CO5070579A1 - Formulaciones de ziprasidona - Google Patents

Formulaciones de ziprasidona

Info

Publication number
CO5070579A1
CO5070579A1 CO99037319A CO99037319A CO5070579A1 CO 5070579 A1 CO5070579 A1 CO 5070579A1 CO 99037319 A CO99037319 A CO 99037319A CO 99037319 A CO99037319 A CO 99037319A CO 5070579 A1 CO5070579 A1 CO 5070579A1
Authority
CO
Colombia
Prior art keywords
ziprasidona
formulations
crystalline ziprasidone
mfi
schizophrenia
Prior art date
Application number
CO99037319A
Other languages
English (en)
Inventor
Frank Robert Busch
Hausberger Angela Carol Gatlin
Rasadi Bijan
Arenson Daniel Ray
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22216447&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5070579(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of CO5070579A1 publication Critical patent/CO5070579A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • A61K9/1688Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Feeding Of Articles By Means Other Than Belts Or Rollers (AREA)
  • Polyamides (AREA)
  • Detergent Compositions (AREA)

Abstract

Composiciones que comprenden partículas de base libre de ziprasidona cristalina o de hidrocloruro de ziprasidona cristalino, que tienen un tamaño medio de partículas inferior a 85 (m, y un vehículo farmacéuticamente aceptable son sustancialmente bioequivalentes y se pueden usar para tratar psicosis, como esquizofrenia. <EMI FILE="99037319_1" ID="1" IMF=JPEG >
CO99037319A 1998-06-15 1999-06-15 Formulaciones de ziprasidona CO5070579A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8922998P 1998-06-15 1998-06-15

Publications (1)

Publication Number Publication Date
CO5070579A1 true CO5070579A1 (es) 2001-08-28

Family

ID=22216447

Family Applications (1)

Application Number Title Priority Date Filing Date
CO99037319A CO5070579A1 (es) 1998-06-15 1999-06-15 Formulaciones de ziprasidona

Country Status (45)

Country Link
US (1) US6150366A (es)
EP (1) EP0965343B1 (es)
JP (2) JP3441676B2 (es)
KR (1) KR100338915B1 (es)
CN (1) CN1307994C (es)
AP (1) AP1216A (es)
AR (1) AR015553A1 (es)
AT (1) ATE240732T1 (es)
AU (1) AU753820B2 (es)
BG (1) BG64691B1 (es)
BR (1) BR9902268A (es)
CA (1) CA2274338C (es)
CO (1) CO5070579A1 (es)
CY (1) CY2003002I1 (es)
CZ (1) CZ297954B6 (es)
DE (1) DE69908021T2 (es)
DK (1) DK0965343T3 (es)
EA (1) EA002223B1 (es)
ES (1) ES2197581T3 (es)
GT (1) GT199900080A (es)
HK (1) HK1024184A1 (es)
HN (1) HN1999000089A (es)
HR (1) HRP990193B1 (es)
HU (1) HU226487B1 (es)
ID (1) ID23546A (es)
IL (1) IL130424A (es)
IS (1) IS2182B (es)
MA (1) MA26647A1 (es)
MY (1) MY121397A (es)
NO (1) NO316713B1 (es)
NZ (1) NZ336271A (es)
OA (1) OA11064A (es)
PA (1) PA8475601A1 (es)
PE (1) PE20000632A1 (es)
PL (2) PL195209B1 (es)
PT (1) PT965343E (es)
RS (1) RS49611B (es)
SG (1) SG77243A1 (es)
SI (1) SI0965343T1 (es)
SK (1) SK286245B6 (es)
TR (1) TR199901379A2 (es)
TW (1) TW590774B (es)
UA (1) UA59383C2 (es)
UY (1) UY25649A1 (es)
ZA (1) ZA993938B (es)

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Also Published As

Publication number Publication date
KR100338915B1 (ko) 2002-05-30
US6150366A (en) 2000-11-21
OA11064A (en) 2002-03-13
CZ212799A3 (cs) 2000-09-13
PL333737A1 (en) 1999-12-20
PE20000632A1 (es) 2000-07-26
IL130424A (en) 2003-10-31
DE69908021D1 (de) 2003-06-26
AP1216A (en) 2003-10-19
EA199900467A3 (ru) 2000-04-24
HRP990193B1 (en) 2003-08-31
RS49611B (sr) 2007-06-04
EA199900467A2 (ru) 1999-12-29
MA26647A1 (fr) 2004-12-20
NO316713B1 (no) 2004-04-13
SK76999A3 (en) 2000-12-11
AU3398399A (en) 1999-12-23
TW590774B (en) 2004-06-11
PL195209B1 (pl) 2007-08-31
SK286245B6 (sk) 2008-06-06
JP4187423B2 (ja) 2008-11-26
HUP9901960A3 (en) 2000-09-28
HK1024184A1 (en) 2000-10-05
IS5079A (is) 1999-12-16
IL130424A0 (en) 2000-06-01
SI0965343T1 (en) 2003-10-31
AP9901579A0 (en) 1999-06-30
DK0965343T3 (da) 2003-08-04
AU753820B2 (en) 2002-10-31
HUP9901960A2 (hu) 2000-08-28
EA002223B1 (ru) 2002-02-28
IS2182B (is) 2006-12-15
HU226487B1 (en) 2009-03-02
JP2000007566A (ja) 2000-01-11
BG64691B1 (bg) 2005-12-30
CN1307994C (zh) 2007-04-04
HU9901960D0 (en) 1999-08-30
ES2197581T3 (es) 2004-01-01
EP0965343B1 (en) 2003-05-21
ID23546A (id) 2000-05-04
YU27199A (sh) 2002-12-10
HN1999000089A (es) 1999-11-03
CY2003002I1 (el) 2009-11-04
PT965343E (pt) 2003-08-29
SG77243A1 (en) 2000-12-19
JP3441676B2 (ja) 2003-09-02
BG103489A (en) 2000-07-31
HRP990193A2 (en) 2000-02-29
KR20000006143A (ko) 2000-01-25
UA59383C2 (uk) 2003-09-15
AR015553A1 (es) 2001-05-02
GT199900080A (es) 2000-11-29
BR9902268A (pt) 2000-05-02
CA2274338C (en) 2003-04-15
CZ297954B6 (cs) 2007-05-09
CA2274338A1 (en) 1999-12-15
ZA993938B (en) 2000-12-14
EP0965343A2 (en) 1999-12-22
JP2002003492A (ja) 2002-01-09
EP0965343A3 (en) 2000-02-23
NZ336271A (en) 2000-10-27
NO992892D0 (no) 1999-06-14
TR199901379A2 (xx) 2000-01-21
DE69908021T2 (de) 2003-11-27
UY25649A1 (es) 2000-02-23
ATE240732T1 (de) 2003-06-15
CN1242987A (zh) 2000-02-02
PA8475601A1 (es) 2000-09-29
MY121397A (en) 2006-01-28
PL195606B1 (pl) 2007-10-31
NO992892L (no) 1999-12-16

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