CL2014002472A1 - Uso de (rs)-s-ciclopropil-s-(4-{[4-{[(1r, 2r)-2-hidroxi-1-metilpropil]oxi}-5-(trifluorometil)pirimidin-2-il] amino}fenil) sulfoximida para el tratamiento de cancer de tiroides, mesoteliomas, carcinomas de celulas escamosas del esofago o carcinomas colangiocelulares; composicion farmaceutica; combinacion farmaceutica. - Google Patents

Uso de (rs)-s-ciclopropil-s-(4-{[4-{[(1r, 2r)-2-hidroxi-1-metilpropil]oxi}-5-(trifluorometil)pirimidin-2-il] amino}fenil) sulfoximida para el tratamiento de cancer de tiroides, mesoteliomas, carcinomas de celulas escamosas del esofago o carcinomas colangiocelulares; composicion farmaceutica; combinacion farmaceutica.

Info

Publication number
CL2014002472A1
CL2014002472A1 CL2014002472A CL2014002472A CL2014002472A1 CL 2014002472 A1 CL2014002472 A1 CL 2014002472A1 CL 2014002472 A CL2014002472 A CL 2014002472A CL 2014002472 A CL2014002472 A CL 2014002472A CL 2014002472 A1 CL2014002472 A1 CL 2014002472A1
Authority
CL
Chile
Prior art keywords
carcinomas
sulfoximide
mesotheliomas
methylpropyl
pyrimidin
Prior art date
Application number
CL2014002472A
Other languages
English (en)
Inventor
Kornacker Martin Dr
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47891732&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2014002472(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of CL2014002472A1 publication Critical patent/CL2014002472A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CL2014002472A 2012-03-21 2014-09-17 Uso de (rs)-s-ciclopropil-s-(4-{[4-{[(1r, 2r)-2-hidroxi-1-metilpropil]oxi}-5-(trifluorometil)pirimidin-2-il] amino}fenil) sulfoximida para el tratamiento de cancer de tiroides, mesoteliomas, carcinomas de celulas escamosas del esofago o carcinomas colangiocelulares; composicion farmaceutica; combinacion farmaceutica. CL2014002472A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102012204506 2012-03-21

Publications (1)

Publication Number Publication Date
CL2014002472A1 true CL2014002472A1 (es) 2014-12-12

Family

ID=47891732

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2014002472A CL2014002472A1 (es) 2012-03-21 2014-09-17 Uso de (rs)-s-ciclopropil-s-(4-{[4-{[(1r, 2r)-2-hidroxi-1-metilpropil]oxi}-5-(trifluorometil)pirimidin-2-il] amino}fenil) sulfoximida para el tratamiento de cancer de tiroides, mesoteliomas, carcinomas de celulas escamosas del esofago o carcinomas colangiocelulares; composicion farmaceutica; combinacion farmaceutica.

Country Status (20)

Country Link
US (1) US20150051232A1 (es)
EP (1) EP2827871A1 (es)
JP (1) JP2015510910A (es)
KR (1) KR20140135215A (es)
CN (1) CN104220075A (es)
AP (1) AP2014007915A0 (es)
AU (1) AU2013234451A1 (es)
CA (1) CA2867746A1 (es)
CL (1) CL2014002472A1 (es)
EA (1) EA201491732A1 (es)
HK (1) HK1204294A1 (es)
MA (1) MA35943B1 (es)
MX (1) MX2014011240A (es)
PH (1) PH12014502075A1 (es)
SA (1) SA113340398B1 (es)
SG (1) SG11201405386SA (es)
TN (1) TN2014000391A1 (es)
TW (1) TW201338779A (es)
WO (1) WO2013139734A1 (es)
ZA (1) ZA201406986B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015071231A1 (de) * 2013-11-14 2015-05-21 Bayer Pharma Aktiengesellschaft Kombinationen von (rs)-s-cyclopropyl-s-(4-{[4-{[(1r, 2r)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluormethyl)pyrimidin-2-yl]amino}phenyl)sulfoximid zur behandlung von tumoren
ES2951596T3 (es) 2014-06-13 2023-10-23 Bach Biosciences Llc Agentes terapéuticos activados por FAP y usos relacionados con los mismos

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1307271A (en) 1970-06-25 1973-02-14 Shell Int Research Sulphoximine derivatives and their use in herbicidal compositions
DE4029650A1 (de) 1990-09-19 1992-03-26 Hoechst Ag 2-anilino-pyrimidine, verfahren zu ihrer herstellung, sie enthaltene mittel und ihre verwendung als fungizide
EP1017394B1 (en) 1997-07-12 2005-12-07 Cancer Research Technology Limited Cyclin dependent kinase inhibiting purine derivatives
US6440965B1 (en) 1997-10-15 2002-08-27 Krenitsky Pharmaceuticals, Inc. Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system
ATE336484T1 (de) 1998-08-29 2006-09-15 Astrazeneca Ab Pyrimidine verbindungen
GB9828511D0 (en) 1998-12-24 1999-02-17 Zeneca Ltd Chemical compounds
JP4771576B2 (ja) * 2000-06-12 2011-09-14 譲治 稲澤 Gasc1遺伝子
GB0016877D0 (en) 2000-07-11 2000-08-30 Astrazeneca Ab Chemical compounds
EP1392662B1 (de) 2001-05-29 2009-01-07 Bayer Schering Pharma Aktiengesellschaft Cdk inhibitorische pyrimidine, deren herstellung und verwendung als arzneimittel
EP1483260A1 (de) 2002-03-11 2004-12-08 Schering Aktiengesellschaft Cdk inhibitorische 2-heteroaryl-pyrimidine, deren herstellung und verwendung als arzneimittel
WO2004041267A1 (en) * 2002-11-06 2004-05-21 Cyclacel Limited Combination comprising a cdk inhibitor and cisplatin
DE10349423A1 (de) 2003-10-16 2005-06-16 Schering Ag Sulfoximinsubstituierte Parimidine als CDK- und/oder VEGF-Inhibitoren, deren Herstellung und Verwendung als Arzneimittel
EP2179991A1 (de) * 2008-10-21 2010-04-28 Bayer Schering Pharma Aktiengesellschaft Sulfoximinsubstituierte Anilino-Pyrimidinderivate als CDK-Inhibitoren, deren Herstellung und Verwendung als Arzneimittel
CN102223885B (zh) * 2008-11-24 2013-04-03 内尔维阿诺医学科学有限公司 用于治疗间皮瘤的cdk抑制剂
EP2424843B1 (en) * 2009-04-30 2014-03-26 Novartis AG Imidazole derivatives and their use as modulators of cyclin dependent kinases
DE102010014426A1 (de) * 2010-04-01 2011-10-06 Bayer Schering Pharma Aktiengesellschaft Verwendung neuer pan-CDK-Inhibitoren zur Behandlung von Tumoren
DE102010014427A1 (de) 2010-04-01 2011-10-06 Bayer Schering Pharma Aktiengesellschaft Kombinationen neuer pan-CDK-Inhibitoren zur Behandlung von Tumoren

Also Published As

Publication number Publication date
ZA201406986B (en) 2016-08-31
AU2013234451A1 (en) 2014-09-25
TN2014000391A1 (en) 2015-12-21
AP2014007915A0 (en) 2014-09-30
CN104220075A (zh) 2014-12-17
MA35943B1 (fr) 2014-12-01
EA201491732A1 (ru) 2015-08-31
MX2014011240A (es) 2014-10-15
SA113340398B1 (ar) 2016-04-04
CA2867746A1 (en) 2013-09-26
JP2015510910A (ja) 2015-04-13
TW201338779A (zh) 2013-10-01
KR20140135215A (ko) 2014-11-25
WO2013139734A1 (de) 2013-09-26
SG11201405386SA (en) 2014-11-27
PH12014502075A1 (en) 2014-12-10
US20150051232A1 (en) 2015-02-19
EP2827871A1 (de) 2015-01-28
HK1204294A1 (en) 2015-11-13

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