UY26839A1 - Productos de derivados de la 4 - fenil - piridina - Google Patents

Productos de derivados de la 4 - fenil - piridina

Info

Publication number
UY26839A1
UY26839A1 UY26839A UY26839A UY26839A1 UY 26839 A1 UY26839 A1 UY 26839A1 UY 26839 A UY26839 A UY 26839A UY 26839 A UY26839 A UY 26839A UY 26839 A1 UY26839 A1 UY 26839A1
Authority
UY
Uruguay
Prior art keywords
derivatives
piridina
fenil
products
pyridine
Prior art date
Application number
UY26839A
Other languages
English (en)
Inventor
Andrew Sleight
Torsten Hoffmann
Patrick Schnider
Sonia Mari Poli
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of UY26839A1 publication Critical patent/UY26839A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36—Opioid-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

La invención se refiere a derivados de N-óxidos de 4 - fenil - piridina y a sales de adición de ácidos farmacéuticamente aceptables de los mismos. Se ha observado que estos compuestos pueden ser utilizados como pro - fármacos para el tratamiento o la prevención de enfermedades, relacionadas al receptor de NK 1.
UY26839A 2000-07-14 2001-07-13 Productos de derivados de la 4 - fenil - piridina UY26839A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP00115287 2000-07-14

Publications (1)

Publication Number Publication Date
UY26839A1 true UY26839A1 (es) 2002-01-31

Family

ID=8169262

Family Applications (1)

Application Number Title Priority Date Filing Date
UY26839A UY26839A1 (es) 2000-07-14 2001-07-13 Productos de derivados de la 4 - fenil - piridina

Country Status (39)

Country Link
US (4) US6593472B2 (es)
EP (1) EP1303490B1 (es)
JP (1) JP3950044B2 (es)
KR (1) KR100501608B1 (es)
CN (1) CN1178917C (es)
AR (1) AR029717A1 (es)
AT (1) ATE400556T1 (es)
AU (1) AU7061901A (es)
BR (1) BRPI0112475B8 (es)
CA (1) CA2415890C (es)
CY (1) CY1108557T1 (es)
CZ (1) CZ303639B6 (es)
DE (1) DE60134749D1 (es)
DK (1) DK1303490T3 (es)
EC (1) ECSP034431A (es)
EG (1) EG24968A (es)
ES (1) ES2309075T3 (es)
GT (1) GT200100137A (es)
HK (1) HK1058198A1 (es)
HR (1) HRP20030003B1 (es)
HU (1) HU230316B1 (es)
IL (2) IL153834A0 (es)
JO (1) JO2372B1 (es)
MA (1) MA26929A1 (es)
ME (1) ME01311B (es)
MX (1) MXPA03000366A (es)
MY (1) MY154976A (es)
NO (1) NO324700B1 (es)
NZ (1) NZ523273A (es)
PA (1) PA8522001A1 (es)
PE (1) PE20020272A1 (es)
PL (1) PL205207B1 (es)
PT (1) PT1303490E (es)
RS (1) RS50932B (es)
RU (1) RU2266284C2 (es)
SI (1) SI1303490T1 (es)
UY (1) UY26839A1 (es)
WO (1) WO2002006236A1 (es)
ZA (1) ZA200210207B (es)

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Also Published As

Publication number Publication date
BRPI0112475B8 (pt) 2021-05-25
US6897226B2 (en) 2005-05-24
PL205207B1 (pl) 2010-03-31
KR100501608B1 (ko) 2005-07-18
EG24968A (en) 2011-03-14
EP1303490A1 (en) 2003-04-23
SI1303490T1 (sl) 2008-10-31
HRP20030003A2 (en) 2003-02-28
US6593472B2 (en) 2003-07-15
NO20030154D0 (no) 2003-01-13
US20040048901A1 (en) 2004-03-11
MY154976A (en) 2015-08-28
YU603A (sh) 2006-01-16
MA26929A1 (fr) 2004-12-20
PE20020272A1 (es) 2002-04-16
ECSP034431A (es) 2003-03-10
ZA200210207B (en) 2004-03-17
US6747026B2 (en) 2004-06-08
CN1178917C (zh) 2004-12-08
ATE400556T1 (de) 2008-07-15
WO2002006236A1 (en) 2002-01-24
ME01311B (me) 2013-12-20
HUP0301311A2 (hu) 2003-08-28
US20030149039A1 (en) 2003-08-07
NO324700B1 (no) 2007-12-03
NZ523273A (en) 2004-08-27
BR0112475B1 (pt) 2013-10-15
CZ303639B6 (cs) 2013-01-23
IL153834A0 (en) 2003-07-31
GT200100137A (es) 2002-05-16
CN1441782A (zh) 2003-09-10
EP1303490B1 (en) 2008-07-09
BR0112475A (pt) 2003-07-29
ES2309075T3 (es) 2008-12-16
JP3950044B2 (ja) 2007-07-25
AR029717A1 (es) 2003-07-10
MXPA03000366A (es) 2003-05-27
KR20030015387A (ko) 2003-02-20
DE60134749D1 (de) 2008-08-21
AU7061901A (en) 2002-01-30
US6806370B2 (en) 2004-10-19
PT1303490E (pt) 2008-09-04
RU2266284C2 (ru) 2005-12-20
HU230316B1 (hu) 2016-01-28
PL365684A1 (en) 2005-01-10
JO2372B1 (en) 2006-12-12
JP2004504301A (ja) 2004-02-12
RS50932B (sr) 2010-08-31
CA2415890A1 (en) 2002-01-24
CA2415890C (en) 2009-04-07
HK1058198A1 (en) 2004-05-07
IL153834A (en) 2008-11-03
NO20030154L (no) 2003-01-13
CY1108557T1 (el) 2014-04-09
US20020045642A1 (en) 2002-04-18
PA8522001A1 (es) 2002-04-25
US20040014793A1 (en) 2004-01-22
HRP20030003B1 (en) 2011-01-31
DK1303490T3 (da) 2008-08-25

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