BG32116A3 - Метод за получаване на 4''-амино-олеандомицинови производни - Google Patents

Метод за получаване на 4''-амино-олеандомицинови производни

Info

Publication number
BG32116A3
BG32116A3 BG038401A BG3840178A BG32116A3 BG 32116 A3 BG32116 A3 BG 32116A3 BG 038401 A BG038401 A BG 038401A BG 3840178 A BG3840178 A BG 3840178A BG 32116 A3 BG32116 A3 BG 32116A3
Authority
BG
Bulgaria
Prior art keywords
amino
derivatives
oleandomicine
obtaining
proven
Prior art date
Application number
BG038401A
Other languages
English (en)
Inventor
Frank Sciavolino
Original Assignee
Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware filed Critical Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware
Publication of BG32116A3 publication Critical patent/BG32116A3/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Метод за получаване на охарактеризирани и доказани в описанието 4''-амино-олеандомицинови производни с формула...................... Патентните претенции са формулирани в 5 точки
BG038401A 1977-02-04 1978-01-16 Метод за получаване на 4''-амино-олеандомицинови производни BG32116A3 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/765,486 US4125705A (en) 1977-02-04 1977-02-04 Semi-synthetic 4-amino-oleandomycin derivatives

Publications (1)

Publication Number Publication Date
BG32116A3 true BG32116A3 (bg) 1982-05-14

Family

ID=25073683

Family Applications (2)

Application Number Title Priority Date Filing Date
BG040058A BG32117A4 (bg) 1977-02-04 1978-01-16 Метод за получаване олеандомицини
BG038401A BG32116A3 (bg) 1977-02-04 1978-01-16 Метод за получаване на 4''-амино-олеандомицинови производни

Family Applications Before (1)

Application Number Title Priority Date Filing Date
BG040058A BG32117A4 (bg) 1977-02-04 1978-01-16 Метод за получаване олеандомицини

Country Status (34)

Country Link
US (1) US4125705A (bg)
JP (2) JPS5398981A (bg)
AR (1) AR215666A1 (bg)
AT (1) AT358169B (bg)
AU (1) AU502293B1 (bg)
BE (1) BE863618A (bg)
BG (2) BG32117A4 (bg)
CA (1) CA1106366A (bg)
CH (1) CH629821A5 (bg)
CS (3) CS200537B2 (bg)
DD (1) DD134523A5 (bg)
DE (1) DE2804509C2 (bg)
DK (1) DK149628C (bg)
ES (1) ES465322A1 (bg)
FI (1) FI65262C (bg)
FR (2) FR2383964A1 (bg)
GB (1) GB1583921A (bg)
GR (1) GR68692B (bg)
HU (2) HU181395B (bg)
IE (1) IE46395B1 (bg)
IL (2) IL53959A0 (bg)
IT (1) IT1094211B (bg)
LU (1) LU79007A1 (bg)
NL (1) NL175997C (bg)
NO (2) NO145955C (bg)
NZ (1) NZ186384A (bg)
PH (2) PH14836A (bg)
PL (3) PL113163B1 (bg)
PT (1) PT67569B (bg)
RO (3) RO79258A (bg)
SE (2) SE445222B (bg)
SU (3) SU805949A3 (bg)
YU (3) YU39504B (bg)
ZA (1) ZA78646B (bg)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4413119A (en) * 1982-03-01 1983-11-01 Pfizer Inc. Semi-synthetic macrolides
US4363803A (en) * 1982-03-01 1982-12-14 Pfizer Inc. 3",4"-Oxyallylene erythromycin and oleandomycin, composition and method of use
JPH0240447U (bg) * 1988-09-14 1990-03-19
US5141926A (en) * 1990-04-18 1992-08-25 Abbott Laboratories Erythromycin derivatives
JPH05155896A (ja) * 1991-01-18 1993-06-22 Yamanouchi Pharmaceut Co Ltd 新規マクロライド化合物及びその製造法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3022219A (en) * 1958-03-07 1962-02-20 Pfizer & Co C Acyl esters of oleandomycin
US3179652A (en) * 1961-09-05 1965-04-20 Pfizer & Co C Antibiotic recovery process and salts produced thereby
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3842069A (en) * 1973-06-21 1974-10-15 Abbott Lab 4"-deoxy-4"-oxoerythromycin b derivatives
US4036853A (en) * 1976-08-06 1977-07-19 Pfizer Inc. Semi-synthetic oleandomycin derivatives-C8 modifications

Also Published As

Publication number Publication date
CA1106366A (en) 1981-08-04
YU39517B (en) 1984-12-31
ATA72078A (de) 1980-01-15
HU181395B (en) 1983-07-28
YU300377A (en) 1982-10-31
NO811914L (no) 1978-08-07
IL61606A0 (en) 1981-01-30
IT1094211B (it) 1985-07-26
PL113163B1 (en) 1980-11-29
NL175997B (nl) 1984-09-03
FI65262C (fi) 1984-04-10
CS200538B2 (en) 1980-09-15
CH629821A5 (fr) 1982-05-14
DE2804509A1 (de) 1978-08-10
SE457085B (sv) 1988-11-28
SU1020004A3 (ru) 1983-05-23
GR68692B (bg) 1982-02-01
FI65262B (fi) 1983-12-30
NO150439B (no) 1984-07-09
YU39518B (en) 1984-12-31
IE780240L (en) 1978-08-04
NL7801259A (nl) 1978-08-08
NO780390L (no) 1978-08-07
US4125705A (en) 1978-11-14
DE2804509C2 (de) 1982-12-02
HU179744B (en) 1982-12-28
BE863618A (fr) 1978-08-03
PT67569A (en) 1978-02-01
IE46395B1 (en) 1983-06-01
PL110793B1 (en) 1980-07-31
YU39504B (en) 1984-12-31
SE8300869D0 (sv) 1983-02-16
GB1583921A (en) 1981-02-04
JPS56135497A (en) 1981-10-22
YU151782A (en) 1982-10-31
CS200537B2 (en) 1980-09-15
FR2396022A1 (fr) 1979-01-26
JPS5398981A (en) 1978-08-29
BG32117A4 (bg) 1982-05-14
AT358169B (de) 1980-08-25
FR2383964B1 (bg) 1981-11-27
PH14836A (en) 1981-12-16
LU79007A1 (fr) 1979-09-06
DK51778A (da) 1978-08-05
ZA78646B (en) 1978-12-27
PL111160B1 (en) 1980-08-30
SU888824A3 (ru) 1981-12-07
PH16491A (en) 1983-10-28
FR2396022B1 (bg) 1980-06-13
AU502293B1 (en) 1979-07-19
JPS5652036B2 (bg) 1981-12-09
FR2383964A1 (fr) 1978-10-13
RO75387A (ro) 1980-11-30
JPS5827799B2 (ja) 1983-06-11
NO150439C (no) 1984-10-17
NO145955C (no) 1982-06-30
NL175997C (nl) 1985-02-01
RO79264A (ro) 1982-06-25
SE7800269L (sv) 1978-08-05
SU805949A3 (ru) 1981-02-15
PL204041A1 (pl) 1979-06-04
YU151882A (en) 1982-10-31
DK149628B (da) 1986-08-18
NO145955B (no) 1982-03-22
DD134523A5 (de) 1979-03-07
ES465322A1 (es) 1978-09-16
NZ186384A (en) 1980-08-26
CS200536B2 (en) 1980-09-15
DK149628C (da) 1987-02-02
IT7820006A0 (it) 1978-02-03
PT67569B (en) 1979-06-18
AR215666A1 (es) 1979-10-31
IL53959A0 (en) 1978-04-30
SE445222B (sv) 1986-06-09
RO79258A (ro) 1982-06-25
FI780355A (fi) 1978-08-05

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