CY1111075T1 - Φαρμακευτικες συνθεσεις που περιεχουν τα παραγωγα της 3-αμινο-αζετιδινης, τα νεα παραγωγα τους και η προετοιμασια τους - Google Patents

Φαρμακευτικες συνθεσεις που περιεχουν τα παραγωγα της 3-αμινο-αζετιδινης, τα νεα παραγωγα τους και η προετοιμασια τους

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Publication number
CY1111075T1
CY1111075T1 CY20101100983T CY101100983T CY1111075T1 CY 1111075 T1 CY1111075 T1 CY 1111075T1 CY 20101100983 T CY20101100983 T CY 20101100983T CY 101100983 T CY101100983 T CY 101100983T CY 1111075 T1 CY1111075 T1 CY 1111075T1
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CY
Cyprus
Prior art keywords
products
preparation
azetidine
amino
denotes
Prior art date
Application number
CY20101100983T
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English (en)
Inventor
Daniel Achard
Hervé Bouchard
Jean Bouquerel
Bruno Filoche
Serge Grisoni
Augustin Hittinger
Michael Myers
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of CY1111075T1 publication Critical patent/CY1111075T1/el

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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Η παρούσα εφεύρεση αφορά τις φαρμακευτικές ενώσεις που περιέχουν ως δραστικό στοιχείο μια ένωση του τύπου (I) όπου το R1 δηλώνει μια ρίζα -NHCOR4 ή -N(R5)-Y-R6, το Υ είναι CO ή SO2, το R4 δηλώνει μια ρίζα -alk-SO2R11, -alk-SO2-CH=CH-R11, Het υποκαθιστούμενο από -SO2-R11 ή φαινύλιο υποκαθιστούμενο από -SO2-R11 ή -alk-SO2-R11, το R5 δηλώνει ένα άτομο υδρογόνου ή μια ρίζα αλκυλίου, το R6 δηλώνει μια ρίζα φαινυλαλκύλιου, Het ή Ar, τα νέα παράγωγα του τύπου (I) και την παρασκευή τους.
CY20101100983T 2000-03-03 2010-10-29 Φαρμακευτικες συνθεσεις που περιεχουν τα παραγωγα της 3-αμινο-αζετιδινης, τα νεα παραγωγα τους και η προετοιμασια τους CY1111075T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0002777A FR2805810B1 (fr) 2000-03-03 2000-03-03 Compositions pharmaceutiques contenant des derives de 3- amino-azetidine, les nouveaux derives et leur preparation
EP01909938A EP1263721B1 (fr) 2000-03-03 2001-03-01 Compositions pharmaceutiques contenant des derives de 3-amino-azetidine, les nouveaux derives et leur preparation

Publications (1)

Publication Number Publication Date
CY1111075T1 true CY1111075T1 (el) 2015-06-11

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CY20101100983T CY1111075T1 (el) 2000-03-03 2010-10-29 Φαρμακευτικες συνθεσεις που περιεχουν τα παραγωγα της 3-αμινο-αζετιδινης, τα νεα παραγωγα τους και η προετοιμασια τους

Country Status (35)

Country Link
EP (1) EP1263721B1 (el)
JP (1) JP2003525269A (el)
KR (1) KR100813740B1 (el)
CN (1) CN1187325C (el)
AR (1) AR034405A1 (el)
AT (1) ATE478840T1 (el)
AU (2) AU3752601A (el)
BG (1) BG107057A (el)
BR (1) BR0108894A (el)
CA (1) CA2400138A1 (el)
CY (1) CY1111075T1 (el)
DE (1) DE60142890D1 (el)
DK (1) DK1263721T3 (el)
DZ (1) DZ3311A1 (el)
EA (1) EA004649B1 (el)
EE (1) EE05081B1 (el)
ES (1) ES2351183T3 (el)
FR (1) FR2805810B1 (el)
HR (1) HRP20020710A2 (el)
HU (1) HUP0300350A2 (el)
IL (2) IL151209A0 (el)
MA (1) MA26879A1 (el)
MX (1) MXPA02008346A (el)
NO (1) NO324523B1 (el)
NZ (1) NZ521076A (el)
OA (1) OA12221A (el)
PL (1) PL365007A1 (el)
PT (1) PT1263721E (el)
SI (1) SI1263721T1 (el)
SK (1) SK12442002A3 (el)
TW (1) TWI294420B (el)
UA (1) UA72319C2 (el)
WO (1) WO2001064633A1 (el)
YU (1) YU65902A (el)
ZA (1) ZA200206916B (el)

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NO324523B1 (no) 2007-11-12
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EE200200486A (et) 2004-02-16
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