DD151448A5 - Verfahren zur herstellung von benzothiazolderivaten - Google Patents

Verfahren zur herstellung von benzothiazolderivaten Download PDF

Info

Publication number
DD151448A5
DD151448A5 DD80220177A DD22017780A DD151448A5 DD 151448 A5 DD151448 A5 DD 151448A5 DD 80220177 A DD80220177 A DD 80220177A DD 22017780 A DD22017780 A DD 22017780A DD 151448 A5 DD151448 A5 DD 151448A5
Authority
DD
German Democratic Republic
Prior art keywords
acid
formula
compound
salt
salts
Prior art date
Application number
DD80220177A
Other languages
German (de)
English (en)
Inventor
Marcel Lepant
Pierre Bessin
Jacqueline Bonnet
Original Assignee
Rolland Sa A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rolland Sa A filed Critical Rolland Sa A
Publication of DD151448A5 publication Critical patent/DD151448A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/64Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • C07D277/66Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82Nitrogen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
DD80220177A 1979-04-03 1980-04-02 Verfahren zur herstellung von benzothiazolderivaten DD151448A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7908303A FR2453163A1 (fr) 1979-04-03 1979-04-03 Derives de benzothiazole, leur procede de preparation et leurs applications en therapeutique

Publications (1)

Publication Number Publication Date
DD151448A5 true DD151448A5 (de) 1981-10-21

Family

ID=9223868

Family Applications (1)

Application Number Title Priority Date Filing Date
DD80220177A DD151448A5 (de) 1979-04-03 1980-04-02 Verfahren zur herstellung von benzothiazolderivaten

Country Status (27)

Country Link
EP (1) EP0017543B1 (es)
JP (1) JPS55133367A (es)
AR (1) AR227884A1 (es)
AT (1) ATE4807T1 (es)
AU (1) AU530911B2 (es)
BE (1) BE882270A (es)
CA (1) CA1144556A (es)
DD (1) DD151448A5 (es)
DE (1) DE3065004D1 (es)
DK (1) DK134880A (es)
ES (2) ES490797A0 (es)
FI (1) FI801023A (es)
FR (1) FR2453163A1 (es)
GR (1) GR67195B (es)
HU (1) HU178851B (es)
IL (1) IL59655A (es)
IT (1) IT8048308A0 (es)
MA (1) MA18772A1 (es)
NO (1) NO800946L (es)
NZ (1) NZ193337A (es)
OA (1) OA06504A (es)
PH (1) PH15451A (es)
PL (1) PL123701B1 (es)
PT (1) PT71035A (es)
SU (1) SU910120A3 (es)
YU (1) YU80780A (es)
ZA (1) ZA801574B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1303043C (zh) 2002-02-05 2007-03-07 住友化学工业株式会社 二芳基化合物的制备方法
TWI458711B (zh) 2010-07-02 2014-11-01 Gilead Sciences Inc 治療性化合物
AP2013006706A0 (en) 2010-07-02 2013-02-28 Gilead Sciences Inc Napht-2-ylacetic acid derivatives to treat AIDS
EP2699558B1 (en) * 2011-04-21 2016-11-23 Gilead Sciences, Inc. Benzothiazole compounds and their pharmaceutical use
US9284323B2 (en) 2012-01-04 2016-03-15 Gilead Sciences, Inc. Naphthalene acetic acid derivatives against HIV infection
US9376392B2 (en) 2012-01-04 2016-06-28 Gilead Sciences, Inc. 2-(tert-butoxy)-2-(7-methylquinolin-6-yl) acetic acid derivatives for treating AIDS
MX2014005002A (es) 2012-04-20 2014-07-09 Gilead Sciences Inc Derivados de acido benzotiazol-6-il acetico y su uso para tratar una infeccion por vih.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2145178C3 (de) * 1970-09-11 1975-12-11 Tokyo Tanabe Co., Ltd., Tokio 2-Phenyl-5-oder -6-benzothiazolylessigsäure-Verblndungen
US3895028A (en) * 1972-09-12 1975-07-15 Tokyo Tanabe Co Alpha-(2-phenylbenzothiazol-5-yl)propionic acid

Also Published As

Publication number Publication date
ES8204989A1 (es) 1982-06-01
ATE4807T1 (de) 1983-10-15
AU5686480A (en) 1980-10-09
FR2453163B1 (es) 1982-07-02
FR2453163A1 (fr) 1980-10-31
DK134880A (da) 1980-10-04
PH15451A (en) 1983-01-18
BE882270A (fr) 1980-09-17
FI801023A (fi) 1980-10-04
ES8200098A1 (es) 1981-11-01
SU910120A3 (ru) 1982-02-28
PL123701B1 (en) 1982-11-30
DE3065004D1 (en) 1983-11-03
EP0017543A1 (fr) 1980-10-15
IL59655A0 (en) 1980-06-30
OA06504A (fr) 1981-07-31
HU178851B (en) 1982-07-28
ES490797A0 (es) 1981-11-01
AU530911B2 (en) 1983-08-04
AR227884A1 (es) 1982-12-30
PT71035A (fr) 1980-04-01
ZA801574B (en) 1981-03-25
NZ193337A (en) 1982-12-07
CA1144556A (en) 1983-04-12
NO800946L (no) 1980-10-06
MA18772A1 (fr) 1980-10-01
IT8048308A0 (it) 1980-04-01
PL223191A1 (es) 1981-01-30
EP0017543B1 (fr) 1983-09-28
IL59655A (en) 1983-05-15
YU80780A (en) 1983-02-28
GR67195B (es) 1981-06-24
ES498313A0 (es) 1982-06-01
JPS55133367A (en) 1980-10-17

Similar Documents

Publication Publication Date Title
DE1668648C3 (de) 3-Benzoylphenylessigsäurederivate, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
DE1595915C3 (de) Pyrrolidinderivate
EP0004279B1 (de) Verfahren zur Herstellung von 4-Pyridon-3-carbonsäuren, 1-Cyclopropyl-4-Pyridon-3-Carbonsäurederivate und diese enthaltende Arzneimittel
DD242229A5 (de) Verfahren zur herstellung von neuen derivaten der alpha-/oxo-2-hexahydro-2,4,5,6,7a thieno (3,2-c) pyridyl-5) phenyl-essig-saurer saeure
DE2205815A1 (de) Piperazinderivate und verfahren zu ihrer herstellung
DE2047658C3 (de) 2-Styryl- und 2-Phenyläthinylbenzylaminderivate, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
DE2803651C2 (es)
DE2122273C3 (de) Substituierte Phenylessigsäureverbindungen, sie enthaltende entzündungshemmende, antipyretische und analgetische Mittel und Verfahren zu ihrer Herstellung
DD151448A5 (de) Verfahren zur herstellung von benzothiazolderivaten
DE1618465C3 (de) Phenylessigsäureester, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
CH622491A5 (en) Process for the preparation of novel hydroxypropylamines
DE2354931C2 (de) trans-2-Phenylbicyclooctan-Verbindungen, Verfahren zu ihrer Herstellung und sie enthaltende pharmazeutische Zubereitungen
DE2907379A1 (de) Benzylidenderivate, verfahren zu ihrer herstellung und sie enthaltende arzneimittel
EP0224849B1 (de) Verfahren zur Herstellung von 4-Mercaptobenzonitrilen und neue 4-Mercaptobenzonitrile
CH356121A (de) Verfahren zur Herstellung von N-monosubstituierten Amiden vona-Aminoalkyl-a-phenyl-essigsäuren
DE862602C (de) Verfahren zur Herstellung von Halogendiamidinen und ihren Salzen
AT220614B (de) Verfahren zur Herstellung neuer substituierter Amine und ihrer Salze
AT270630B (de) Verfahren zur Herstellung von neuen Pyrrolinderivaten und ihren Salzen
DE1793802A1 (de) Organische verbindungen mit 2 bis 4 dicyanacetatgruppen
AT226710B (de) Verfahren zur Herstellung von neuen Dihydrochinoxalonen-(2) und von deren Salzen
AT367029B (de) Verfahren zur herstellung von neuen racemischen oder optisch aktiven phenylessigsaeureamiden
AT357515B (de) Verfahren zur herstellung von neuen thieno- thienylcarbonylphenyl-alkansaeuren, von deren derivaten und den salzen
AT350574B (de) Verfahren zur herstellung von neuen chinol-2-on -4-yl-alkansaeuren und von deren basenadditons- salzen
AT277246B (de) Verfahren zur Herstellung von neuen Pyridincarbonsäuren und von deren Salzen
AT330181B (de) Verfahren zur herstellung von neuen chinolinessigsaurederivaten und ihren salzen