CO2018008707A2 - Inhibidores de la proteína quinasa 1 que interactúa con el receptor - Google Patents

Inhibidores de la proteína quinasa 1 que interactúa con el receptor

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Publication number
CO2018008707A2
CO2018008707A2 CONC2018/0008707A CO2018008707A CO2018008707A2 CO 2018008707 A2 CO2018008707 A2 CO 2018008707A2 CO 2018008707 A CO2018008707 A CO 2018008707A CO 2018008707 A2 CO2018008707 A2 CO 2018008707A2
Authority
CO
Colombia
Prior art keywords
inhibitors
interacts
receptor
protein kinase
compositions
Prior art date
Application number
CONC2018/0008707A
Other languages
English (en)
Inventor
Joseph P Lyssikatos
Zachary K Sweeney
Anthony A Estrada
Jianwen A Feng
Brian Fox
Colin Philip Leslie
Alfonso Pozzan
Vicente Fidalgo Javier De
Original Assignee
Denali Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Denali Therapeutics Inc filed Critical Denali Therapeutics Inc
Publication of CO2018008707A2 publication Critical patent/CO2018008707A2/es

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    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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Abstract

La presente descripción se refiere en general a compuestos y composiciones y a su uso como inhibidores de quinasa.
CONC2018/0008707A 2016-02-05 2018-08-21 Inhibidores de la proteína quinasa 1 que interactúa con el receptor CO2018008707A2 (es)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US201662292202P 2016-02-05 2016-02-05
US201662341019P 2016-05-24 2016-05-24
US201662363775P 2016-07-18 2016-07-18
US201662385217P 2016-09-08 2016-09-08
US201662417219P 2016-11-03 2016-11-03
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