NO331001B1 - Fremgangsmate for fremstilling av et fenylalaninderivat, mellomprodukt i fremgangsmaten, samt fremgangsmate for fremstilling av mellomproduktet - Google Patents

Fremgangsmate for fremstilling av et fenylalaninderivat, mellomprodukt i fremgangsmaten, samt fremgangsmate for fremstilling av mellomproduktet

Info

Publication number
NO331001B1
NO331001B1 NO20044087A NO20044087A NO331001B1 NO 331001 B1 NO331001 B1 NO 331001B1 NO 20044087 A NO20044087 A NO 20044087A NO 20044087 A NO20044087 A NO 20044087A NO 331001 B1 NO331001 B1 NO 331001B1
Authority
NO
Norway
Prior art keywords
preparation
phenylalanine derivative
phenylalanine
derivative
Prior art date
Application number
NO20044087A
Other languages
English (en)
Other versions
NO20044087L (no
Inventor
Isao Inoue
Toru Kuroda
Ryuzo Yoshioka
Original Assignee
Mitsubishi Tanabe Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Tanabe Pharma Corp filed Critical Mitsubishi Tanabe Pharma Corp
Publication of NO20044087L publication Critical patent/NO20044087L/no
Publication of NO331001B1 publication Critical patent/NO331001B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20044087A 2002-02-28 2004-09-27 Fremgangsmate for fremstilling av et fenylalaninderivat, mellomprodukt i fremgangsmaten, samt fremgangsmate for fremstilling av mellomproduktet NO331001B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002052605 2002-02-28
PCT/JP2003/002181 WO2003072536A1 (en) 2002-02-28 2003-02-27 A process for preparing a phenylalanine derivative and intermediates thereof

Publications (2)

Publication Number Publication Date
NO20044087L NO20044087L (no) 2004-09-27
NO331001B1 true NO331001B1 (no) 2011-09-05

Family

ID=27764341

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20044087A NO331001B1 (no) 2002-02-28 2004-09-27 Fremgangsmate for fremstilling av et fenylalaninderivat, mellomprodukt i fremgangsmaten, samt fremgangsmate for fremstilling av mellomproduktet

Country Status (22)

Country Link
US (1) US7476758B2 (no)
EP (1) EP1478619B1 (no)
KR (1) KR100681224B1 (no)
CN (2) CN100480233C (no)
AR (1) AR038624A1 (no)
AT (1) ATE495147T1 (no)
AU (1) AU2003208618B2 (no)
BR (1) BR0308027A (no)
CA (1) CA2476022C (no)
DE (1) DE60335704D1 (no)
ES (1) ES2359302T3 (no)
HK (1) HK1069382A1 (no)
IL (1) IL163429A (no)
MX (1) MXPA04008359A (no)
MY (1) MY140707A (no)
NO (1) NO331001B1 (no)
NZ (1) NZ534957A (no)
PL (1) PL211046B1 (no)
RU (1) RU2280641C2 (no)
TW (1) TWI327996B (no)
WO (1) WO2003072536A1 (no)
ZA (1) ZA200406747B (no)

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AR078521A1 (es) 2009-10-08 2011-11-16 Eisai R&D Man Co Ltd Compuesto pirazolotiazol
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AU2019373242B2 (en) 2018-10-30 2023-07-13 Gilead Sciences, Inc. Compounds for inhibition of alpha 4 beta 7 integrin
KR102659859B1 (ko) 2018-10-30 2024-04-25 길리애드 사이언시즈, 인코포레이티드 알파4β7 인테그린의 억제를 위한 화합물
EP3873884A1 (en) 2018-10-30 2021-09-08 Gilead Sciences, Inc. Quinoline derivatives as alpha4beta7 integrin inhibitors
US11174256B2 (en) 2018-10-30 2021-11-16 Gilead Sciences, Inc. Imidazopyridine derivatives
KR20220047323A (ko) 2019-08-14 2022-04-15 길리애드 사이언시즈, 인코포레이티드 알파 4 베타 7 인테그린의 저해용 화합물

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Also Published As

Publication number Publication date
AU2003208618A1 (en) 2003-09-09
DE60335704D1 (de) 2011-02-24
US20050165107A1 (en) 2005-07-28
RU2280641C2 (ru) 2006-07-27
TW200303854A (en) 2003-09-16
KR20040091665A (ko) 2004-10-28
KR100681224B1 (ko) 2007-02-09
RU2004128935A (ru) 2006-02-20
AR038624A1 (es) 2005-01-19
EP1478619A1 (en) 2004-11-24
AU2003208618B2 (en) 2008-06-19
CN100522930C (zh) 2009-08-05
CN1646482A (zh) 2005-07-27
HK1069382A1 (en) 2005-05-20
ZA200406747B (en) 2005-08-31
EP1478619B1 (en) 2011-01-12
MY140707A (en) 2010-01-15
ES2359302T3 (es) 2011-05-20
NO20044087L (no) 2004-09-27
ATE495147T1 (de) 2011-01-15
TWI327996B (en) 2010-08-01
PL371386A1 (en) 2005-06-13
CA2476022A1 (en) 2003-09-04
MXPA04008359A (es) 2004-11-26
CA2476022C (en) 2008-07-15
NZ534957A (en) 2006-11-30
PL211046B1 (pl) 2012-04-30
WO2003072536A1 (en) 2003-09-04
IL163429A (en) 2012-07-31
CN1817853A (zh) 2006-08-16
CN100480233C (zh) 2009-04-22
BR0308027A (pt) 2004-12-28
US7476758B2 (en) 2009-01-13

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Legal Events

Date Code Title Description
CHAD Change of the owner's name or address (par. 44 patent law, par. patentforskriften)

Owner name: MITSUBISHI TANABE PHARMA CORP (JP)

CHAD Change of the owner's name or address (par. 44 patent law, par. patentforskriften)

Owner name: MITSUBISHI TANABE PHARMA CORP, JP

MM1K Lapsed by not paying the annual fees