CS212220B2 - Method of making the 3,3-ethylendioxy-4,5-seko-19-norandrost-9-en-5, 17-dione - Google Patents

Method of making the 3,3-ethylendioxy-4,5-seko-19-norandrost-9-en-5, 17-dione Download PDF

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Publication number
CS212220B2
CS212220B2 CS794117A CS411779A CS212220B2 CS 212220 B2 CS212220 B2 CS 212220B2 CS 794117 A CS794117 A CS 794117A CS 411779 A CS411779 A CS 411779A CS 212220 B2 CS212220 B2 CS 212220B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
compound
chem
mixed anhydride
grignard reagent
Prior art date
Application number
CS794117A
Other languages
Czech (cs)
English (en)
Inventor
Gary F Cooper
Horn Albert R Van
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of CS212220B2 publication Critical patent/CS212220B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/26Radicals substituted by doubly bound oxygen or sulfur atoms or by two such atoms singly bound to the same carbon atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/54Preparation of carboxylic acid anhydrides
    • C07C51/56Preparation of carboxylic acid anhydrides from organic acids, their salts, their esters or their halides, e.g. by carboxylation

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CS794117A 1978-06-19 1979-06-14 Method of making the 3,3-ethylendioxy-4,5-seko-19-norandrost-9-en-5, 17-dione CS212220B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/916,443 US4158012A (en) 1978-06-19 1978-06-19 Steroid synthesis process using mixed anhydride

Publications (1)

Publication Number Publication Date
CS212220B2 true CS212220B2 (en) 1982-03-26

Family

ID=25437272

Family Applications (2)

Application Number Title Priority Date Filing Date
CS794117A CS212220B2 (en) 1978-06-19 1979-06-14 Method of making the 3,3-ethylendioxy-4,5-seko-19-norandrost-9-en-5, 17-dione
CS794430A CS212221B2 (en) 1978-06-19 1979-06-14 Method of making the (+) 3a, 7a-trans-4-/7,7-/ethylenedioxy /-oxooktyl/-7a beta-methylperhydroindane-1,5-dion

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS794430A CS212221B2 (en) 1978-06-19 1979-06-14 Method of making the (+) 3a, 7a-trans-4-/7,7-/ethylenedioxy /-oxooktyl/-7a beta-methylperhydroindane-1,5-dion

Country Status (16)

Country Link
US (1) US4158012A (de)
EP (1) EP0006355B1 (de)
JP (3) JPS552675A (de)
AT (1) ATE7600T1 (de)
CS (2) CS212220B2 (de)
DD (1) DD144269A5 (de)
DE (1) DE2967004D1 (de)
DK (2) DK246479A (de)
ES (1) ES481650A1 (de)
HK (1) HK96787A (de)
HU (2) HU186974B (de)
MY (1) MY8700665A (de)
PL (2) PL123780B1 (de)
SG (1) SG38287G (de)
SU (1) SU999977A3 (de)
YU (1) YU41160B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4400524A (en) * 1981-07-28 1983-08-23 The Upjohn Company Grignard reagents prepared from 5-halopentan-2-one propylene ketals
JPS58134577A (ja) * 1982-02-05 1983-08-10 Nippon Kogaku Kk <Nikon> 電気光学的光制御素子
NL8602767A (nl) * 1986-10-31 1988-05-16 Gantax Nv Organisch zuuranhydride, alsmede farmaceutisch preparaat op basis van een prodrug.
CA2243402A1 (en) * 1997-07-22 1999-01-22 Hideo Suwa Process for producing maleic anhydride
JP4822548B2 (ja) * 2007-04-23 2011-11-24 レーザーテック株式会社 欠陥検査装置
CN109293723A (zh) * 2018-09-21 2019-02-01 山东斯瑞生物医药有限公司 雌甾-4,9-二烯-3,17-二酮的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1255101A (fr) * 1960-01-22 1961-03-03 Chimiotherapie Lab Franc Procédé d'alcoylation d'intermédiaires de la synthèse de 10-alcoyl 19-nor stéroïdes
US3117979A (en) * 1960-01-22 1964-01-14 Roussel Uclaf Esters of 10beta-substituted 4, 5-seco-delta9(11)-19-nor-androstene-17beta-ol-3, 5-dines, intermediates and process
NL126395C (de) * 1962-03-06
NL130550C (de) * 1966-05-26
US3984473A (en) * 1968-10-04 1976-10-05 Hoffmann-La Roche Inc. Stereospecific total steroidal synthesis via substituted C/D-trans indanones
US3686215A (en) * 1969-03-27 1972-08-22 Syntex Corp Production of 5,6,7,7a-tetrahydroindan-5-ones
SE367181B (de) * 1969-05-14 1974-05-20 Takeda Chemical Industries Ltd
US3813417A (en) * 1970-08-26 1974-05-28 Hoffmann La Roche Cycloalkyl(f)(l)benzopyrans
DE2228474A1 (de) * 1972-06-08 1973-12-20 Schering Ag Neue bicycloalkan-derivate

Also Published As

Publication number Publication date
PL216413A1 (de) 1980-03-24
JPH0129792B2 (de) 1989-06-14
MY8700665A (en) 1987-12-31
HU186974B (en) 1985-10-28
DK129491A (da) 1991-07-02
JPS6425772A (en) 1989-01-27
EP0006355B1 (de) 1984-05-23
YU142779A (en) 1983-02-28
DE2967004D1 (en) 1984-06-28
DK246479A (da) 1979-12-20
CS212221B2 (en) 1982-03-26
JPS6425747A (en) 1989-01-27
SG38287G (en) 1987-07-24
JPH0316333B2 (de) 1991-03-05
DK129491D0 (da) 1991-07-02
SU999977A3 (ru) 1983-02-23
EP0006355A1 (de) 1980-01-09
HK96787A (en) 1987-12-24
DD144269A5 (de) 1980-10-08
JPS645034B2 (de) 1989-01-27
US4158012A (en) 1979-06-12
HU181503B (en) 1983-10-28
PL118827B1 (en) 1981-10-31
PL123780B1 (en) 1982-11-30
ATE7600T1 (de) 1984-06-15
ES481650A1 (es) 1980-04-16
JPS552675A (en) 1980-01-10
YU41160B (en) 1986-12-31

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