PT82523B - Processo para a preparacao de compostos antipsicoticos com um anel condensado derivados da piridinilpiperazina e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de compostos antipsicoticos com um anel condensado derivados da piridinilpiperazina e de composicoes farmaceuticas que os contem

Info

Publication number
PT82523B
PT82523B PT82523A PT8252386A PT82523B PT 82523 B PT82523 B PT 82523B PT 82523 A PT82523 A PT 82523A PT 8252386 A PT8252386 A PT 8252386A PT 82523 B PT82523 B PT 82523B
Authority
PT
Portugal
Prior art keywords
pyridinylpiperazine
preparation
pharmaceutical compositions
compositions containing
condensed ring
Prior art date
Application number
PT82523A
Other languages
English (en)
Other versions
PT82523A (en
Inventor
Joseph P Yevich
James Stewart New
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of PT82523A publication Critical patent/PT82523A/pt
Publication of PT82523B publication Critical patent/PT82523B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT82523A 1985-05-06 1986-05-06 Processo para a preparacao de compostos antipsicoticos com um anel condensado derivados da piridinilpiperazina e de composicoes farmaceuticas que os contem PT82523B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73120185A 1985-05-06 1985-05-06

Publications (2)

Publication Number Publication Date
PT82523A PT82523A (en) 1986-06-01
PT82523B true PT82523B (pt) 1988-10-14

Family

ID=24938510

Family Applications (1)

Application Number Title Priority Date Filing Date
PT82523A PT82523B (pt) 1985-05-06 1986-05-06 Processo para a preparacao de compostos antipsicoticos com um anel condensado derivados da piridinilpiperazina e de composicoes farmaceuticas que os contem

Country Status (25)

Country Link
JP (1) JPH0753728B2 (pt)
KR (1) KR940000829B1 (pt)
CN (1) CN1017901B (pt)
AT (1) AT398572B (pt)
AU (1) AU593244B2 (pt)
BE (1) BE904724A (pt)
CA (1) CA1278792C (pt)
CH (1) CH672787A5 (pt)
DE (1) DE3615180C2 (pt)
DK (1) DK165745C (pt)
EG (1) EG18206A (pt)
ES (6) ES8801250A1 (pt)
FI (1) FI85484C (pt)
FR (1) FR2581385B1 (pt)
GB (1) GB2174703B (pt)
GR (1) GR861149B (pt)
HU (1) HU195509B (pt)
IE (1) IE59201B1 (pt)
IT (1) IT1208607B (pt)
LU (1) LU86421A1 (pt)
MY (1) MY100777A (pt)
NL (1) NL8601146A (pt)
PT (1) PT82523B (pt)
SE (1) SE465270B (pt)
ZA (1) ZA862046B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5801186A (en) * 1987-11-20 1998-09-01 Hoechst Marion Roussel, Inc. 3- 4-(1-substituted-4-piperazinyl)butyl!-4-thiazolidinone and related compounds
US4880930A (en) * 1987-11-30 1989-11-14 New James S Psychotropic acyclic amide derivatives
US4780466A (en) * 1988-03-17 1988-10-25 Hoechst-Roussel Pharmaceuticals, Inc. Arylpiperazinylalkoxy derivatives of cyclic imides
IE903410A1 (en) * 1989-10-09 1991-04-10 Novo Nordisk As Indole derivatives, their preparation and use
US5272148A (en) * 1992-09-09 1993-12-21 Hoechst-Roussel Pharmaceuticals Incorporated Heteroarenylpiperazines
FR2738822B1 (fr) * 1995-09-15 1997-10-31 Synthelabo Derives de 4-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)quinolein-2(1h)-one, leur preparation et leur application en therapeutique
FR2738823B1 (fr) * 1995-09-15 1997-10-31 Synthelabo Derives de 3-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)-3,4-dihydroquinolein-2(1h)-one,leur preparation et leur application en therapeutique
FR2738824B1 (fr) * 1995-09-15 1997-10-31 Synthelabo Derives de 3-(omega(4-(thieno(3,2-c)pyridin-4-yl)piperazin-1 -yl)alkyl)-3,4-dihydroquinazolin-2(1h)-one,leur preparation et leur application en therapeutique
JP3335362B2 (ja) * 1995-09-15 2002-10-15 サノフィ―サンテラボ キノレイン−2(1h)−オン誘導体セロトニンアンタゴニスト
FR2761071B1 (fr) * 1997-03-20 1999-12-03 Synthelabo Derives de quinolein-2(1h)-one et de dihydroquinolein-2(1h)- one, leur preparation et leur application en therapeutique
FR2797874B1 (fr) * 1999-08-27 2002-03-29 Adir Nouveaux derives de la pyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4367335A (en) * 1981-08-03 1983-01-04 Mead Johnson & Company Thiazolidinylalkylene piperazine derivatives
US4452799A (en) * 1981-12-23 1984-06-05 Mead Johnson & Company Benzisothiazole and benzisoxazole piperazine derivatives
US4361565A (en) * 1981-12-28 1982-11-30 Mead Johnson & Company 2-[4-[(4,4-Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyridines

Also Published As

Publication number Publication date
GB2174703B (en) 1988-10-26
AU593244B2 (en) 1990-02-08
HU195509B (en) 1988-05-30
FI85484B (fi) 1992-01-15
DK165745C (da) 1993-06-14
DE3615180C2 (de) 1996-03-07
JPH0753728B2 (ja) 1995-06-07
HUT43848A (en) 1987-12-28
GR861149B (en) 1986-09-09
IT1208607B (it) 1989-07-10
NL8601146A (nl) 1986-12-01
ES8900253A1 (es) 1989-05-16
ATA121486A (de) 1994-05-15
SE8602061D0 (sv) 1986-05-05
GB2174703A (en) 1986-11-12
ES8801250A1 (es) 1987-12-16
AU5679586A (en) 1986-11-13
LU86421A1 (fr) 1986-12-05
FI85484C (fi) 1992-04-27
ES554659A0 (es) 1987-12-16
FR2581385A1 (fr) 1986-11-07
CN86103071A (zh) 1987-03-18
GB8610810D0 (en) 1986-06-11
ES9000005A1 (es) 1989-11-01
ES557809A0 (es) 1988-09-01
ES557855A0 (es) 1989-05-16
PT82523A (en) 1986-06-01
ES8802149A1 (es) 1988-04-01
ZA862046B (en) 1986-11-26
SE465270B (sv) 1991-08-19
ES557757A0 (es) 1988-04-01
IE59201B1 (en) 1994-01-26
ES8900138A1 (es) 1989-01-16
ES557839A0 (es) 1989-01-16
FI861820A0 (fi) 1986-04-30
DK207186D0 (da) 1986-05-05
IE861193L (en) 1986-11-06
AT398572B (de) 1994-12-27
BE904724A (fr) 1986-11-05
MY100777A (en) 1991-02-14
SE8602061L (sv) 1986-11-07
FI861820A (fi) 1986-11-07
CH672787A5 (pt) 1989-12-29
DK165745B (da) 1993-01-11
JPS61268681A (ja) 1986-11-28
DE3615180A1 (de) 1986-11-06
KR940000829B1 (ko) 1994-02-02
CN1017901B (zh) 1992-08-19
EG18206A (en) 1992-09-30
ES8802614A1 (es) 1988-09-01
KR860009008A (ko) 1986-12-19
CA1278792C (en) 1991-01-08
FR2581385B1 (fr) 1991-10-04
DK207186A (da) 1986-11-07
IT8620313A0 (it) 1986-05-06

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