DE60308040D1 - HERSTELLUNG VON 1H-IMIDAZOc4,5-CÜCHINOLIN-4-AMINEN BER 1H-IMIDAZOc4,5-CÜCHINOLIN-4-PHTHALIMIDZWISCHENPRODUKTE - Google Patents

HERSTELLUNG VON 1H-IMIDAZOc4,5-CÜCHINOLIN-4-AMINEN BER 1H-IMIDAZOc4,5-CÜCHINOLIN-4-PHTHALIMIDZWISCHENPRODUKTE

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Publication number
DE60308040D1
DE60308040D1 DE60308040T DE60308040T DE60308040D1 DE 60308040 D1 DE60308040 D1 DE 60308040D1 DE 60308040 T DE60308040 T DE 60308040T DE 60308040 T DE60308040 T DE 60308040T DE 60308040 D1 DE60308040 D1 DE 60308040D1
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DE
Germany
Prior art keywords
cuchinolin
imidazoc4
ber
amine
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60308040T
Other languages
English (en)
Other versions
DE60308040T2 (de
Inventor
Valeriano Merli
Silvia Mantovani
Stefano Bianchi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teva Pharmaceutical Works PLC
Original Assignee
Teva Pharmaceutical Works PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharmaceutical Works PLC filed Critical Teva Pharmaceutical Works PLC
Application granted granted Critical
Publication of DE60308040D1 publication Critical patent/DE60308040D1/de
Publication of DE60308040T2 publication Critical patent/DE60308040T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
DE60308040T 2002-07-23 2003-07-23 Herstellung von 1H-Imidazo-4,5-C]-Chinolin-4-Aminen Ber 1H-Imidazo-4,5-C]-Chinolin-4-Phthalimid-Zwischenprodukten Expired - Fee Related DE60308040T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US39760702P 2002-07-23 2002-07-23
US397607P 2002-07-23
PCT/US2003/023153 WO2004009593A1 (en) 2002-07-23 2003-07-23 Preparation of 1h-imidazo[4,5-c]quinolin-4-amines via1h-imidazo [4,5-c]quinolin-4-phthalimide intermediates

Publications (2)

Publication Number Publication Date
DE60308040D1 true DE60308040D1 (de) 2006-10-12
DE60308040T2 DE60308040T2 (de) 2007-04-19

Family

ID=30771087

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60308040T Expired - Fee Related DE60308040T2 (de) 2002-07-23 2003-07-23 Herstellung von 1H-Imidazo-4,5-C]-Chinolin-4-Aminen Ber 1H-Imidazo-4,5-C]-Chinolin-4-Phthalimid-Zwischenprodukten

Country Status (17)

Country Link
US (3) US6852861B2 (de)
EP (1) EP1543002B1 (de)
JP (1) JP2006502121A (de)
KR (1) KR20050028047A (de)
CN (1) CN1315828C (de)
AT (1) ATE338044T1 (de)
AU (1) AU2003259226A1 (de)
CA (1) CA2493227A1 (de)
DE (1) DE60308040T2 (de)
DK (1) DK1543002T3 (de)
ES (1) ES2271650T3 (de)
HR (1) HRP20050159A2 (de)
IL (1) IL166309A (de)
MX (1) MXPA05000893A (de)
PL (1) PL374884A1 (de)
PT (1) PT1543002E (de)
WO (1) WO2004009593A1 (de)

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EA200700244A1 (ru) * 2004-12-27 2007-06-29 Ю Эс Ви ЛИМИТЕД СПОСОБ ПОЛУЧЕНИЯ 4-АМИНО-1-ИЗОБУТИЛ-1H-ИМИДАЗО-[4,5-c]ХИНОЛИНА (ИМИХИМОД)
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AR052447A1 (es) * 2004-12-30 2007-03-21 3M Innovative Properties Co Etansulfonato de 1-(2-metipropil)-1h-imidazo[4,5-c] [1,5] naftiridin-4- amina y metansulfonato de 1-(2- metipropil)-1h-imidazo[4,5 -c] [1,5] naftiridin-4-amina
US8436176B2 (en) * 2004-12-30 2013-05-07 Medicis Pharmaceutical Corporation Process for preparing 2-methyl-1-(2-methylpropyl)-1H-imidazo[4,5-c][1,5]naphthyridin-4-amine
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PL1830876T3 (pl) * 2004-12-30 2015-09-30 Meda Ab Zastosowanie imikwimodu do leczenia przerzutów do skóry wywodzących się od guza stanowiącego raka piersi
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JP5122980B2 (ja) 2005-02-09 2013-01-16 スリーエム イノベイティブ プロパティズ カンパニー アルキルオキシ置換チアゾロキノリン類およびアルキルオキシ置換チアゾロナフチリデン類
JP2008532933A (ja) * 2005-02-11 2008-08-21 コーリー ファーマシューティカル グループ，インコーポレイテッド 置換イミダゾキノリン類および置換イミダゾナフチリジン類
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JP2008531568A (ja) 2005-02-23 2008-08-14 コーリー ファーマシューティカル グループ，インコーポレイテッド ヒドロキシアルキルで置換されたイミダゾナフチリジン
JP2008535832A (ja) 2005-04-01 2008-09-04 コーリー ファーマシューティカル グループ，インコーポレイテッド ピラゾロピリジン−１，４−ジアミン、およびそのアナログ
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Also Published As

Publication number Publication date
DE60308040T2 (de) 2007-04-19
DK1543002T3 (da) 2006-12-27
IL166309A0 (en) 2006-01-15
PT1543002E (pt) 2006-11-30
WO2004009593A1 (en) 2004-01-29
US20040138459A1 (en) 2004-07-15
HRP20050159A2 (en) 2005-08-31
ES2271650T3 (es) 2007-04-16
US20050113404A1 (en) 2005-05-26
KR20050028047A (ko) 2005-03-21
CA2493227A1 (en) 2004-01-29
ATE338044T1 (de) 2006-09-15
PL374884A1 (en) 2005-11-14
AU2003259226A1 (en) 2004-02-09
US6852861B2 (en) 2005-02-08
CN1315828C (zh) 2007-05-16
EP1543002A1 (de) 2005-06-22
CN1681814A (zh) 2005-10-12
EP1543002B1 (de) 2006-08-30
JP2006502121A (ja) 2006-01-19
US20070060755A1 (en) 2007-03-15
US7153967B2 (en) 2006-12-26
MXPA05000893A (es) 2005-09-30
IL166309A (en) 2010-04-15

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