DK137082B - Analogifremgangsmade til fremstilling af 3-aminoidazolcarboxylsyrederivater - Google Patents

Analogifremgangsmade til fremstilling af 3-aminoidazolcarboxylsyrederivater

Info

Publication number
DK137082B
DK137082B DK567275AA DK567275A DK137082B DK 137082 B DK137082 B DK 137082B DK 567275A A DK567275A A DK 567275AA DK 567275 A DK567275 A DK 567275A DK 137082 B DK137082 B DK 137082B
Authority
DK
Denmark
Prior art keywords
aminoidazole
preparation
carboxylic acid
acid derivatives
analogical procedure
Prior art date
Application number
DK567275AA
Other languages
English (en)
Other versions
DK567275A (da
DK137082C (da
Inventor
K H Mayer
S Petersen
E Klauke
F Hoffmeister
W Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of DK567275A publication Critical patent/DK567275A/da
Publication of DK137082B publication Critical patent/DK137082B/da
Application granted granted Critical
Publication of DK137082C publication Critical patent/DK137082C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK567275A 1974-12-13 1975-12-12 Analogifremgangsmaade til fremstilling af 3-aminoindazolcarboxylsyrederivater DK137082C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (3)

Publication Number Publication Date
DK567275A DK567275A (da) 1976-06-14
DK137082B true DK137082B (da) 1978-01-16
DK137082C DK137082C (da) 1978-06-19

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
DK567275A DK137082C (da) 1974-12-13 1975-12-12 Analogifremgangsmaade til fremstilling af 3-aminoindazolcarboxylsyrederivater

Country Status (27)

Country Link
US (1) US4051252A (da)
JP (1) JPS5182266A (da)
AT (1) AT343653B (da)
BE (1) BE836528A (da)
CA (1) CA1059523A (da)
CH (1) CH622250A5 (da)
CS (1) CS189731B2 (da)
DD (1) DD125484A5 (da)
DE (1) DE2458965C3 (da)
DK (1) DK137082C (da)
ES (1) ES443429A1 (da)
FI (1) FI753493A (da)
FR (1) FR2293928A1 (da)
GB (1) GB1490306A (da)
HK (1) HK52580A (da)
HU (1) HU173557B (da)
IE (1) IE42208B1 (da)
IL (1) IL48642A (da)
KE (1) KE3078A (da)
LU (1) LU73993A1 (da)
NL (1) NL7514521A (da)
NO (1) NO145382C (da)
PL (1) PL99858B1 (da)
SE (1) SE419645B (da)
SU (1) SU604487A3 (da)
YU (1) YU315275A (da)
ZA (1) ZA757777B (da)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
EP1698627A1 (en) * 2000-09-15 2006-09-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
ZA200301703B (en) * 2000-09-15 2004-03-02 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
JP4105949B2 (ja) 2000-09-15 2008-06-25 バーテックス ファーマシューティカルズ インコーポレイテッド プロテインキナーゼインヒビターとして有用なピラゾール化合物
PT1355905E (pt) * 2000-12-21 2007-05-31 Vertex Pharma Compostos de pirazole úteis como inibidores de proteínaquinase
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
EP1432416B1 (en) 2001-09-26 2011-01-19 Pfizer Italia S.r.l. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
EP1472245A2 (en) * 2002-02-06 2004-11-03 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
ATE468336T1 (de) 2002-03-15 2010-06-15 Vertex Pharma Azolylaminoazine als proteinkinasehemmer
MXPA04011417A (es) 2002-05-17 2005-02-14 Pharmacia Italia Spa Derivados de aminoindazol activos como inhibidores de cinasa, procedimiento para su preparacion y composiciones farmaceuticas que los comprenden.
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
EA200500299A1 (ru) 2002-08-02 2005-08-25 Вертекс Фармасьютикалз Инкорпорейтед Пиразольные композиции, используемые в качестве ингибиторов gsk-3
US7199119B2 (en) * 2002-10-31 2007-04-03 Amgen Inc. Antiinflammation agents
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
AU2004297235A1 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
EP1917259B1 (en) 2005-08-18 2012-01-25 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
WO2007056164A2 (en) 2005-11-03 2007-05-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
NZ571705A (en) * 2006-04-14 2012-03-30 Abbott Lab Process for the preparation of indazolyl ureas that inhibit vanilloid subtype 1 (VR1) receptors
JP2010509231A (ja) 2006-11-02 2010-03-25 バーテックス ファーマシューティカルズ インコーポレイテッド プロテインキナーゼの阻害剤として有用なアミノピリジンおよびアミノピリミジン
ATE474835T1 (de) 2006-12-19 2010-08-15 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyrimidine
NZ579485A (en) 2007-03-09 2012-02-24 Vertex Pharma Aminopyrimidines useful as inhibitors of protein kinases
AU2008226461A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyridines useful as inhibitors of protein kinases
CA2679884A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
AU2008240313A1 (en) 2007-04-13 2008-10-23 Aj Park Aminopyrimidines useful as kinase inhibitors
AU2008247595A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
AU2008247592A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
CN101801959A (zh) 2007-05-02 2010-08-11 沃泰克斯药物股份有限公司 可用作激酶抑制剂的氨基嘧啶类化合物
EP2164842A2 (en) * 2007-05-24 2010-03-24 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
EP2176261B1 (en) 2007-07-31 2012-12-19 Vertex Pharmaceuticals Incorporated Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
JP2012501971A (ja) * 2008-09-03 2012-01-26 バーテックス ファーマシューティカルズ インコーポレイテッド 共結晶および共結晶を含む薬学的処方物
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
UA116542C2 (uk) 2012-07-24 2018-04-10 Біал - Портела Енд Ка, С.А. Сполуки сечовини та їх застосування як інгібіторів ферментів
CN104662002A (zh) * 2012-07-27 2015-05-27 比亚尔-珀特拉和Ca股份公司 取代脲类化合物的合成方法
JP6449277B2 (ja) 2013-07-24 2019-01-09 ビアル−ポルテラ エ コンパニア，ソシエダッド アノニマ イミダゾールカルボキサミドおよびｆａａｈ阻害剤としてのそれらの使用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (da) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
ZA757777B (en) 1976-11-24
ATA939775A (de) 1977-10-15
SE419645B (sv) 1981-08-17
PL99858B1 (pl) 1978-08-31
DE2458965A1 (de) 1976-06-16
CA1059523A (en) 1979-07-31
KE3078A (en) 1980-10-03
HU173557B (hu) 1979-06-28
SU604487A3 (ru) 1978-04-25
NO145382C (no) 1982-03-10
IE42208L (en) 1976-06-13
US4051252A (en) 1977-09-27
CH622250A5 (da) 1981-03-31
NL7514521A (nl) 1976-06-15
YU315275A (en) 1982-02-28
AT343653B (de) 1978-06-12
IL48642A0 (en) 1976-02-29
CS189731B2 (en) 1979-04-30
DK567275A (da) 1976-06-14
DE2458965B2 (de) 1979-02-22
GB1490306A (en) 1977-11-02
DK137082C (da) 1978-06-19
FR2293928B1 (da) 1979-09-21
NO145382B (no) 1981-11-30
NO754024L (da) 1976-06-15
IL48642A (en) 1979-12-30
IE42208B1 (en) 1980-06-18
FR2293928A1 (fr) 1976-07-09
LU73993A1 (da) 1976-11-11
DE2458965C3 (de) 1979-10-11
AU8717075A (en) 1977-06-09
ES443429A1 (es) 1977-04-16
DD125484A5 (da) 1977-04-20
SE7513990L (sv) 1976-06-14
BE836528A (fr) 1976-06-11
HK52580A (en) 1980-09-26
FI753493A (da) 1976-06-14
JPS5182266A (en) 1976-07-19

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