BR0010693A - Derivados azaindol para tratamento de depressão - Google Patents
Derivados azaindol para tratamento de depressãoInfo
- Publication number
- BR0010693A BR0010693A BR0010693-3A BR0010693A BR0010693A BR 0010693 A BR0010693 A BR 0010693A BR 0010693 A BR0010693 A BR 0010693A BR 0010693 A BR0010693 A BR 0010693A
- Authority
- BR
- Brazil
- Prior art keywords
- treating depression
- azaindole derivatives
- depression
- affected
- ring
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Abstract
Patente de Invenção: "DERIVADOS AZAINDOL PARA TRATAMENTO DE DEPRESSãO". Compostos úteis no tratamento de doenças afetadas por desordens dos sistemas neurológicos afetados - serotonina, tais como depressão e ansiedade, são providos tendo a fórmula (1) onde: R~ 1~ e R~ 2~ formam um anel carbocíclico ou heterocíclico de 5 a 7 átomos, onde o dito anel pode ser saturado ou insaturado; e X é independentemente hidrogênio, ciano, carbamoíla, halogênio ou alcóxi; ou seus sais farmaceuticamente aceitáveis.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US29673699A | 1999-04-22 | 1999-04-22 | |
PCT/US2000/010628 WO2000064898A1 (en) | 1999-04-22 | 2000-04-20 | Azaindole derivatives for the treatment of depression |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0010693A true BR0010693A (pt) | 2002-02-05 |
Family
ID=23143341
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0010693-3A BR0010693A (pt) | 1999-04-22 | 2000-04-20 | Derivados azaindol para tratamento de depressão |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1171439A1 (pt) |
JP (1) | JP2002543079A (pt) |
CN (1) | CN1348451A (pt) |
AR (1) | AR028475A1 (pt) |
AU (1) | AU4364400A (pt) |
BR (1) | BR0010693A (pt) |
CA (1) | CA2367681A1 (pt) |
WO (1) | WO2000064898A1 (pt) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2003082869A1 (en) * | 2002-03-28 | 2003-10-09 | Eisai Co., Ltd. | Azaindoles as inhibitors of c-jun n-terminal kinases |
DE602005016836D1 (de) | 2004-11-26 | 2009-11-05 | Janssen Pharmaceutica Nv | Chotischer und anxiolytischer aktivität |
WO2008063888A2 (en) | 2006-11-22 | 2008-05-29 | Plexxikon, Inc. | Compounds modulating c-fms and/or c-kit activity and uses therefor |
EP2170830B1 (en) | 2007-07-17 | 2014-10-15 | Plexxikon, Inc. | 2-FLUORO-BENZENESULFONAMIDE COMPOUNDS AS Raf KINASE MODULATORS |
MY172424A (en) | 2009-04-03 | 2019-11-25 | Hoffmann La Roche | Propane- i-sulfonic acid {3- (4-chloro-phenyl)-1h-pyrrolo [2, 3-b] pyridine-3-carconyl] -2, 4-difluoro-phenyl} -amide compositions and uses thereof |
PE20120508A1 (es) | 2009-06-17 | 2012-05-09 | Vertex Pharma | Inhibidores de la replicacion de los virus de la gripe |
BR112012012156A2 (pt) | 2009-11-06 | 2015-09-08 | Plexxikon Inc | compostos e métodos para modulação de cinase, e indicações para esta |
CN103492381A (zh) | 2010-12-16 | 2014-01-01 | 沃泰克斯药物股份有限公司 | 流感病毒复制的抑制剂 |
TR201816421T4 (tr) | 2011-02-07 | 2018-11-21 | Plexxikon Inc | Kinaz modülasyonu için bileşikler ve metotlar ve bunların endikasyonları. |
AR085279A1 (es) | 2011-02-21 | 2013-09-18 | Plexxikon Inc | Formas solidas de {3-[5-(4-cloro-fenil)-1h-pirrolo[2,3-b]piridina-3-carbonil]-2,4-difluor-fenil}-amida del acido propano-1-sulfonico |
UA118010C2 (uk) | 2011-08-01 | 2018-11-12 | Вертекс Фармасьютікалз Інкорпорейтед | Інгібітори реплікації вірусів грипу |
US9150570B2 (en) | 2012-05-31 | 2015-10-06 | Plexxikon Inc. | Synthesis of heterocyclic compounds |
EP3068776B1 (en) | 2013-11-13 | 2019-05-29 | Vertex Pharmaceuticals Incorporated | Inhibitors of influenza viruses replication |
SG10201804021TA (en) | 2013-11-13 | 2018-07-30 | Vertex Pharma | Methods of preparing inhibitors of influenza viruses replication |
JP6857617B2 (ja) | 2015-05-13 | 2021-04-14 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | インフルエンザウイルスの複製の阻害剤 |
WO2016183116A1 (en) | 2015-05-13 | 2016-11-17 | Vertex Pharmaceuticals Incorporated | Methods of preparing inhibitors of influenza viruses replication |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5521197A (en) * | 1994-12-01 | 1996-05-28 | Eli Lilly And Company | 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists |
US5576321A (en) * | 1995-01-17 | 1996-11-19 | Eli Lilly And Company | Compounds having effects on serotonin-related systems |
US5627196A (en) * | 1995-01-17 | 1997-05-06 | Eli Lilly And Company | Compounds having effects on serotonin-related systems |
-
2000
- 2000-04-19 AR ARP000101879A patent/AR028475A1/es unknown
- 2000-04-20 WO PCT/US2000/010628 patent/WO2000064898A1/en not_active Application Discontinuation
- 2000-04-20 CN CN00806589A patent/CN1348451A/zh active Pending
- 2000-04-20 CA CA002367681A patent/CA2367681A1/en not_active Abandoned
- 2000-04-20 JP JP2000614250A patent/JP2002543079A/ja active Pending
- 2000-04-20 EP EP00923540A patent/EP1171439A1/en not_active Withdrawn
- 2000-04-20 AU AU43644/00A patent/AU4364400A/en not_active Abandoned
- 2000-04-20 BR BR0010693-3A patent/BR0010693A/pt not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JP2002543079A (ja) | 2002-12-17 |
AR028475A1 (es) | 2003-05-14 |
AU4364400A (en) | 2000-11-10 |
CN1348451A (zh) | 2002-05-08 |
CA2367681A1 (en) | 2000-11-02 |
EP1171439A1 (en) | 2002-01-16 |
WO2000064898A1 (en) | 2000-11-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR0010693A (pt) | Derivados azaindol para tratamento de depressão | |
ATE370138T1 (de) | Neue imidazopyridine und ihre verwendung | |
BRPI0314308B8 (pt) | antagonistas de opióide, seus usos, e composição farmacêutica | |
BR0108610A (pt) | Compostos azapolicìclicos condensados com arila | |
TR200201505T2 (tr) | Terapötik maddeler olarak pirazolopirimidinler | |
BR0113448A (pt) | Composto da fórmula ou um sal ou solvato deste ou um derivado destes fisiologicamente funcional, composição farmacêutica, uso do composto ou de um sal ou solvato deste ou de um derivado destes fisiologicamente funcional, e , métodos para tratar uma condição ou estado de doença mediados pela p38 quinase ou mediados pelas citoquinas, e mediados pela jnk quinase ou mediados pelas citoquinas, e ,para tratar duas ou mais condições ou doenças independentemente mediadas pela atividade da p38 e da jnk quinase | |
ES2161418T3 (es) | Compuestos de piridilfurano y de piridiltiofeno y uso farmaceutico de los mismos. | |
MXPA04012965A (es) | Inhibidores virales. | |
BR0311541A (pt) | indol, azaindol e 4-aquenil piperidina amidas heterocìclicas relacionadas | |
DE69911448D1 (de) | Pyrazolopyrimidinone, cgmp pde5 inhibitoren, zur behandlung von sexuellen funktionsstörungen | |
BR0312232A (pt) | Inibidores de caspases e seus usos | |
ES2158778B1 (es) | Compuestos de sales de paroxetina, su preparacion y uso, y composiciones farmaceuticas que los contienen. | |
NO20072046L (no) | Halogensubstituerte benzodiazepinderivater | |
BR9914040A (pt) | Derivados de [1,2,4]triazolo[1,5-c]pirimidina e seu uso, medicamento, antagonista, agente para prevenir ou tratar doenças, bem como processo para prevenção ou tratamento de distúrbios | |
DE60305514D1 (de) | Neue verwendung von benzothiazolderivaten | |
NO990433L (no) | Nye forbindelser og blandinger for behandling av sykdommer i forbindelse med tryptase-aktivitet | |
BR0315777A (pt) | Uso de derivados de piperazina como antagonistas ccr1 | |
ATE242246T1 (de) | (1,2,3)-triazolo(4,5-d)pyrimidin-derivate als antithrombotische mittel | |
WO2002079169A8 (en) | Cyano-substituted dihydropyrimidine compounds and their use to treat diseases | |
BR9807950A (pt) | Composto, composição farmacêutica, uso de um composto, e, processos para tratar ou reduzir o risco de doenças ou condições humanas, o risco de doença inflamatória o risco da dor e para a preparação de um composto | |
WO2002079149A3 (en) | Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases | |
MXPA01007940A (es) | Derivados de azabicicloalcano y usos terapeuticos de los mismos. | |
BR0213417A (pt) | Compostos e composições de tetraciclicazaindóis e indolinas tendo atividade de 5-ht e seus usos | |
BR0213037A (pt) | Derivados de pirimidina | |
ATE482211T1 (de) | Imidazoä1,2-aüpyridin-anxiolytika |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA10 | Dismissal: dismissal - article 33 of industrial property law | ||
B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired | ||
B25D | Requested change of name of applicant approved |