AU593244B2 - Antipsychotic fused-ring pyroidinylpiperazine derivatives - Google Patents

Antipsychotic fused-ring pyroidinylpiperazine derivatives

Info

Publication number: AU593244B2
Authority: AU; Australia
Prior art keywords: pyroidinylpiperazine; antipsychotic; fused; derivatives; ring
Prior art date: 1985-05-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

AU56795/86A

Other languages

English (en)

Other versions

AU5679586A (en

Inventor

James Stewart New

Joseph P. Yevich

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bristol Myers Squibb Co

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-05-06

Filing date

1986-04-29

Publication date

1990-02-08

1986-04-29 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1986-11-13 Publication of AU5679586A publication Critical patent/AU5679586A/en

1990-02-08 Application granted granted Critical

1990-02-08 Publication of AU593244B2 publication Critical patent/AU593244B2/en

1993-08-05 Assigned to BRISTOL-MYERS SQUIBB COMPANY reassignment BRISTOL-MYERS SQUIBB COMPANY Request to Amend Deed and Register Assignors: BRISTOL-MYERS COMPANY

2006-04-29 Anticipated expiration legal-status Critical

Status Expired legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

AU56795/86A 1985-05-06 1986-04-29 Antipsychotic fused-ring pyroidinylpiperazine derivatives Expired AU593244B2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US73120185A	1985-05-06	1985-05-06
US731201		1985-05-06

Publications (2)

Publication Number	Publication Date
AU5679586A AU5679586A (en)	1986-11-13
AU593244B2 true AU593244B2 (en)	1990-02-08

Family

ID=24938510

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU56795/86A Expired AU593244B2 (en)	1985-05-06	1986-04-29	Antipsychotic fused-ring pyroidinylpiperazine derivatives

Country Status (25)

Country	Link
JP (1)	JPH0753728B2 (ja)
KR (1)	KR940000829B1 (ja)
CN (1)	CN1017901B (ja)
AT (1)	AT398572B (ja)
AU (1)	AU593244B2 (ja)
BE (1)	BE904724A (ja)
CA (1)	CA1278792C (ja)
CH (1)	CH672787A5 (ja)
DE (1)	DE3615180C2 (ja)
DK (1)	DK165745C (ja)
EG (1)	EG18206A (ja)
ES (6)	ES8801250A1 (ja)
FI (1)	FI85484C (ja)
FR (1)	FR2581385B1 (ja)
GB (1)	GB2174703B (ja)
GR (1)	GR861149B (ja)
HU (1)	HU195509B (ja)
IE (1)	IE59201B1 (ja)
IT (1)	IT1208607B (ja)
LU (1)	LU86421A1 (ja)
MY (1)	MY100777A (ja)
NL (1)	NL8601146A (ja)
PT (1)	PT82523B (ja)
SE (1)	SE465270B (ja)
ZA (1)	ZA862046B (ja)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5801186A (en) *	1987-11-20	1998-09-01	Hoechst Marion Roussel, Inc.	3- 4-(1-substituted-4-piperazinyl)butyl!-4-thiazolidinone and related compounds
US4880930A (en) *	1987-11-30	1989-11-14	New James S	Psychotropic acyclic amide derivatives
US4780466A (en) *	1988-03-17	1988-10-25	Hoechst-Roussel Pharmaceuticals, Inc.	Arylpiperazinylalkoxy derivatives of cyclic imides
IE903410A1 (en) *	1989-10-09	1991-04-10	Novo Nordisk As	Indole derivatives, their preparation and use
US5272148A (en) *	1992-09-09	1993-12-21	Hoechst-Roussel Pharmaceuticals Incorporated	Heteroarenylpiperazines
FR2738822B1 (fr) *	1995-09-15	1997-10-31	Synthelabo	Derives de 4-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)quinolein-2(1h)-one, leur preparation et leur application en therapeutique
FR2738823B1 (fr) *	1995-09-15	1997-10-31	Synthelabo	Derives de 3-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)-3,4-dihydroquinolein-2(1h)-one,leur preparation et leur application en therapeutique
FR2738824B1 (fr) *	1995-09-15	1997-10-31	Synthelabo	Derives de 3-(omega(4-(thieno(3,2-c)pyridin-4-yl)piperazin-1 -yl)alkyl)-3,4-dihydroquinazolin-2(1h)-one,leur preparation et leur application en therapeutique
JP3335362B2 (ja) *	1995-09-15	2002-10-15	サノフィ―サンテラボ	キノレイン−２（１ｈ）−オン誘導体セロトニンアンタゴニスト
FR2761071B1 (fr) *	1997-03-20	1999-12-03	Synthelabo	Derives de quinolein-2(1h)-one et de dihydroquinolein-2(1h)- one, leur preparation et leur application en therapeutique
FR2797874B1 (fr) *	1999-08-27	2002-03-29	Adir	Nouveaux derives de la pyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4367335A (en) *	1981-08-03	1983-01-04	Mead Johnson & Company	Thiazolidinylalkylene piperazine derivatives
US4452799A (en) *	1981-12-23	1984-06-05	Mead Johnson & Company	Benzisothiazole and benzisoxazole piperazine derivatives
US4361565A (en) *	1981-12-28	1982-11-30	Mead Johnson & Company	2-[4-[(4,4-Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyridines

1986
- 1986-03-11 CA CA000503794A patent/CA1278792C/en not_active Expired - Fee Related
- 1986-03-19 ZA ZA862046A patent/ZA862046B/xx unknown
- 1986-04-29 GR GR861149A patent/GR861149B/el unknown
- 1986-04-29 EG EG250/86A patent/EG18206A/xx active
- 1986-04-29 AU AU56795/86A patent/AU593244B2/en not_active Expired
- 1986-04-30 FI FI861820A patent/FI85484C/fi not_active IP Right Cessation
- 1986-05-02 GB GB08610810A patent/GB2174703B/en not_active Expired
- 1986-05-02 KR KR1019860003445A patent/KR940000829B1/ko not_active IP Right Cessation
- 1986-05-05 CN CN86103071A patent/CN1017901B/zh not_active Expired
- 1986-05-05 DE DE3615180A patent/DE3615180C2/de not_active Expired - Lifetime
- 1986-05-05 IE IE119386A patent/IE59201B1/en not_active IP Right Cessation
- 1986-05-05 SE SE8602061A patent/SE465270B/sv not_active IP Right Cessation
- 1986-05-05 NL NL8601146A patent/NL8601146A/nl active Search and Examination
- 1986-05-05 ES ES554659A patent/ES8801250A1/es not_active Expired
- 1986-05-05 CH CH1830/86A patent/CH672787A5/de not_active IP Right Cessation
- 1986-05-05 LU LU86421A patent/LU86421A1/fr unknown
- 1986-05-05 FR FR8606471A patent/FR2581385B1/fr not_active Expired - Lifetime
- 1986-05-05 DK DK207186A patent/DK165745C/da not_active IP Right Cessation
- 1986-05-05 BE BE0/216623A patent/BE904724A/fr not_active IP Right Cessation
- 1986-05-06 IT IT8620313A patent/IT1208607B/it active
- 1986-05-06 PT PT82523A patent/PT82523B/pt unknown
- 1986-05-06 AT AT0121486A patent/AT398572B/de not_active IP Right Cessation
- 1986-05-06 HU HU861860A patent/HU195509B/hu unknown
- 1986-05-06 JP JP61103726A patent/JPH0753728B2/ja not_active Expired - Lifetime
1987
- 1987-09-25 ES ES557757A patent/ES8802149A1/es not_active Expired
- 1987-10-01 MY MYPI87002712A patent/MY100777A/en unknown
1988
- 1988-01-28 ES ES557809A patent/ES8802614A1/es not_active Expired
- 1988-05-26 ES ES557839A patent/ES8900138A1/es not_active Expired
- 1988-11-16 ES ES557855A patent/ES8900253A1/es not_active Expired
1989
- 1989-02-27 ES ES557865A patent/ES9000005A1/es not_active Expired

Also Published As

Publication number	Publication date
GB2174703B (en)	1988-10-26
HU195509B (en)	1988-05-30
FI85484B (fi)	1992-01-15
DK165745C (da)	1993-06-14
DE3615180C2 (de)	1996-03-07
JPH0753728B2 (ja)	1995-06-07
HUT43848A (en)	1987-12-28
GR861149B (en)	1986-09-09
IT1208607B (it)	1989-07-10
NL8601146A (nl)	1986-12-01
ES8900253A1 (es)	1989-05-16
ATA121486A (de)	1994-05-15
SE8602061D0 (sv)	1986-05-05
GB2174703A (en)	1986-11-12
ES8801250A1 (es)	1987-12-16
AU5679586A (en)	1986-11-13
LU86421A1 (fr)	1986-12-05
FI85484C (fi)	1992-04-27
ES554659A0 (es)	1987-12-16
FR2581385A1 (fr)	1986-11-07
CN86103071A (zh)	1987-03-18
GB8610810D0 (en)	1986-06-11
ES9000005A1 (es)	1989-11-01
ES557809A0 (es)	1988-09-01
ES557855A0 (es)	1989-05-16
PT82523A (en)	1986-06-01
ES8802149A1 (es)	1988-04-01
ZA862046B (en)	1986-11-26
SE465270B (sv)	1991-08-19
ES557757A0 (es)	1988-04-01
IE59201B1 (en)	1994-01-26
ES8900138A1 (es)	1989-01-16
ES557839A0 (es)	1989-01-16
FI861820A0 (fi)	1986-04-30
DK207186D0 (da)	1986-05-05
IE861193L (en)	1986-11-06
AT398572B (de)	1994-12-27
BE904724A (fr)	1986-11-05
MY100777A (en)	1991-02-14
SE8602061L (sv)	1986-11-07
FI861820A (fi)	1986-11-07
CH672787A5 (ja)	1989-12-29
DK165745B (da)	1993-01-11
JPS61268681A (ja)	1986-11-28
DE3615180A1 (de)	1986-11-06
KR940000829B1 (ko)	1994-02-02
CN1017901B (zh)	1992-08-19
EG18206A (en)	1992-09-30
PT82523B (pt)	1988-10-14
ES8802614A1 (es)	1988-09-01
KR860009008A (ko)	1986-12-19
CA1278792C (en)	1991-01-08
FR2581385B1 (fr)	1991-10-04
DK207186A (da)	1986-11-07
IT8620313A0 (it)	1986-05-06

Publication	Publication Date	Title
AU572402B2 (en)	1988-05-05	25-avermectin derivatives
AU5912086A (en)	1986-12-24	Substituted 3-phenyl-cyanopyrrole derivatives
AU583607B2 (en)	1989-05-04	Indole derivatives
AU585351B2 (en)	1989-06-15	3-benzazepine derivatives
AU583343B2 (en)	1989-04-27	Heterocyclic compounds
AU6418286A (en)	1987-04-30	3-quinuclidinylmethyl derivatives
AU591210B2 (en)	1989-11-30	1-acyl-2-aminomethyl azacylclic derivatives
AU6416986A (en)	1987-04-30	Heterocyclic compounds
AU6398586A (en)	1987-04-30	Benzoheterocyclylcarboxamide derivatives
AU589685B2 (en)	1989-10-19	New derivatives
AU6538686A (en)	1987-05-21	5-phenyl-2-oxazole derivatives
AU6101086A (en)	1987-02-12	7-formamidoceph-3-em-4-carboxylate derivatives
AU6150386A (en)	1987-02-19	Guanine derivatives
AU593244B2 (en)	1990-02-08	Antipsychotic fused-ring pyroidinylpiperazine derivatives
AU5397486A (en)	1986-08-26	Heterocyclic derivatives
AU5638686A (en)	1986-10-23	Cyclohexylamidazole derivatives
AU562773B2 (en)	1987-06-18	Tetrahydroimidazoquinazolinone derivatives
AU6202986A (en)	1987-03-05	6-phenoxymethyl-4-hydroxytetrahydropyran-2-one derivatives
AU581066B2 (en)	1989-02-09	Cyanoalkanimidamidophenylpyridazinone derivatives
AU5511986A (en)	1986-10-13	2-arylbenzothiazine derivatives
AU561320B2 (en)	1987-05-07	Clycoside derivatives
AU5363090A (en)	1990-09-13	Novel terahydroisoquinoline derivatives
AU576962B2 (en)	1988-09-08	Substituted hexahydro arylquinolizine derivatives
AU6031086A (en)	1987-01-22	Dihydroquinolinone derivatives
AU586700B2 (en)	1989-07-20	N-sulfanoyl-3-halo-propionamidine derivatives