ZA200007222B - Glycopeptide derivatives and pharmaceutical compositions containing the same. - Google Patents

Glycopeptide derivatives and pharmaceutical compositions containing the same.

Info

Publication number
ZA200007222B
ZA200007222B ZA200007222A ZA200007222A ZA200007222B ZA 200007222 B ZA200007222 B ZA 200007222B ZA 200007222 A ZA200007222 A ZA 200007222A ZA 200007222 A ZA200007222 A ZA 200007222A ZA 200007222 B ZA200007222 B ZA 200007222B
Authority
ZA
South Africa
Prior art keywords
pharmaceutical compositions
compositions containing
same
derivatives
glycopeptide derivatives
Prior art date
Application number
ZA200007222A
Other languages
English (en)
Inventor
J Kevin Judice
Bernice Lam
Martin Sheringham Linsell
Sean Gary Trapp
Gaung Yang
Paul Ross Fatheree
Michael Leadbetter
Yongqi Mu
Yan Zhu
Original Assignee
Advanced Medicine Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Advanced Medicine Inc filed Critical Advanced Medicine Inc
Publication of ZA200007222B publication Critical patent/ZA200007222B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA200007222A 1998-12-23 2000-12-06 Glycopeptide derivatives and pharmaceutical compositions containing the same. ZA200007222B (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US11372898P 1998-12-23 1998-12-23
US12931399P 1999-04-14 1999-04-14
US16402499P 1999-11-04 1999-11-04
US16997899P 1999-12-10 1999-12-10
PCT/US1999/030543 WO2000039156A1 (en) 1998-12-23 1999-12-22 Glycopeptide derivatives and pharmaceutical compositions containing the same

Publications (1)

Publication Number Publication Date
ZA200007222B true ZA200007222B (en) 2002-03-06

Family

ID=27493926

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200007222A ZA200007222B (en) 1998-12-23 2000-12-06 Glycopeptide derivatives and pharmaceutical compositions containing the same.

Country Status (23)

Country Link
US (9) US6392012B1 (pt)
EP (1) EP1140993B1 (pt)
JP (1) JP4362017B2 (pt)
KR (1) KR100665204B1 (pt)
CN (1) CN1249081C (pt)
AT (1) ATE242783T1 (pt)
AU (1) AU768204B2 (pt)
BR (1) BRPI9914221B8 (pt)
CA (1) CA2336445C (pt)
CZ (1) CZ301184B6 (pt)
DE (1) DE69908819T2 (pt)
DK (1) DK1140993T3 (pt)
ES (1) ES2201825T3 (pt)
HK (1) HK1040721B (pt)
HU (1) HU230190B1 (pt)
IL (2) IL140093A0 (pt)
NO (1) NO326066B1 (pt)
NZ (1) NZ508594A (pt)
PL (1) PL198311B1 (pt)
PT (1) PT1140993E (pt)
SI (1) SI1140993T1 (pt)
WO (1) WO2000039156A1 (pt)
ZA (1) ZA200007222B (pt)

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SI1278549T1 (sl) * 2000-05-02 2009-04-30 Theravance Inc Sestavek, ki vsebuje ciklodekstrin in glikopeptidni antibiotik
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US6770621B2 (en) * 2000-05-02 2004-08-03 Theravance, Inc. Polyacid glycopeptide derivatives
US6828299B2 (en) 2000-06-22 2004-12-07 Theravance, Inc. Polyhydroxy glycopeptide derivatives
ES2302733T3 (es) * 2000-06-22 2008-08-01 Theravance, Inc. Derivados carboxi-sacaridos de glucopeptido.
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US6872804B2 (en) 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
US6905669B2 (en) * 2001-04-24 2005-06-14 Supergen, Inc. Compositions and methods for reestablishing gene transcription through inhibition of DNA methylation and histone deacetylase
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) * 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
ATE322975T1 (de) 2001-09-19 2006-04-15 Procter & Gamble Farbbedruckte mehrschichtstruktur, ein damit hergestellter absorbierender artikel und verfahren zu deren herstellung
TWI335332B (en) 2001-10-12 2011-01-01 Theravance Inc Cross-linked vancomycin-cephalosporin antibiotics
US7652039B2 (en) 2002-05-17 2010-01-26 Sequella, Inc. Methods of use and compositions for the diagnosis and treatment of infectious disease
US20040033986A1 (en) 2002-05-17 2004-02-19 Protopopova Marina Nikolaevna Anti tubercular drug: compositions and methods
JP4347799B2 (ja) 2002-05-24 2009-10-21 セラヴァンス, インコーポレーテッド 架橋グリコペプチド−セファロスポリン抗生物質
WO2003106399A2 (en) 2002-06-17 2003-12-24 Theravance, Inc. PROCESS FOR PREPARING N-PROTECTED β-AMINO ALDEHYDE COMPOUNDS
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US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US6900175B2 (en) * 2002-11-18 2005-05-31 Vicuron Pharmaceuticals Inc. Methods of administering dalbavancin for treatment of bacterial infections
ATE450540T1 (de) * 2003-05-23 2009-12-15 Theravance Inc Quervernetzte glycopeptid-cephalosporin- antibiotika
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DE102004055582A1 (de) * 2004-11-18 2006-05-24 Bayer Cropscience Ag N-Heterocyclyl-phthalsäurediamide
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US7368422B2 (en) * 2005-02-28 2008-05-06 Novartis Vaccines And Diagnostics Inc. Semi-synthetic rearranged vancomycin/desmethyl-vancomycin-based glycopeptides with antibiotic activity
US7632918B2 (en) * 2005-02-28 2009-12-15 Novartis Vaccines And Diagnostics, Inc. Semi-synthetic glycopeptides with antibiotic activity
US20070185015A1 (en) * 2005-02-28 2007-08-09 Chiron Corporation and North China Pharmaceutical Corporation Semi-synthetic desmethyl-vancomycin-based glycopeptides with antibiotic activity
EP1933881B1 (en) 2005-09-22 2019-03-13 Medivas, LLC Solid polymer delivery compositions and methods for use thereof
JP5192384B2 (ja) 2005-09-22 2013-05-08 メディバス エルエルシー ビス−(α−アミノ)−ジオール−ジエステル含有ポリ(エステルアミド)およびポリ(エステルウレタン)組成物および使用の方法
US20070173438A1 (en) * 2006-01-13 2007-07-26 The Scripps Research Institute [PSI[CH2NH]PG4] glycopeptide antibiotic analogs
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
KR20100109934A (ko) 2007-12-26 2010-10-11 시오노기세야쿠 가부시키가이샤 글리코펩티드 항생 물질 배당화 유도체
EP2238102A4 (en) * 2007-12-26 2011-03-09 Lead Therapeutics Inc NEW HALF-SYNTHETIC GLYCOPEPTIDES AS ANTIBACTERIAL AGENTS
WO2009123713A1 (en) 2008-04-01 2009-10-08 Cornell University Organo-soluble chitosan salts and chitosan-derived biomaterials prepared thereof
GB2465863A (en) * 2008-12-05 2010-06-09 Lead Therapeutics Inc Semi-synthetic heptapeptidic glycopeptides for the treatment of bacterial infections
CN101928330B (zh) * 2009-06-26 2013-10-16 上海来益生物药物研究开发中心有限责任公司 一种新的化合物及其应用
WO2012129493A1 (en) * 2011-03-24 2012-09-27 Seachaid Pharmaceuticals, Inc. Vancomycin derivatives
EP3049115A1 (en) * 2013-09-23 2016-08-03 Jawaharlal Nehru Centre For Advanced Scientific Research Vancomycin-sugar conjugates and uses thereof
EP3240574A1 (en) * 2014-12-25 2017-11-08 Jawaharlal Nehru Centre For Advanced Scientific Research Glycopeptides and uses thereof
WO2017121863A1 (en) * 2016-01-15 2017-07-20 Universität Hamburg Methods for the production of rhamnosylated flavonoids
CN108698974A (zh) * 2016-01-28 2018-10-23 阿卡特肖勒公司 光裂解底漆组合物和使用方法
CN107325159A (zh) 2016-04-29 2017-11-07 中国科学院上海药物研究所 一类万古霉素衍生物、其制备方法、药物组合物和用途
IL270686B (en) * 2017-05-22 2022-09-01 Insmed Inc Derivatives of glycopeptides and their uses
CN107987131B (zh) * 2017-11-16 2021-03-09 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的化合物、其制备方法和应用
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用
NL2023883B1 (en) * 2019-09-24 2021-04-26 Univ Leiden Antibiotic compounds
CN111620931B (zh) * 2020-06-12 2021-12-17 苏州博源医疗科技有限公司 万古霉素衍生物及其制备方法和应用
CN114213284B (zh) * 2022-01-04 2023-08-01 丽珠集团福州福兴医药有限公司 (9h-芴-9-基)-癸基(2-氧代乙基)氨基甲酸甲酯及其合成方法

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Also Published As

Publication number Publication date
US8030445B2 (en) 2011-10-04
BRPI9914221B8 (pt) 2021-05-25
BR9914221A (pt) 2001-06-26
NO20006323L (no) 2001-02-12
JP2002533472A (ja) 2002-10-08
CN1315961A (zh) 2001-10-03
CZ200122A3 (en) 2001-06-13
US20040204346A1 (en) 2004-10-14
SI1140993T1 (en) 2003-12-31
HUP0400887A3 (en) 2012-09-28
US6962970B2 (en) 2005-11-08
DE69908819D1 (de) 2003-07-17
US20060241024A1 (en) 2006-10-26
US20050239690A1 (en) 2005-10-27
KR100665204B1 (ko) 2007-01-04
EP1140993B1 (en) 2003-06-11
JP4362017B2 (ja) 2009-11-11
KR20010085857A (ko) 2001-09-07
NO326066B1 (no) 2008-09-08
NZ508594A (en) 2003-05-30
PL348451A1 (en) 2002-05-20
US7723470B2 (en) 2010-05-25
HU230190B1 (hu) 2015-09-28
HUP0400887A2 (hu) 2004-08-30
PL198311B1 (pl) 2008-06-30
US6392012B1 (en) 2002-05-21
AU768204B2 (en) 2003-12-04
CA2336445C (en) 2011-07-19
CA2336445A1 (en) 2000-07-06
US6949681B2 (en) 2005-09-27
DK1140993T3 (da) 2003-10-06
NO20006323D0 (no) 2000-12-12
CZ301184B6 (cs) 2009-12-02
US7351791B2 (en) 2008-04-01
US20080103292A1 (en) 2008-05-01
ATE242783T1 (de) 2003-06-15
HK1040721B (zh) 2003-10-17
EP1140993A1 (en) 2001-10-10
CN1249081C (zh) 2006-04-05
AU3127300A (en) 2000-07-31
US20090215982A1 (en) 2009-08-27
US6455669B1 (en) 2002-09-24
US7101964B2 (en) 2006-09-05
ES2201825T3 (es) 2004-03-16
HK1040721A1 (en) 2002-06-21
DE69908819T2 (de) 2004-05-06
PT1140993E (pt) 2003-10-31
US20030060598A1 (en) 2003-03-27
IL140093A (en) 2006-06-11
US6444786B1 (en) 2002-09-03
IL140093A0 (en) 2002-02-10
BR9914221B1 (pt) 2013-12-31
WO2000039156A1 (en) 2000-07-06

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