UA85079C2 - Derivatives of n-(1,5-diphenyl-1h-pyrazol-3-yl) sulphonamide with cb1 receptor affinity - Google Patents

Derivatives of n-(1,5-diphenyl-1h-pyrazol-3-yl) sulphonamide with cb1 receptor affinity

Info

Publication number: UA85079C2
Authority: UA; Ukraine
Prior art keywords: unsubstituted; alkyl; substituted; sulphonamide; pyrazol
Prior art date: 2004-01-12

Application number

UAA200608995A

Other languages

English (en)

Inventor

Франсис Барт

Кристиан Конжи

Серж Мартинес

Мюриэлль Ринальди-Кармона

Original Assignee

Санофи-Авентис

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-01-12

Filing date

2005-01-07

Publication date

2008-12-25

2005-01-07 Application filed by Санофи-Авентис filed Critical Санофи-Авентис

2008-12-25 Publication of UA85079C2 publication Critical patent/UA85079C2/ru

Links

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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

UAA200608995A 2004-01-12 2005-01-07 Derivatives of n-(1,5-diphenyl-1h-pyrazol-3-yl) sulphonamide with cb1 receptor affinity UA85079C2 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0400257A FR2864958B1 (fr)	2004-01-12	2004-01-12	Derive de n-[(1,5-diphenyl-1h-pyrazol-3-yl)methyl] sulfonamide, leur preparation et leur application en therapeutique.

Publications (1)

Publication Number	Publication Date
UA85079C2 true UA85079C2 (en)	2008-12-25

Family

ID=34684951

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UAA200608995A UA85079C2 (en)	2004-01-12	2005-01-07	Derivatives of n-(1,5-diphenyl-1h-pyrazol-3-yl) sulphonamide with cb1 receptor affinity

Country Status (31)

Country	Link
US (1)	US7294645B2 (ru)
EP (1)	EP1720837B1 (ru)
JP (1)	JP4723514B2 (ru)
KR (1)	KR20060105050A (ru)
CN (1)	CN1910157A (ru)
AR (1)	AR047096A1 (ru)
AT (1)	ATE465995T1 (ru)
AU (1)	AU2005209441B2 (ru)
CA (1)	CA2551141C (ru)
CR (1)	CR8468A (ru)
CY (1)	CY1110651T1 (ru)
DE (1)	DE602005020907D1 (ru)
DK (1)	DK1720837T3 (ru)
EC (1)	ECSP066695A (ru)
ES (1)	ES2344850T3 (ru)
FR (1)	FR2864958B1 (ru)
HR (1)	HRP20100283T8 (ru)
IL (1)	IL176710A0 (ru)
MA (1)	MA28422B1 (ru)
NO (1)	NO20063621L (ru)
NZ (1)	NZ548442A (ru)
PL (1)	PL1720837T3 (ru)
PT (1)	PT1720837E (ru)
RS (1)	RS51365B (ru)
RU (1)	RU2366657C2 (ru)
SI (1)	SI1720837T1 (ru)
TN (1)	TNSN06203A1 (ru)
TW (1)	TWI323255B (ru)
UA (1)	UA85079C2 (ru)
WO (1)	WO2005073197A1 (ru)
ZA (1)	ZA200605657B (ru)

Families Citing this family (22)

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US7030141B2 (en) *	2001-11-29	2006-04-18	Christopher Franklin Bigge	Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade
FR2880023B1 (fr) *	2004-12-23	2007-02-23	Sanofi Aventis Sa	Derives de n-[(4,5-diphenyl-3-alkyl-2-thienyl) methyl] amine leur preparation et leur application en therapeutique
FR2880890B1 (fr) *	2005-01-19	2007-03-30	Sanofi Aventis Sa	Derives de n-[(4,5-diphenyl-2-thienyl)methyl]sulfonamide, leur preparation et leur application en therapeutique
FR2881744B1 (fr) *	2005-02-09	2007-04-27	Sanofi Aventis Sa	Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique
FR2894579B1 (fr) *	2005-12-12	2008-01-18	Sanofi Aventis Sa	Derives diaryltriazolmethylamine, leur preparation et leur application en therapeutique.
FR2894578B1 (fr) *	2005-12-12	2008-02-01	Sanofi Aventis Sa	Derives heterocycliques, leur preparation et leur application en therapeutique.
EP1829867A1 (en)	2006-03-03	2007-09-05	Laboratorios Del Dr. Esteve, S.A.	Imidazole compounds having pharmaceutical activity towards the sigma receptor
FR2899899A1 (fr) *	2006-04-14	2007-10-19	Sanofi Aventis Sa	Derives d'aminomethyl pyridine, leur preparation et leur application en therapeutique
EP1878723B1 (fr) *	2006-07-11	2010-05-26	Sanofi-Aventis	Dérivés de N-[(1,5-diphényl-1H-pyrazol-3-yl)méthyl]sulfonamide antagonistes des récepteurs CB1 des cannabinoïdes
JP2008019205A (ja) *	2006-07-12	2008-01-31	Sanofi-Aventis	Ｎ−［（１，５−ジフェニル−１ｈ−ピラゾール−３−イル）メチル］スルホンアミド誘導体、その調製法および治療におけるその応用
US7297710B1 (en) *	2006-07-12	2007-11-20	Sanofi-Aventis	Derivatives of N-[(1,5-diphenyl-1H-pyrazol-3-yl)methyl]sulfonamide, their preparation and their application in therapeutics
WO2008062424A2 (en) *	2006-07-31	2008-05-29	Cadila Healthcare Limited	Substituted 4,5-dihydro-1h-pyrazole derivatives as cannabinoid modulators
US7875647B2 (en)	2006-09-29	2011-01-25	Green Cross Corporation	Heteroaryl-pyrazole derivatives as cannabinoid CB1 receptor antagonists
EP1911747A1 (en) *	2006-10-11	2008-04-16	Laboratorios del Dr. Esteve S.A.	Sulfonamide substituted pyrazoline compounds, their preparation and use as CB1 modulators
FR2911136B1 (fr) *	2007-01-05	2009-02-20	Sanofi Aventis Sa	Derives de n-(4-cyano-1h-pyrazol-3-yl)methylamine substitues leur preparation et leur application en therapeutique.
FR2919184A1 (fr) *	2007-07-26	2009-01-30	Sanofi Aventis Sa	L'acide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4- methylpyrazole-3-carboxylique, ses esters, ses sels pharmaceutiquement acceptables et leurs solvates pour leur utilisation comme medicament.
AU2013302473B2 (en) *	2012-08-16	2017-08-10	Janssen Pharmaceutica Nv	Pyrrolopyrazoles as N-type calcium channel blockers
BR112015003393A2 (pt)	2012-08-16	2017-07-04	Janssen Pharmaceutica Nv	pirazóis substituídos como bloqueadores de canal de cálcio de tipo-n
EP2945624B1 (en) *	2013-01-17	2018-04-18	F.Hoffmann-La Roche Ag	Oxytocin receptor agonists for the treatment of cns diseases
US9453002B2 (en)	2013-08-16	2016-09-27	Janssen Pharmaceutica Nv	Substituted imidazoles as N-type calcium channel blockers
KR101685993B1 (ko)	2014-05-15	2016-12-13	한국과학기술연구원	전압개폐 칼슘이온채널 억제 활성화능을 갖는 ｎ-(피라졸릴메틸)아릴설폰아마이드 화합물 및 이를 포함하는 약학적 조성물
US20240000806A1 (en) *	2020-11-20	2024-01-04	University Of Pittsburgh - Of The Commonwealth System Of Higher Education	Methods and materials for inhibiting cb1 activity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2713225B1 (fr) *	1993-12-02	1996-03-01	Sanofi Sa	N-pipéridino-3-pyrazolecarboxamide substitué.
FR2692575B1 (fr) *	1992-06-23	1995-06-30	Sanofi Elf	Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.

2004
- 2004-01-12 FR FR0400257A patent/FR2864958B1/fr not_active Expired - Fee Related
2005
- 2005-01-07 DK DK05717379.1T patent/DK1720837T3/da active
- 2005-01-07 JP JP2006548341A patent/JP4723514B2/ja not_active Expired - Fee Related
- 2005-01-07 AU AU2005209441A patent/AU2005209441B2/en not_active Ceased
- 2005-01-07 SI SI200531060T patent/SI1720837T1/sl unknown
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- 2005-01-07 NZ NZ548442A patent/NZ548442A/en not_active IP Right Cessation
- 2005-01-07 KR KR1020067016046A patent/KR20060105050A/ko not_active Application Discontinuation
- 2005-01-07 CA CA2551141A patent/CA2551141C/fr not_active Expired - Fee Related
- 2005-01-07 AT AT05717379T patent/ATE465995T1/de active
- 2005-01-07 PT PT05717379T patent/PT1720837E/pt unknown
- 2005-01-07 WO PCT/FR2005/000031 patent/WO2005073197A1/fr active Application Filing
- 2005-01-07 ZA ZA200605657A patent/ZA200605657B/xx unknown
- 2005-01-07 RU RU2006129297/04A patent/RU2366657C2/ru not_active IP Right Cessation
- 2005-01-07 CN CNA2005800022298A patent/CN1910157A/zh active Pending
- 2005-01-07 ES ES05717379T patent/ES2344850T3/es active Active
- 2005-01-07 PL PL05717379T patent/PL1720837T3/pl unknown
- 2005-01-07 DE DE602005020907T patent/DE602005020907D1/de active Active
- 2005-01-07 EP EP05717379A patent/EP1720837B1/fr active Active
- 2005-01-07 UA UAA200608995A patent/UA85079C2/ru unknown
- 2005-01-10 AR ARP050100070A patent/AR047096A1/es unknown
- 2005-01-11 TW TW094100683A patent/TWI323255B/zh not_active IP Right Cessation
2006
- 2006-06-19 MA MA29118A patent/MA28422B1/fr unknown
- 2006-06-21 CR CR8468A patent/CR8468A/es unknown
- 2006-06-23 TN TNP2006000203A patent/TNSN06203A1/en unknown
- 2006-07-05 IL IL176710A patent/IL176710A0/en not_active IP Right Cessation
- 2006-07-06 US US11/428,928 patent/US7294645B2/en active Active
- 2006-07-11 EC EC2006006695A patent/ECSP066695A/es unknown
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2010
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Also Published As

Publication number	Publication date
AR047096A1 (es)	2006-01-04
EP1720837A1 (fr)	2006-11-15
ATE465995T1 (de)	2010-05-15
PL1720837T3 (pl)	2010-09-30
TW200535135A (en)	2005-11-01
NZ548442A (en)	2009-10-30
EP1720837B1 (fr)	2010-04-28
HRP20100283T8 (en)	2010-10-31
KR20060105050A (ko)	2006-10-09
RS51365B (en)	2011-02-28
CA2551141C (fr)	2011-06-07
MA28422B1 (fr)	2007-02-01
CR8468A (es)	2007-03-06
ECSP066695A (es)	2006-10-31
ZA200605657B (en)	2007-12-27
SI1720837T1 (sl)	2010-08-31
IL176710A0 (en)	2006-10-31
PT1720837E (pt)	2010-05-14
TNSN06203A1 (en)	2007-11-15
DK1720837T3 (da)	2010-08-23
AU2005209441A1 (en)	2005-08-11
FR2864958A1 (fr)	2005-07-15
JP4723514B2 (ja)	2011-07-13
FR2864958B1 (fr)	2006-02-24
DE602005020907D1 (de)	2010-06-10
ES2344850T3 (es)	2010-09-08
CN1910157A (zh)	2007-02-07
NO20063621L (no)	2006-10-10
US20070021486A1 (en)	2007-01-25
AU2005209441B2 (en)	2010-12-23
CA2551141A1 (fr)	2005-08-11
TWI323255B (en)	2010-04-11
CY1110651T1 (el)	2015-06-10
JP2007517839A (ja)	2007-07-05
HRP20100283T1 (hr)	2010-08-31
US7294645B2 (en)	2007-11-13
WO2005073197A1 (fr)	2005-08-11
RU2006129297A (ru)	2008-02-20
RU2366657C2 (ru)	2009-09-10

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