TW360653B - A oxadiazole compound having colon motility stimulating properties, its preparation process and its pharmaceutical composition - Google Patents
A oxadiazole compound having colon motility stimulating properties, its preparation process and its pharmaceutical compositionInfo
- Publication number
- TW360653B TW360653B TW085101860A TW85101860A TW360653B TW 360653 B TW360653 B TW 360653B TW 085101860 A TW085101860 A TW 085101860A TW 85101860 A TW85101860 A TW 85101860A TW 360653 B TW360653 B TW 360653B
- Authority
- TW
- Taiwan
- Prior art keywords
- alkyl
- hydrogen
- dioxane
- alk
- aryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP95200501 | 1995-03-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
TW360653B true TW360653B (en) | 1999-06-11 |
Family
ID=8220055
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW085101860A TW360653B (en) | 1995-03-01 | 1996-02-15 | A oxadiazole compound having colon motility stimulating properties, its preparation process and its pharmaceutical composition |
Country Status (25)
Country | Link |
---|---|
US (1) | US5854261A (zh) |
EP (1) | EP0812321B1 (zh) |
JP (1) | JP3980056B2 (zh) |
KR (1) | KR100443554B1 (zh) |
CN (1) | CN1092656C (zh) |
AR (1) | AR003932A1 (zh) |
AT (1) | ATE384716T1 (zh) |
AU (1) | AU702932B2 (zh) |
BR (1) | BR9607316A (zh) |
CA (1) | CA2212893C (zh) |
CZ (1) | CZ286992B6 (zh) |
DE (1) | DE69637412T2 (zh) |
EA (1) | EA001084B1 (zh) |
ES (1) | ES2301166T3 (zh) |
FI (1) | FI973562A (zh) |
HU (1) | HUP9702395A3 (zh) |
IL (1) | IL117315A (zh) |
MY (1) | MY113584A (zh) |
NO (1) | NO309425B1 (zh) |
NZ (1) | NZ301699A (zh) |
PL (1) | PL183712B1 (zh) |
TR (1) | TR199700876T1 (zh) |
TW (1) | TW360653B (zh) |
WO (1) | WO1996026937A1 (zh) |
ZA (1) | ZA961652B (zh) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9603755D0 (en) * | 1996-02-22 | 1996-04-24 | Pfizer Ltd | Therapeutic agents |
US6107313A (en) * | 1998-10-02 | 2000-08-22 | Combichem, Inc. | Dopamine receptor antagonists |
US7332508B2 (en) * | 2002-12-18 | 2008-02-19 | Novo Nordisk A/S | Substituted homopiperidine, piperidine or pyrrolidine derivatives |
GB0910667D0 (en) * | 2009-06-19 | 2009-08-05 | Glaxo Wellcome Mfg Pte Ltd | Novel compounds |
DK2758394T3 (en) | 2011-09-19 | 2015-04-20 | Suven Life Sciences Ltd | HETEROARYL COMPOUNDS AS 5-HT4 RECEPTOR LIGANDS |
JP2019533022A (ja) * | 2016-10-24 | 2019-11-14 | ユマニティ セラピューティクス,インコーポレーテッド | 化合物及びその使用 |
CA3083000A1 (en) | 2017-10-24 | 2019-05-02 | Yumanity Therapeutics, Inc. | Compounds and uses thereof |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1183847A (en) * | 1981-10-01 | 1985-03-12 | Georges Van Daele | N-(3-hydroxy-4-piperidinyl)benzamide derivatives |
US5374637A (en) * | 1989-03-22 | 1994-12-20 | Janssen Pharmaceutica N.V. | N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives |
GB9005014D0 (en) * | 1990-03-06 | 1990-05-02 | Janssen Pharmaceutica Nv | N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives |
US5492919A (en) * | 1991-08-03 | 1996-02-20 | Smithkline Beecham P.L.C. | 5-HT4 receptor antagonists |
GB9202797D0 (en) * | 1992-02-11 | 1992-03-25 | Milsom Jonathan | Glazed units |
US5708174A (en) * | 1992-03-12 | 1998-01-13 | Smithkline Beecham P.L.C. | Heterocyclic-esters or -amides used as 5-HT4 receptor antagonists |
MX9306311A (es) * | 1992-10-13 | 1994-04-29 | Smithkline Beecham Plc | Compuestos antagonistas del receptor de 5-ht4, procedimiento para su preparacion y composiciones farmaceuticas que los contienen |
JPH08502741A (ja) * | 1992-11-05 | 1996-03-26 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | 5−ht▲下4▼レセプターアンタゴニスト用のピペリジン誘導体 |
JPH06157518A (ja) * | 1992-11-27 | 1994-06-03 | Yamanouchi Pharmaceut Co Ltd | 新規なオキサジアゾール誘導体又はその塩 |
WO1995032965A1 (fr) * | 1994-06-01 | 1995-12-07 | Yamanouchi Pharmaceutical Co. Ltd. | Derive de l'oxadiazole et composition medicinale a base de ce dernier |
-
1996
- 1996-02-15 TW TW085101860A patent/TW360653B/zh not_active IP Right Cessation
- 1996-02-21 CA CA002212893A patent/CA2212893C/en not_active Expired - Lifetime
- 1996-02-21 BR BR9607316A patent/BR9607316A/pt not_active Application Discontinuation
- 1996-02-21 PL PL96322019A patent/PL183712B1/pl not_active IP Right Cessation
- 1996-02-21 AT AT96903000T patent/ATE384716T1/de not_active IP Right Cessation
- 1996-02-21 CZ CZ19972723A patent/CZ286992B6/cs not_active IP Right Cessation
- 1996-02-21 KR KR1019970705701A patent/KR100443554B1/ko not_active IP Right Cessation
- 1996-02-21 AU AU47188/96A patent/AU702932B2/en not_active Ceased
- 1996-02-21 NZ NZ301699A patent/NZ301699A/en not_active IP Right Cessation
- 1996-02-21 EA EA199700205A patent/EA001084B1/ru not_active IP Right Cessation
- 1996-02-21 HU HU9702395A patent/HUP9702395A3/hu unknown
- 1996-02-21 WO PCT/EP1996/000784 patent/WO1996026937A1/en active IP Right Grant
- 1996-02-21 CN CN96192300A patent/CN1092656C/zh not_active Expired - Fee Related
- 1996-02-21 DE DE69637412T patent/DE69637412T2/de not_active Expired - Lifetime
- 1996-02-21 ES ES96903000T patent/ES2301166T3/es not_active Expired - Lifetime
- 1996-02-21 US US08/894,340 patent/US5854261A/en not_active Expired - Lifetime
- 1996-02-21 EP EP96903000A patent/EP0812321B1/en not_active Expired - Lifetime
- 1996-02-21 TR TR97/00876T patent/TR199700876T1/xx unknown
- 1996-02-21 JP JP52601096A patent/JP3980056B2/ja not_active Expired - Lifetime
- 1996-02-29 IL IL11731596A patent/IL117315A/xx not_active IP Right Cessation
- 1996-02-29 ZA ZA9601652A patent/ZA961652B/xx unknown
- 1996-02-29 MY MYPI96000748A patent/MY113584A/en unknown
- 1996-02-29 AR ARP960101592A patent/AR003932A1/es unknown
-
1997
- 1997-08-19 NO NO973808A patent/NO309425B1/no not_active IP Right Cessation
- 1997-08-29 FI FI973562A patent/FI973562A/fi not_active Application Discontinuation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Annulment or lapse of patent due to non-payment of fees |