ATE495147T1 - Ein verfahren zur herstellung eines phenylalaninderivats und zwischenprodukte davon - Google Patents

Ein verfahren zur herstellung eines phenylalaninderivats und zwischenprodukte davon

Info

Publication number
ATE495147T1
ATE495147T1 AT03707122T AT03707122T ATE495147T1 AT E495147 T1 ATE495147 T1 AT E495147T1 AT 03707122 T AT03707122 T AT 03707122T AT 03707122 T AT03707122 T AT 03707122T AT E495147 T1 ATE495147 T1 AT E495147T1
Authority
AT
Austria
Prior art keywords
producing
intermediate products
phenylalanine derivative
phenylalanine
derivative
Prior art date
Application number
AT03707122T
Other languages
English (en)
Inventor
Isao Inoue
Toru Kuroda
Ryuzo Yoshioka
Original Assignee
Mitsubishi Tanabe Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Tanabe Pharma Corp filed Critical Mitsubishi Tanabe Pharma Corp
Application granted granted Critical
Publication of ATE495147T1 publication Critical patent/ATE495147T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT03707122T 2002-02-28 2003-02-27 Ein verfahren zur herstellung eines phenylalaninderivats und zwischenprodukte davon ATE495147T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002052605 2002-02-28
PCT/JP2003/002181 WO2003072536A1 (en) 2002-02-28 2003-02-27 A process for preparing a phenylalanine derivative and intermediates thereof

Publications (1)

Publication Number Publication Date
ATE495147T1 true ATE495147T1 (de) 2011-01-15

Family

ID=27764341

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03707122T ATE495147T1 (de) 2002-02-28 2003-02-27 Ein verfahren zur herstellung eines phenylalaninderivats und zwischenprodukte davon

Country Status (22)

Country Link
US (1) US7476758B2 (de)
EP (1) EP1478619B1 (de)
KR (1) KR100681224B1 (de)
CN (2) CN100522930C (de)
AR (1) AR038624A1 (de)
AT (1) ATE495147T1 (de)
AU (1) AU2003208618B2 (de)
BR (1) BR0308027A (de)
CA (1) CA2476022C (de)
DE (1) DE60335704D1 (de)
ES (1) ES2359302T3 (de)
HK (1) HK1069382A1 (de)
IL (1) IL163429A (de)
MX (1) MXPA04008359A (de)
MY (1) MY140707A (de)
NO (1) NO331001B1 (de)
NZ (1) NZ534957A (de)
PL (1) PL211046B1 (de)
RU (1) RU2280641C2 (de)
TW (1) TWI327996B (de)
WO (1) WO2003072536A1 (de)
ZA (1) ZA200406747B (de)

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JP2008542407A (ja) 2005-06-09 2008-11-27 ユセベ ファルマ ソシエテ アノニム ２，６キノリニル誘導体、それらを調製するための方法及び薬剤としてのそれらの使用
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EA201290165A1 (ru) 2009-10-21 2012-11-30 Глаксо Груп Лимитед Способ получения производного фенилаланина
CN112969504B (zh) 2018-10-30 2024-04-09 吉利德科学公司 用于抑制α4β7整合素的化合物
CA3114240C (en) 2018-10-30 2023-09-05 Gilead Sciences, Inc. Imidazopyridine derivatives as alpha4beta7 integrin inhibitors
CA3115820A1 (en) 2018-10-30 2020-05-07 Gilead Sciences, Inc. Compounds for inhibition of .alpha.4.beta.7 integrin
WO2020092375A1 (en) 2018-10-30 2020-05-07 Gilead Sciences, Inc. Quinoline derivatives as alpha4beta7 integrin inhibitors
CA3148613A1 (en) 2019-08-14 2021-02-18 Gilead Sciences, Inc. Phenylalanine derived compounds and their use as inhinitors of alpha 4 beta 7 integrin

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Also Published As

Publication number Publication date
KR100681224B1 (ko) 2007-02-09
CN1817853A (zh) 2006-08-16
PL371386A1 (en) 2005-06-13
MY140707A (en) 2010-01-15
US20050165107A1 (en) 2005-07-28
ES2359302T3 (es) 2011-05-20
AU2003208618B2 (en) 2008-06-19
CN1646482A (zh) 2005-07-27
KR20040091665A (ko) 2004-10-28
US7476758B2 (en) 2009-01-13
NO20044087L (no) 2004-09-27
EP1478619B1 (de) 2011-01-12
WO2003072536A1 (en) 2003-09-04
CN100480233C (zh) 2009-04-22
RU2004128935A (ru) 2006-02-20
HK1069382A1 (en) 2005-05-20
TWI327996B (en) 2010-08-01
ZA200406747B (en) 2005-08-31
RU2280641C2 (ru) 2006-07-27
AR038624A1 (es) 2005-01-19
MXPA04008359A (es) 2004-11-26
AU2003208618A1 (en) 2003-09-09
DE60335704D1 (de) 2011-02-24
CN100522930C (zh) 2009-08-05
EP1478619A1 (de) 2004-11-24
TW200303854A (en) 2003-09-16
CA2476022C (en) 2008-07-15
CA2476022A1 (en) 2003-09-04
PL211046B1 (pl) 2012-04-30
NZ534957A (en) 2006-11-30
BR0308027A (pt) 2004-12-28
NO331001B1 (no) 2011-09-05
IL163429A (en) 2012-07-31

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties