DE60037455T2
(de)
|
1999-09-17 |
2008-11-27 |
Abbott Gmbh & Co. Kg |
Kinaseinhibitoren als arzneimittel
|
CN1321628C
(zh)
|
2000-06-28 |
2007-06-20 |
史密斯克莱·比奇曼公司 |
湿磨方法
|
WO2004035580A1
(en)
|
2002-10-21 |
2004-04-29 |
Aprea Ab |
Reactivation of wild type p53 in human tumour cells by a low molecular weight compound
|
US20050203063A1
(en)
|
2003-09-12 |
2005-09-15 |
Raymond Deshaies |
Proteasome pathway inhibitors and related methods
|
UY28931A1
(es)
|
2004-06-03 |
2005-12-30 |
Bayer Pharmaceuticals Corp |
Derivados de pirrolotriazina utiles para tratar trastornos hiper-proliferativos y enfermedades asociadas con angiogenesis
|
AR053090A1
(es)
|
2004-07-20 |
2007-04-25 |
Osi Pharm Inc |
Imidazotriazinas como inhibidores de proteina quinasas y su uso para la preparacion de medicamentos
|
UY29177A1
(es)
|
2004-10-25 |
2006-05-31 |
Astex Therapeutics Ltd |
Derivados sustituidos de purina, purinona y deazapurina, composiciones que los contienen métodos para su preparación y sus usos
|
JP5335432B2
(ja)
|
2005-11-17 |
2013-11-06 |
オーエスアイ・フアーマシユーテイカルズ・エル・エル・シー |
縮合2環系mTOR阻害剤
|
CN101466710B
(zh)
|
2005-12-02 |
2013-05-29 |
拜尔健康护理有限责任公司 |
用于治疗与血管生成有关的过度增殖性病症和疾病的取代的4-氨基-吡咯并三嗪衍生物
|
PE20070855A1
(es)
|
2005-12-02 |
2007-10-14 |
Bayer Pharmaceuticals Corp |
Derivados de 4-amino-pirrolotriazina sustituida como inhibidores de quinasas
|
MY162590A
(en)
|
2005-12-13 |
2017-06-30 |
Incyte Holdings Corp |
Heteroaryl substituted pyrrolo[2,3-b] pyridines and pyrrolo[2,3-b] pyrimidines as janus kinase inhibitors
|
ES2562428T3
(es)
|
2005-12-15 |
2016-03-04 |
Rigel Pharmaceuticals, Inc. |
Inhibidores de cinasa y sus usos
|
JP5313875B2
(ja)
|
2006-04-12 |
2013-10-09 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
増殖性疾患の処置のためのタンパク質キナーゼplk1の阻害剤として有用な4,5−ジヒドロ−[1,2,4]トリアゾロ[4,3−f]プテリジン
|
EP2016077A2
(en)
|
2006-04-25 |
2009-01-21 |
Astex Therapeutics Limited |
Pharmaceutical compounds
|
US8097630B2
(en)
|
2006-10-10 |
2012-01-17 |
Rigel Pharmaceuticals, Inc. |
Pinane-substituted pyrimidinediamine derivatives useful as Axl inhibitors
|
MX2009006345A
(es)
|
2006-12-14 |
2009-06-23 |
Vertex Pharma |
Compuestos utiles como inhibidores de proteina cinasa.
|
ME01832B
(me)
|
2006-12-29 |
2014-12-20 |
Rigel Pharmaceuticals Inc |
Policiklični heteroaril supstituisani triazoli koji su korisni kao axl inhibitori
|
EP2074115B1
(en)
|
2006-12-29 |
2018-03-07 |
Rigel Pharmaceuticals, Inc. |
N3-heteroaryl substituted triazoles and n5-heteroaryl substituted triazoles useful as axl inhibitors
|
CA2710043C
(en)
|
2006-12-29 |
2016-02-09 |
Rigel Pharmaceuticals, Inc. |
Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as axl inhibitors
|
WO2008098139A2
(en)
|
2007-02-07 |
2008-08-14 |
The Regents Of The University Of Colorado |
Axl tyrosine kinase inhibitors and methods of making and using the same
|
CA2695753A1
(en)
|
2007-08-15 |
2009-02-19 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as protein kinases inhibitors
|
GB0719803D0
(en)
|
2007-10-10 |
2007-11-21 |
Cancer Rec Tech Ltd |
Therapeutic compounds and their use
|
KR20100089090A
(ko)
|
2007-10-25 |
2010-08-11 |
아스트라제네카 아베 |
세포 증식 장애의 치료에 유용한 피리딘 및 피라진 유도체
|
ES2424259T3
(es)
|
2007-10-26 |
2013-09-30 |
Rigel Pharmaceuticals, Inc. |
Triazoles sustituidos con arilo policíclico y heteroarilo policíclico, útiles como agentes inhibidores del Axl
|
EA201001030A1
(ru)
|
2007-12-19 |
2011-02-28 |
Амген Инк. |
Конденсированные соединения пиридина, пиримидина и триазина в качестве ингибиторов клеточного цикла
|
AR070127A1
(es)
|
2008-01-11 |
2010-03-17 |
Novartis Ag |
Pirrolo - pirimidinas y pirrolo -piridinas
|
CN102131783A
(zh)
|
2008-04-16 |
2011-07-20 |
马克斯普朗克科学发展组织 |
作为axl激酶抑制剂的喹啉衍生物
|
CA2728729C
(en)
|
2008-06-23 |
2016-09-27 |
Vertex Pharmaceuticals Incorporated |
Protein kinase inhibitors
|
ES2537480T3
(es)
|
2008-07-09 |
2015-06-08 |
Rigel Pharmaceuticals, Inc. |
Triazoles sustituidos con heteroarilo policíclicos útiles como inhibidores de Axl
|
ES2399319T3
(es)
|
2008-07-09 |
2013-03-27 |
Rigel Pharmaceuticals, Inc. |
Triazoles sustituidos con heteroarilos bicíclicos que contienen puentes útiles como inhibidores de AXL
|
WO2010014755A1
(en)
|
2008-07-29 |
2010-02-04 |
The Regents Of The University Of Colorado |
Methods and compounds for enhancing anti-cancer therapy
|
US20100075973A1
(en)
|
2008-08-28 |
2010-03-25 |
Takeda Pharmaceutical Company Limited |
Polo-like kinase inhibitors
|
EP2376491B1
(en)
|
2008-12-19 |
2015-03-04 |
Cephalon, Inc. |
Pyrrolotriazines as alk and jak2 inhibitors
|
SG172857A1
(en)
|
2009-02-09 |
2011-08-29 |
Supergen Inc |
Pyrrolopyrimidinyl axl kinase inhibitors
|
US8765754B2
(en)
|
2009-04-29 |
2014-07-01 |
Locus Pharmaceuticals, Inc. |
Pyrrolotriazine compounds
|
EA025520B1
(ru)
|
2009-05-22 |
2017-01-30 |
Инсайт Холдингс Корпорейшн |
N-(ГЕТЕРО)АРИЛПИРРОЛИДИНОВЫЕ ПРОИЗВОДНЫЕ ПИРАЗОЛ-4-ИЛ-ПИРРОЛО[2,3-d]ПИРИМИДИНОВ И ПИРРОЛ-3-ИЛ-ПИРРОЛО[2,3-d]ПИРИМИДИНОВ В КАЧЕСТВЕ ИНГИБИТОРОВ ЯНУС-КИНАЗЫ
|
AR077280A1
(es)
|
2009-06-29 |
2011-08-17 |
Incyte Corp |
Pirimidinonas como inhibidores de pi3k, y composiciones farmaceuticas que los comprenden
|
TW201113285A
(en)
|
2009-09-01 |
2011-04-16 |
Incyte Corp |
Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
AU2010298190A1
(en)
|
2009-09-25 |
2012-05-03 |
Vertex Pharmaceuticals Incorporated |
Methods for preparing pyrimidine derivatives useful as protein kinase inhibitors
|
EP2311809A1
(en)
|
2009-10-16 |
2011-04-20 |
Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. |
Quinolinyloxyphenylsulfonamides
|
US8604217B2
(en)
|
2009-11-12 |
2013-12-10 |
Selvita S.A. |
Compound, a process for its preparation, a pharmaceutical composition, use of a compound, a method for modulating or regulating serine/threonine kinases and a serine/threonine kinases modulating agent
|
WO2011075630A1
(en)
|
2009-12-18 |
2011-06-23 |
Incyte Corporation |
Substituted fused aryl and heteroaryl derivatives as pi3k inhibitors
|
SI3354652T1
(sl)
|
2010-03-10 |
2020-08-31 |
Incyte Holdings Corporation |
Derivati piperidin-4-il azetidina kot inhibitorji JAK1
|
EP2552922A1
(en)
|
2010-03-31 |
2013-02-06 |
Bristol-Myers Squibb Company |
Substituted pyrrolotriazines as protein kinase inhibitors
|
CN102471342A
(zh)
|
2010-05-05 |
2012-05-23 |
沃泰克斯药物股份有限公司 |
用作PKC-θ抑制剂的4取代的吡唑并吡啶类
|
EP2423208A1
(en)
|
2010-08-28 |
2012-02-29 |
Lead Discovery Center GmbH |
Pharmaceutically active compounds as Axl inhibitors
|
EP2661268A2
(en)
|
2010-10-08 |
2013-11-13 |
Elan Pharmaceuticals Inc. |
Inhibitors of polo-like kinase
|
ITRM20100537A1
(it)
|
2010-10-12 |
2012-04-12 |
Consiglio Nazionale Ricerche |
Aptamero inibitore del recettore tirosina chinasi axl per uso in terapia
|
BR112013012502A2
(pt)
|
2010-11-19 |
2019-03-06 |
Incyte Corporation |
pirrolopiridina ciclobutil substituída e derivados de pirrolopirimidina derivativos como inibidores de jak
|
US9034884B2
(en)
|
2010-11-19 |
2015-05-19 |
Incyte Corporation |
Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as JAK inhibitors
|
TW201249844A
(en)
|
2010-12-20 |
2012-12-16 |
Incyte Corp |
N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
|
RU2568258C2
(ru)
|
2011-02-28 |
2015-11-20 |
Саншайн Лейк Фарма Ко., Лтд |
Замещенные соединения хинолина и способы их использования
|
DK2688887T3
(en)
|
2011-03-23 |
2015-06-29 |
Amgen Inc |
DEHYDRATED tricyclic DUALINHIBITORER OF CDK 4/6 AND FLT3
|
WO2012135800A1
(en)
|
2011-04-01 |
2012-10-04 |
University Of Utah Research Foundation |
Substituted n-phenylpyrimidin-2-amine analogs as inhibitors of the axl kinase
|
MY165963A
(en)
|
2011-06-20 |
2018-05-18 |
Incyte Holdings Corp |
Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors
|
AU2012280508A1
(en)
|
2011-07-01 |
2013-12-12 |
Bayer Intellectual Property Gmbh |
Hydroxymethylaryl-substituted pyrrolotriazines as ALK1 inhibitors
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
SI2751109T1
(sl)
|
2011-09-02 |
2017-03-31 |
Incyte Holdings Corporation |
Heterociklilamini kot inhibitorji pi3k
|
CN102408411B
(zh)
|
2011-09-19 |
2014-10-22 |
北京康辰药业股份有限公司 |
一种含喹啉基的羟肟酸类化合物及其制备方法、以及含有该化合物的药物组合物及其应用
|
CN103958510B
(zh)
|
2011-10-03 |
2016-10-19 |
北卡罗来纳大学教堂山分校 |
用于治疗癌症的吡咯并嘧啶化合物
|
SG10201510307WA
(en)
|
2011-11-14 |
2016-01-28 |
Cephalon Inc |
Uracil derivatives as axl and c-met kinase inhibitors
|
US8993756B2
(en)
|
2011-12-06 |
2015-03-31 |
Merck Sharp & Dohme Corp. |
Pyrrolopyrimidines as janus kinase inhibitors
|
PL2810937T3
(pl)
|
2012-01-31 |
2017-07-31 |
Daiichi Sankyo Company, Limited |
Pochodna pirydonu
|
WO2013162061A1
(ja)
|
2012-04-26 |
2013-10-31 |
第一三共株式会社 |
二環性ピリミジン化合物
|
US9193733B2
(en)
|
2012-05-18 |
2015-11-24 |
Incyte Holdings Corporation |
Piperidinylcyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors
|
JP6318156B2
(ja)
|
2012-09-06 |
2018-04-25 |
プレキシコン インコーポレーテッドPlexxikon Inc. |
キナーゼをモジュレートするための化合物および方法、ならびにその指標
|
BR112015006828A8
(pt)
|
2012-09-26 |
2019-09-17 |
Univ California |
composto, ou um sal farmaceuticamente aceitável do mesmo; composição farmacêutica; uso do composto; e método para modular a atividade de uma proteína ire1
|
US9562047B2
(en)
|
2012-10-17 |
2017-02-07 |
The University Of North Carolina At Chapel Hill |
Pyrazolopyrimidine compounds for the treatment of cancer
|
SG10201703533VA
(en)
|
2012-11-01 |
2017-06-29 |
Incyte Corp |
Tricyclic fused thiophene derivatives as jak inhibitors
|
JP6218848B2
(ja)
|
2012-11-20 |
2017-10-25 |
プロキナーゼ ゲゼルシャフト ミット ベシュレンクテル ハフツング |
プロテインキナーゼ阻害剤としてのチオエーテル誘導体
|
US20140199728A1
(en)
|
2013-01-14 |
2014-07-17 |
Amgen Inc. |
Methods of using cell-cycle inhibitors to modulate one or more properties of a cell culture
|
TW201522337A
(zh)
|
2013-03-12 |
2015-06-16 |
Arqule Inc |
經取代之三環吡唑並-嘧啶化合物類
|
TWI649308B
(zh)
|
2013-07-24 |
2019-02-01 |
小野藥品工業股份有限公司 |
喹啉衍生物
|
JP6493218B2
(ja)
|
2013-11-08 |
2019-04-03 |
小野薬品工業株式会社 |
ピロロピリミジン誘導体
|
EA201691302A1
(ru)
|
2014-02-03 |
2017-03-31 |
Кадила Хелзкэр Лимитед |
Новые гетероциклические соединения
|
ES2746839T3
(es)
|
2014-12-18 |
2020-03-09 |
Pfizer |
Derivados de pirimidina y triazina y su uso como inhibidores de AXL
|
US9840503B2
(en)
|
2015-05-11 |
2017-12-12 |
Incyte Corporation |
Heterocyclic compounds and uses thereof
|
WO2017027717A1
(en)
|
2015-08-12 |
2017-02-16 |
Incyte Corporation |
Bicyclic fused pyrimidine compounds as tam inhibitors
|
US10053465B2
(en)
|
2015-08-26 |
2018-08-21 |
Incyte Corporation |
Pyrrolopyrimidine derivatives as TAM inhibitors
|
US20180296561A1
(en)
|
2015-10-07 |
2018-10-18 |
The University Of North Carolina At Chapel Hill |
The Methods For Treatment Of Tumors
|
WO2017065183A1
(ja)
|
2015-10-13 |
2017-04-20 |
日本農薬株式会社 |
オキシム基を有する縮合複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法
|
EP3373932B1
(en)
|
2015-11-14 |
2022-03-30 |
Sunshine Lake Pharma Co., Ltd. |
Crystalline form of a substituted quinoline compound and pharmaceutical compositions thereof
|
US9695150B2
(en)
|
2015-11-14 |
2017-07-04 |
Calitor Sciences, Llc |
Crystalline form of a substituted quinoline compound and pharmaceutical compositions thereof
|
CA3019145A1
(en)
|
2016-03-28 |
2017-10-05 |
Incyte Corporation |
Pyrrolotriazine compounds as tam inhibitors
|
EP3445339B1
(en)
|
2016-04-22 |
2023-08-23 |
Incyte Corporation |
Formulations of an lsd1 inhibitor
|
WO2017223414A1
(en)
*
|
2016-06-24 |
2017-12-28 |
Incyte Corporation |
HETEROCYCLIC COMPOUNDS AS PI3K-γ INHIBITORS
|
JOP20170153A1
(ar)
|
2016-07-15 |
2019-01-30 |
Lilly Co Eli |
نظائر urocortin-2 جديدة معدلة بحمض دهني لعلاج داء السكري وأمراض الكلى المزمنة
|
LT3484524T
(lt)
|
2016-07-15 |
2022-12-27 |
Ionis Pharmaceuticals, Inc. |
Junginiai ir būdai, skirti smn2 moduliavimui
|
RS62872B1
(sr)
|
2017-09-27 |
2022-02-28 |
Incyte Corp |
Soli derivata pirrolotriazina korisne kao tam inhibitori
|
JP2021529765A
(ja)
|
2018-06-29 |
2021-11-04 |
インサイト・コーポレイションIncyte Corporation |
Axl/mer阻害剤の製剤
|