ZA200707471B - Novel derivatives of phosphinic amino acids, preparation method thereof and pharmaceutical compositions containing same - Google Patents

Novel derivatives of phosphinic amino acids, preparation method thereof and pharmaceutical compositions containing same

Info

Publication number: ZA200707471B
Authority: ZA; South Africa
Prior art keywords: preparation; amino acids; pharmaceutical compositions; compositions containing; containing same
Prior art date: 2005-03-01

Application number

ZA200707471A

Other languages

English (en)

Inventor

Dive Vincent

Jullien Nicolas

Scalbert Elizabeth

Yiotakis Athanasios

Makaritis Anastasios

Original Assignee

Servier Lab

Commissariat Energie Atomique

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-03-01

Filing date

2006-02-28

Publication date

2008-12-31

2006-02-28 Application filed by Servier Lab, Commissariat Energie Atomique filed Critical Servier Lab

2008-12-31 Publication of ZA200707471B publication Critical patent/ZA200707471B/xx

Links

150000001413 amino acids Chemical class 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1
238000002360 preparation method Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
- C07F9/653—Five-membered rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- C07F9/32—Esters thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6596—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having atoms other than oxygen, sulfur, selenium, tellurium, nitrogen or phosphorus as ring hetero atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Cardiology (AREA)
Biochemistry (AREA)
Heart & Thoracic Surgery (AREA)
Molecular Biology (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Hematology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Ophthalmology & Optometry (AREA)
Hospice & Palliative Care (AREA)
Diabetes (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

ZA200707471A 2005-03-01 2006-02-28 Novel derivatives of phosphinic amino acids, preparation method thereof and pharmaceutical compositions containing same ZA200707471B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0502043A FR2882752B1 (fr)	2005-03-01	2005-03-01	Nouveaux derives d'aminoacides phosphiniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number	Publication Date
ZA200707471B true ZA200707471B (en)	2008-12-31

Family

ID=35033564

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200707471A ZA200707471B (en)	2005-03-01	2006-02-28	Novel derivatives of phosphinic amino acids, preparation method thereof and pharmaceutical compositions containing same

Country Status (20)

Country	Link
US (1)	US7521469B2 (ru)
EP (1)	EP1853615A1 (ru)
JP (1)	JP4659843B2 (ru)
KR (1)	KR20080011275A (ru)
CN (1)	CN101133070A (ru)
AR (1)	AR055565A1 (ru)
AU (1)	AU2006219790B2 (ru)
BR (1)	BRPI0607482A2 (ru)
CA (1)	CA2601025C (ru)
EA (1)	EA012447B1 (ru)
FR (1)	FR2882752B1 (ru)
GE (1)	GEP20105026B (ru)
MA (1)	MA29315B1 (ru)
MX (1)	MX2007010665A (ru)
MY (1)	MY143558A (ru)
NO (1)	NO20074942L (ru)
NZ (1)	NZ560750A (ru)
UA (1)	UA91214C2 (ru)
WO (1)	WO2006092495A1 (ru)
ZA (1)	ZA200707471B (ru)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2934267B1 (fr) *	2008-07-23	2010-08-13	Pharmaleads	Derives aminophosphiniques utiles dans le traitement de la douleur

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5476847A (en) *	1994-06-29	1995-12-19	Schering Corporation	Derivatives of phosphinic acid useful as endothelin converting enzyme inhibitors
IT1276710B1 (it) *	1995-06-14	1997-11-03	Zambon Spa	Derivati dell'acido fosfinico ad attivita' inibitrice delle metallopeptidasi
FR2755135B1 (fr) *	1996-10-25	2002-12-27	Inst Nat Sante Rech Med	Nouveaux derives d'(alpha-aminophosphino)peptides, leur procede de preparation et les compositions qui les contiennent

2005
- 2005-03-01 FR FR0502043A patent/FR2882752B1/fr not_active Expired - Fee Related
2006
- 2006-02-27 MY MYPI20060824A patent/MY143558A/en unknown
- 2006-02-28 ZA ZA200707471A patent/ZA200707471B/xx unknown
- 2006-02-28 WO PCT/FR2006/000446 patent/WO2006092495A1/fr active Application Filing
- 2006-02-28 GE GEAP200610296A patent/GEP20105026B/en unknown
- 2006-02-28 BR BRPI0607482-0A patent/BRPI0607482A2/pt not_active IP Right Cessation
- 2006-02-28 US US11/885,301 patent/US7521469B2/en not_active Expired - Fee Related
- 2006-02-28 KR KR1020077022456A patent/KR20080011275A/ko not_active Application Discontinuation
- 2006-02-28 CA CA2601025A patent/CA2601025C/fr not_active Expired - Fee Related
- 2006-02-28 EP EP06725994A patent/EP1853615A1/fr not_active Withdrawn
- 2006-02-28 EA EA200701819A patent/EA012447B1/ru not_active IP Right Cessation
- 2006-02-28 AU AU2006219790A patent/AU2006219790B2/en not_active Expired - Fee Related
- 2006-02-28 MX MX2007010665A patent/MX2007010665A/es active IP Right Grant
- 2006-02-28 NZ NZ560750A patent/NZ560750A/en unknown
- 2006-02-28 CN CNA2006800068686A patent/CN101133070A/zh active Pending
- 2006-02-28 JP JP2007557535A patent/JP4659843B2/ja not_active Expired - Fee Related
- 2006-02-28 UA UAA200710758A patent/UA91214C2/ru unknown
- 2006-03-01 AR ARP060100755A patent/AR055565A1/es not_active Application Discontinuation
2007
- 2007-09-06 MA MA30192A patent/MA29315B1/fr unknown
- 2007-10-01 NO NO20074942A patent/NO20074942L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EA012447B1 (ru)	2009-10-30
EP1853615A1 (fr)	2007-11-14
AU2006219790A1 (en)	2006-09-08
MY143558A (en)	2011-05-31
BRPI0607482A2 (pt)	2009-09-08
EA200701819A1 (ru)	2008-02-28
JP2008531661A (ja)	2008-08-14
FR2882752A1 (fr)	2006-09-08
CN101133070A (zh)	2008-02-27
UA91214C2 (ru)	2010-07-12
NO20074942L (no)	2007-10-01
CA2601025C (fr)	2011-01-25
AR055565A1 (es)	2007-08-22
CA2601025A1 (fr)	2006-09-08
JP4659843B2 (ja)	2011-03-30
NZ560750A (en)	2010-12-24
US20080153890A1 (en)	2008-06-26
GEP20105026B (en)	2010-06-25
US7521469B2 (en)	2009-04-21
MX2007010665A (es)	2007-12-12
MA29315B1 (fr)	2008-03-03
WO2006092495A1 (fr)	2006-09-08
KR20080011275A (ko)	2008-02-01
FR2882752B1 (fr)	2007-05-04
AU2006219790B2 (en)	2011-03-17

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