YU315275A - Process for preparing 3-amino-indazole carboxylic acid derivatives - Google Patents

Process for preparing 3-amino-indazole carboxylic acid derivatives

Info

Publication number
YU315275A
YU315275A YU03152/75A YU315275A YU315275A YU 315275 A YU315275 A YU 315275A YU 03152/75 A YU03152/75 A YU 03152/75A YU 315275 A YU315275 A YU 315275A YU 315275 A YU315275 A YU 315275A
Authority
YU
Yugoslavia
Prior art keywords
amino
preparing
carboxylic acid
acid derivatives
indazole carboxylic
Prior art date
Application number
YU03152/75A
Other languages
English (en)
Inventor
H Mayer
S Petersen
E Klauke
F Hoffmeister
W Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of YU315275A publication Critical patent/YU315275A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
YU03152/75A 1974-12-13 1975-12-12 Process for preparing 3-amino-indazole carboxylic acid derivatives YU315275A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
YU315275A true YU315275A (en) 1982-02-28

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
YU03152/75A YU315275A (en) 1974-12-13 1975-12-12 Process for preparing 3-amino-indazole carboxylic acid derivatives

Country Status (27)

Country Link
US (1) US4051252A (hu)
JP (1) JPS5182266A (hu)
AT (1) AT343653B (hu)
BE (1) BE836528A (hu)
CA (1) CA1059523A (hu)
CH (1) CH622250A5 (hu)
CS (1) CS189731B2 (hu)
DD (1) DD125484A5 (hu)
DE (1) DE2458965C3 (hu)
DK (1) DK137082C (hu)
ES (1) ES443429A1 (hu)
FI (1) FI753493A (hu)
FR (1) FR2293928A1 (hu)
GB (1) GB1490306A (hu)
HK (1) HK52580A (hu)
HU (1) HU173557B (hu)
IE (1) IE42208B1 (hu)
IL (1) IL48642A (hu)
KE (1) KE3078A (hu)
LU (1) LU73993A1 (hu)
NL (1) NL7514521A (hu)
NO (1) NO145382C (hu)
PL (1) PL99858B1 (hu)
SE (1) SE419645B (hu)
SU (1) SU604487A3 (hu)
YU (1) YU315275A (hu)
ZA (1) ZA757777B (hu)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
EP1698627A1 (en) * 2000-09-15 2006-09-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
MXPA03002299A (es) 2000-09-15 2003-06-06 Vertex Pharma Compuestos de pirazol utiles como inhibidores de proteina cinasa.
ZA200301701B (en) * 2000-09-15 2004-03-01 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
MXPA03005605A (es) 2000-12-21 2003-10-06 Vertex Pharma Compuestos de pirazol utiles como inhibidores de la proteina cinasa.
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
CZ2004359A3 (cs) 2001-09-26 2004-09-15 Pharmacia Italia S.P.A. Aminoindazolové deriváty aktivní jako inhibitory kinázy, způsob jejich přípravy a farmaceutické prostředky obsahující tyto deriváty
SG159380A1 (en) * 2002-02-06 2010-03-30 Vertex Pharma Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
DE60332604D1 (de) 2002-03-15 2010-07-01 Vertex Pharma Azolylaminoazine als proteinkinasehemmer
WO2003097610A1 (en) 2002-05-17 2003-11-27 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
NZ550883A (en) 2002-08-02 2008-06-30 Vertex Pharma Pyrazole compositions useful as inhibitors of glycogen synthase kinase-3 (GSK-3)
AU2003270701B2 (en) * 2002-10-31 2009-11-12 Amgen Inc. Antiinflammation agents
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
WO2005056547A2 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
AU2006279376B2 (en) 2005-08-18 2011-04-14 Vertex Pharmaceuticals Incoporated Pyrazine kinase inhibitors
US7820685B2 (en) 2005-11-03 2010-10-26 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
MX2008013205A (es) * 2006-04-14 2008-10-22 Abbott Lab Procedimiento para la preparacion de indazolil ureas que inhibien receptores de vanilloides del subtipo 1 (vr1).
DE602007004750D1 (de) 2006-11-02 2010-03-25 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyridine und aminopyrimidine
NZ577768A (en) 2006-12-19 2012-01-12 Vertex Pharma Aminopyrimidines useful as inhibitors of protein kinases
NZ579483A (en) 2007-03-09 2012-07-27 Vertex Pharma Aminopyridines useful as inhibitors of protein kinases
ES2435997T3 (es) 2007-03-09 2013-12-26 Vertex Pharmaceuticals, Inc. Aminopirimidinas útiles como inhibidores de las proteínas cinasas
ES2374335T3 (es) 2007-03-09 2012-02-15 Vertex Pharmaceuticals Incorporated Aminopirimidinas útiles como inhibidores de proteína quinasas.
EP2146982A2 (en) 2007-04-13 2010-01-27 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
JP5389786B2 (ja) 2007-05-02 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害として有用なアミノピリミジン
EP2155730A2 (en) * 2007-05-02 2010-02-24 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
NZ580884A (en) * 2007-05-02 2012-02-24 Vertex Pharma Thiazoles and pyrazoles useful as kinase inhibitors
WO2008147626A2 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
EP2176261B1 (en) 2007-07-31 2012-12-19 Vertex Pharmaceuticals Incorporated Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
RU2011112802A (ru) * 2008-09-03 2012-10-10 Вертекс Фармасьютикалз Инкорпорейтед (Us) Сокристаллы и содержащие их фармацевтические композиции
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
CN104487422B (zh) 2012-07-24 2017-07-25 比亚尔-珀特拉和Ca股份公司 脲类化合物及其作为酶抑制剂的用途
US20150197503A1 (en) * 2012-07-27 2015-07-16 Bial-Portela & Cª, S.A. Process for the synthesis of substituted urea compounds
LT3024825T (lt) 2013-07-24 2017-12-11 Bial - Portela & C, S.A. Imidazolo karboksamidai ir jų panaudojimas kaip faah inhibitorių

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3274203A (en) * 1963-05-31 1966-09-20 Du Pont 1-carbamyl and thiocarbamyl-3-amino-4-nonsubstituted and substituted pyrazoles
NL6707299A (hu) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
CH622250A5 (hu) 1981-03-31
SE419645B (sv) 1981-08-17
NO145382C (no) 1982-03-10
FR2293928A1 (fr) 1976-07-09
ES443429A1 (es) 1977-04-16
NO754024L (hu) 1976-06-15
DK137082B (da) 1978-01-16
DD125484A5 (hu) 1977-04-20
DK137082C (da) 1978-06-19
LU73993A1 (hu) 1976-11-11
ZA757777B (en) 1976-11-24
GB1490306A (en) 1977-11-02
DK567275A (da) 1976-06-14
NL7514521A (nl) 1976-06-15
DE2458965A1 (de) 1976-06-16
HU173557B (hu) 1979-06-28
CA1059523A (en) 1979-07-31
CS189731B2 (en) 1979-04-30
FI753493A (hu) 1976-06-14
ATA939775A (de) 1977-10-15
IL48642A (en) 1979-12-30
DE2458965C3 (de) 1979-10-11
NO145382B (no) 1981-11-30
BE836528A (fr) 1976-06-11
IE42208L (en) 1976-06-13
DE2458965B2 (de) 1979-02-22
SU604487A3 (ru) 1978-04-25
IL48642A0 (en) 1976-02-29
HK52580A (en) 1980-09-26
JPS5182266A (en) 1976-07-19
AU8717075A (en) 1977-06-09
KE3078A (en) 1980-10-03
PL99858B1 (pl) 1978-08-31
US4051252A (en) 1977-09-27
IE42208B1 (en) 1980-06-18
AT343653B (de) 1978-06-12
SE7513990L (sv) 1976-06-14
FR2293928B1 (hu) 1979-09-21

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