DE60334787D1 - Substituierte amide - Google Patents

Substituierte amide

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Publication number
DE60334787D1
DE60334787D1 DE60334787T DE60334787T DE60334787D1 DE 60334787 D1 DE60334787 D1 DE 60334787D1 DE 60334787 T DE60334787 T DE 60334787T DE 60334787 T DE60334787 T DE 60334787T DE 60334787 D1 DE60334787 D1 DE 60334787D1
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Germany
Prior art keywords
treatment
disorders
useful
compounds
receptor
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60334787T
Other languages
English (en)
Inventor
William K Hagmann
Linus S Lin
Shrenik K Shah
Ravindra N Guthikonda
Hongbo Qi
Linda L Chang
Ping Liu
Helen M Armstrong
James P Jewell
Thomas J Lanza
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Merck Sharp and Dohme LLC
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Merck Sharp and Dohme LLC
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Publication of DE60334787D1 publication Critical patent/DE60334787D1/de
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
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EP1558252B1 (de) 2002-08-02 2007-10-10 Merck & Co., Inc. Substituierte furo[2,3-b]pyridin derivate
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US6972295B2 (en) 2005-12-06
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JP3813152B2 (ja) 2006-08-23
US7816534B2 (en) 2010-10-19
US20050234061A1 (en) 2005-10-20
WO2003077847A2 (en) 2003-09-25
US20040058820A1 (en) 2004-03-25
US20090258884A1 (en) 2009-10-15
ATE486842T1 (de) 2010-11-15
EP1496838A2 (de) 2005-01-19
EP1496838A4 (de) 2008-07-02
CA2478183A1 (en) 2003-09-25
NZ534757A (en) 2006-07-28
JP5025980B2 (ja) 2012-09-12
EP1496838B1 (de) 2010-11-03
WO2003077847A3 (en) 2004-11-04
AU2003218068A1 (en) 2003-09-29
JP2005519958A (ja) 2005-07-07
US20080171692A1 (en) 2008-07-17

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