02 1999-06-15 Paroxetin-methansulfonat i krystallinsk form, farmaceutisk præparat indeholdende dette og andvendelse af forbindelsen til f
DK00201290T DK1020464T3 (da) 1998-07-02 2000-04-10 Paroxetin-methansulfonat
DK200000390U DK200000390U1 (da) 1998-07-02 2000-12-27 Farmaceutiske præparater til oral indgivelse, der omfatter paroxetin-methansulfonat.

Country Status (35)

Country Link
US (4) US6063927A (fr)
EP (5) EP1089996B1 (fr)
JP (1) JP2002519422A (fr)
KR (1) KR20010053336A (fr)
CN (1) CN1127502C (fr)
AR (2) AR011759A1 (fr)
AT (4) AT3185U3 (fr)
AU (4) AU713131B3 (fr)
BE (3) BE1012403A5 (fr)
BR (1) BR9911682A (fr)
CA (1) CA2269999A1 (fr)
CH (1) CH689805A8 (fr)
DE (5) DE29907248U1 (fr)
DK (7) DK199900176U3 (fr)
ES (4) ES2158778B1 (fr)
FI (2) FI4209U1 (fr)
FR (2) FR2780728B1 (fr)
GB (5) GB2367003A (fr)
GR (3) GR990100140A (fr)
HK (1) HK1037877A1 (fr)
HU (1) HUP0102334A3 (fr)
IE (5) IES20000894A2 (fr)
IL (1) IL140628A (fr)
IT (1) IT1312540B1 (fr)
LU (1) LU90388B1 (fr)
NL (4) NL1011875C2 (fr)
NO (1) NO319030B1 (fr)
NZ (1) NZ509180A (fr)
PL (1) PL345214A1 (fr)
PT (4) PT1020464E (fr)
SE (1) SE9901462A0 (fr)
SI (3) SI0970955T1 (fr)
SK (1) SK20262000A3 (fr)
TR (1) TR200100054T2 (fr)
WO (1) WO2000001694A1 (fr)

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Also Published As

Publication number Publication date
DE69911774D1 (de) 2003-11-06
ATE202777T1 (de) 2001-07-15
BE1012403A5 (fr) 2000-10-03
KR20010053336A (ko) 2001-06-25
SK20262000A3 (sk) 2001-07-10
GR3034328T3 (en) 2000-12-29
TR200100054T2 (tr) 2001-06-21
GR3036208T3 (en) 2001-10-31
CH689805A5 (fr) 1999-11-30
NO991944L (no) 2000-01-03
GB9920332D0 (en) 1999-11-03
BE1011664A6 (fr) 1999-11-09
SI1020464T1 (en) 2001-12-31
GR1003350B (el) 2000-03-29
IE990344A1 (en) 2000-05-03
DE60000003D1 (de) 2001-08-09
BR9911682A (pt) 2001-12-26
EP1020463A1 (fr) 2000-07-19
AR018197A1 (es) 2001-10-31
CN1315949A (zh) 2001-10-03
DK200000390U1 (da) 2000-12-27
EP0970955A1 (fr) 2000-01-12
GB2377637A (en) 2003-01-22
IT1312540B1 (it) 2002-04-22
EP1288214A1 (fr) 2003-03-05
SI1089996T1 (en) 2004-04-30
NL1011875C2 (nl) 2000-03-24
FI990922A0 (fi) 1999-04-23
AU713877B3 (en) 1999-12-09
BE1012420A6 (fr) 2000-10-03
EP1089996A1 (fr) 2001-04-11
IES20000894A2 (en) 2001-05-30
NO319030B1 (no) 2005-06-06
GB0026487D0 (en) 2000-12-13
FIU990190U0 (fi) 1999-04-23
AU732211B2 (en) 2001-04-12
AR011759A1 (es) 2000-09-13
SI0970955T1 (en) 2001-02-28
NL1012271A1 (nl) 1999-07-12
PT1089996E (pt) 2004-02-27
ES2157881T3 (es) 2001-09-01
IES81166B2 (en) 2000-05-31
FR2780728B1 (fr) 2001-02-16
PT970955E (pt) 2000-11-30
PT102291A (pt) 2000-05-31
CH689805A8 (fr) 2000-02-29
DE69911774T2 (de) 2004-08-05
EP0970955B1 (fr) 2000-08-02
NL1012271C2 (nl) 1999-09-23
FR2802098A1 (fr) 2001-06-15
IES990343A2 (en) 2000-01-02
US20020035130A1 (en) 2002-03-21
DK1020464T3 (da) 2001-09-24
US20010023253A1 (en) 2001-09-20
HK1037877A1 (en) 2002-02-22
AU3619199A (en) 2000-01-24
NL1011875A1 (nl) 2000-01-07
US20020193406A1 (en) 2002-12-19
PT1020464E (pt) 2001-10-30
DE60000003T2 (de) 2002-03-21
ES2209428T3 (es) 2004-06-16
CA2269999A1 (fr) 2000-01-02
EP1020464A1 (fr) 2000-07-19
ES2158778A1 (es) 2001-09-01
ES2149044T3 (es) 2000-10-16
AT3185U3 (de) 2000-01-25
IL140628A (en) 2004-06-20
ES2158778B1 (es) 2002-03-16
IL140628A0 (en) 2002-02-10
SE9901462D0 (sv) 1999-04-23
GR990100140A (el) 2000-03-31
LU90388B1 (fr) 2001-01-29
DK1089996T3 (da) 2004-02-09
GB2352395B (en) 2004-02-11
ITMI990866A1 (it) 2000-10-23
DE69900007D1 (de) 2000-09-07
GB9909505D0 (en) 1999-06-23
DK199900234U1 (da) 2000-12-22
AU713131B3 (en) 1999-11-25
DE29907248U1 (de) 1999-09-09
PT102291B (pt) 2002-07-31
GB0119695D0 (en) 2001-10-03
GB0216752D0 (en) 2002-08-28
ATE195121T1 (de) 2000-08-15
JP2002519422A (ja) 2002-07-02
US6063927A (en) 2000-05-16
DE19918588A1 (de) 2000-01-27
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AT3185U2 (de) 1999-11-25
FI112077B (fi) 2003-10-31
NL1012272C1 (nl) 1999-07-12
PL345214A1 (en) 2001-12-03
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FI990922A (fi) 2000-01-03
HUP0102334A3 (en) 2003-12-29
HUP0102334A2 (hu) 2002-05-29
GB2352395A (en) 2001-01-31
GB2336364B (en) 2000-05-10
SE9901462L (fr)
GB2339428A (en) 2000-01-26
EP1089996B1 (fr) 2003-10-01
NL1011874C1 (nl) 1999-07-12
GB2367003A (en) 2002-03-27
WO2000001694A1 (fr) 2000-01-13
DE69900007T2 (de) 2001-06-07
CN1127502C (zh) 2003-11-12
GB2336364A (en) 1999-10-20
IES20000893A2 (en) 2001-05-30
DK199900176U3 (da) 1999-08-13
ATE251155T1 (de) 2003-10-15
FI4209U1 (fi) 1999-11-10
IE20000633A1 (en) 2001-10-17
NZ509180A (en) 2001-06-29
EP1020464B1 (fr) 2001-07-04
AU732211C (en) 2004-05-06
AU2392899A (en) 2000-01-20
SE9901462A0 (sv) 2000-01-03
DK199900234U4 (da) 2000-12-22
FR2780728A1 (fr) 2000-01-07

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