NO145382C - Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater. - Google Patents

Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater.

Info

Publication number
NO145382C
NO145382C NO754024A NO754024A NO145382C NO 145382 C NO145382 C NO 145382C NO 754024 A NO754024 A NO 754024A NO 754024 A NO754024 A NO 754024A NO 145382 C NO145382 C NO 145382C
Authority
NO
Norway
Prior art keywords
amino
preparation
acid derivatives
therapeutic active
analogue procedure
Prior art date
Application number
NO754024A
Other languages
English (en)
Other versions
NO145382B (no
NO754024L (no
Inventor
Karl Heinrich Mayer
Siegfried Petersen
Erich Klauke
Friedrich Hoffmeister
Wolfgang Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO754024L publication Critical patent/NO754024L/no
Publication of NO145382B publication Critical patent/NO145382B/no
Publication of NO145382C publication Critical patent/NO145382C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
NO754024A 1974-12-13 1975-11-28 Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater. NO145382C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (3)

Publication Number Publication Date
NO754024L NO754024L (no) 1976-06-15
NO145382B NO145382B (no) 1981-11-30
NO145382C true NO145382C (no) 1982-03-10

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
NO754024A NO145382C (no) 1974-12-13 1975-11-28 Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater.

Country Status (27)

Country Link
US (1) US4051252A (no)
JP (1) JPS5182266A (no)
AT (1) AT343653B (no)
BE (1) BE836528A (no)
CA (1) CA1059523A (no)
CH (1) CH622250A5 (no)
CS (1) CS189731B2 (no)
DD (1) DD125484A5 (no)
DE (1) DE2458965C3 (no)
DK (1) DK137082C (no)
ES (1) ES443429A1 (no)
FI (1) FI753493A (no)
FR (1) FR2293928A1 (no)
GB (1) GB1490306A (no)
HK (1) HK52580A (no)
HU (1) HU173557B (no)
IE (1) IE42208B1 (no)
IL (1) IL48642A (no)
KE (1) KE3078A (no)
LU (1) LU73993A1 (no)
NL (1) NL7514521A (no)
NO (1) NO145382C (no)
PL (1) PL99858B1 (no)
SE (1) SE419645B (no)
SU (1) SU604487A3 (no)
YU (1) YU315275A (no)
ZA (1) ZA757777B (no)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
MXPA03002294A (es) * 2000-09-15 2005-09-08 Vertex Pharma Compuestos de pirazol utiles como inhibidores de proteina cinasa.
ZA200301703B (en) * 2000-09-15 2004-03-02 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
EP1345922B1 (en) 2000-12-21 2006-05-31 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
EP1432416B1 (en) 2001-09-26 2011-01-19 Pfizer Italia S.r.l. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
PL372198A1 (en) * 2002-02-06 2005-07-11 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
AU2003218215A1 (en) 2002-03-15 2003-09-29 Vertex Pharmaceuticals, Inc. Azolylaminoazines as inhibitors of protein kinases
EP1506176B1 (en) 2002-05-17 2013-04-24 Pfizer Italia S.r.l. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY141867A (en) 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
JP4733388B2 (ja) 2002-08-02 2011-07-27 バーテックス ファーマシューティカルズ インコーポレイテッド Ｇｓｋ−３のインヒビターとして有用なピラゾール組成物
AU2003270701B2 (en) * 2002-10-31 2009-11-12 Amgen Inc. Antiinflammation agents
US7601718B2 (en) 2003-02-06 2009-10-13 Vertex Pharmaceuticals Incorporated Compositions useful as inhibitors of protein kinases
CA2548172A1 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
EP1917259B1 (en) 2005-08-18 2012-01-25 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
RU2427578C2 (ru) * 2005-11-03 2011-08-27 Вертекс Фармасьютикалз Инкорпорейтед Аминопиримидины в качестве ингибиторов киназ
JP2009533474A (ja) * 2006-04-14 2009-09-17 アボット・ラボラトリーズ バニロイドサブタイプ１（ｖｒ１）受容体を阻害するインダゾリルウレアの製造方法
MX2009004807A (es) 2006-11-02 2009-06-15 Vertex Pharma Aminopiridinas y aminopirimidinas utiles como inhibidores de proteina cinasa.
MX2009006690A (es) 2006-12-19 2009-07-31 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
MX2009009592A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopiridinas utiles como inhibidores de proteinas cinasas.
RU2009137390A (ru) 2007-03-09 2011-04-20 Вертекс Фармасьютикалз Инкорпорейтед (Us) Аминопиримидины, пригодные в качестве ингибиторов протеинкиназ
WO2008112642A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
NZ580343A (en) 2007-04-13 2012-03-30 Vertex Pharma Aminopyrimidines useful as kinase inhibitors
CN101679378A (zh) 2007-05-02 2010-03-24 沃泰克斯药物股份有限公司 用作激酶抑制剂的噻唑和吡唑
JP5572087B2 (ja) * 2007-05-02 2014-08-13 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害として有用なアミノピリミジン
JP5389786B2 (ja) 2007-05-02 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害として有用なアミノピリミジン
JP2010528021A (ja) * 2007-05-24 2010-08-19 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼのインヒビターとして有用なチアゾールおよびピラゾール
MX2010001137A (es) 2007-07-31 2010-03-31 Vertex Pharma Procesopara preparar 5-fluoro-1h-pirazol[3,4-b]piridin-3-amina y derivados del mismo.
EP2323622A1 (en) * 2008-09-03 2011-05-25 Vertex Pharmaceuticals Incorporated Co-crystals and pharmaceutical formulations comprising the same
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
AR091888A1 (es) 2012-07-24 2015-03-11 Bial Portela & Ca Sa Compuestos de urea y su uso como inhibidores de enzimas
WO2014017938A2 (en) * 2012-07-27 2014-01-30 BIAL - PORTELA & Cª, S.A. Process for the synthesis of substituted urea compounds
PL3024825T3 (pl) 2013-07-24 2017-12-29 BIAL - PORTELA & Cª, S.A. Imidazolokarboksyamidy i ich zastosowanie jako inhibitorów faah

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (no) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
DK137082B (da) 1978-01-16
US4051252A (en) 1977-09-27
NO145382B (no) 1981-11-30
IE42208B1 (en) 1980-06-18
FI753493A (no) 1976-06-14
NL7514521A (nl) 1976-06-15
HK52580A (en) 1980-09-26
DK137082C (da) 1978-06-19
CH622250A5 (no) 1981-03-31
IL48642A (en) 1979-12-30
LU73993A1 (no) 1976-11-11
DE2458965A1 (de) 1976-06-16
ES443429A1 (es) 1977-04-16
ZA757777B (en) 1976-11-24
AT343653B (de) 1978-06-12
IL48642A0 (en) 1976-02-29
SE7513990L (sv) 1976-06-14
GB1490306A (en) 1977-11-02
NO754024L (no) 1976-06-15
FR2293928A1 (fr) 1976-07-09
KE3078A (en) 1980-10-03
CA1059523A (en) 1979-07-31
JPS5182266A (en) 1976-07-19
IE42208L (en) 1976-06-13
AU8717075A (en) 1977-06-09
FR2293928B1 (no) 1979-09-21
ATA939775A (de) 1977-10-15
PL99858B1 (pl) 1978-08-31
BE836528A (fr) 1976-06-11
CS189731B2 (en) 1979-04-30
SU604487A3 (ru) 1978-04-25
DE2458965B2 (de) 1979-02-22
DD125484A5 (no) 1977-04-20
HU173557B (hu) 1979-06-28
DE2458965C3 (de) 1979-10-11
SE419645B (sv) 1981-08-17
DK567275A (da) 1976-06-14
YU315275A (en) 1982-02-28

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