IL117315A - Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing them - Google Patents
Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL117315A IL117315A IL11731596A IL11731596A IL117315A IL 117315 A IL117315 A IL 117315A IL 11731596 A IL11731596 A IL 11731596A IL 11731596 A IL11731596 A IL 11731596A IL 117315 A IL117315 A IL 117315A
- Authority
- IL
- Israel
- Prior art keywords
- prokinetic
- preparation
- pharmaceutical compositions
- compositions containing
- oxadiazole derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP95200501 | 1995-03-01 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL117315A0 IL117315A0 (en) | 1996-06-18 |
IL117315A true IL117315A (en) | 2000-07-26 |
Family
ID=8220055
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL11731596A IL117315A (en) | 1995-03-01 | 1996-02-29 | Prokinetic piperidine substituted oxadiazole derivatives their preparation and pharmaceutical compositions containing them |
Country Status (25)
Country | Link |
---|---|
US (1) | US5854261A (xx) |
EP (1) | EP0812321B1 (xx) |
JP (1) | JP3980056B2 (xx) |
KR (1) | KR100443554B1 (xx) |
CN (1) | CN1092656C (xx) |
AR (1) | AR003932A1 (xx) |
AT (1) | ATE384716T1 (xx) |
AU (1) | AU702932B2 (xx) |
BR (1) | BR9607316A (xx) |
CA (1) | CA2212893C (xx) |
CZ (1) | CZ286992B6 (xx) |
DE (1) | DE69637412T2 (xx) |
EA (1) | EA001084B1 (xx) |
ES (1) | ES2301166T3 (xx) |
FI (1) | FI973562A0 (xx) |
HU (1) | HUP9702395A3 (xx) |
IL (1) | IL117315A (xx) |
MY (1) | MY113584A (xx) |
NO (1) | NO309425B1 (xx) |
NZ (1) | NZ301699A (xx) |
PL (1) | PL183712B1 (xx) |
TR (1) | TR199700876T1 (xx) |
TW (1) | TW360653B (xx) |
WO (1) | WO1996026937A1 (xx) |
ZA (1) | ZA961652B (xx) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9603755D0 (en) * | 1996-02-22 | 1996-04-24 | Pfizer Ltd | Therapeutic agents |
US6107313A (en) * | 1998-10-02 | 2000-08-22 | Combichem, Inc. | Dopamine receptor antagonists |
US7332508B2 (en) | 2002-12-18 | 2008-02-19 | Novo Nordisk A/S | Substituted homopiperidine, piperidine or pyrrolidine derivatives |
GB0910667D0 (en) * | 2009-06-19 | 2009-08-05 | Glaxo Wellcome Mfg Pte Ltd | Novel compounds |
MX337721B (es) | 2011-09-19 | 2016-03-16 | Suven Life Sciences Ltd | Compuestos de heteroarilo como ligandos del receptor 5-ht4. |
JP2019533022A (ja) * | 2016-10-24 | 2019-11-14 | ユマニティ セラピューティクス,インコーポレーテッド | 化合物及びその使用 |
CA3083000A1 (en) | 2017-10-24 | 2019-05-02 | Yumanity Therapeutics, Inc. | Compounds and uses thereof |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1183847A (en) * | 1981-10-01 | 1985-03-12 | Georges Van Daele | N-(3-hydroxy-4-piperidinyl)benzamide derivatives |
US5374637A (en) * | 1989-03-22 | 1994-12-20 | Janssen Pharmaceutica N.V. | N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives |
GB9005014D0 (en) * | 1990-03-06 | 1990-05-02 | Janssen Pharmaceutica Nv | N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives |
AU2363492A (en) * | 1991-08-03 | 1993-03-02 | Smithkline Beecham Plc | 5-ht4 receptor antagonists |
GB9202797D0 (en) * | 1992-02-11 | 1992-03-25 | Milsom Jonathan | Glazed units |
US5708174A (en) * | 1992-03-12 | 1998-01-13 | Smithkline Beecham P.L.C. | Heterocyclic-esters or -amides used as 5-HT4 receptor antagonists |
MX9306311A (es) * | 1992-10-13 | 1994-04-29 | Smithkline Beecham Plc | Compuestos antagonistas del receptor de 5-ht4, procedimiento para su preparacion y composiciones farmaceuticas que los contienen |
JPH08502741A (ja) * | 1992-11-05 | 1996-03-26 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | 5−ht▲下4▼レセプターアンタゴニスト用のピペリジン誘導体 |
JPH06157518A (ja) * | 1992-11-27 | 1994-06-03 | Yamanouchi Pharmaceut Co Ltd | 新規なオキサジアゾール誘導体又はその塩 |
WO1995032965A1 (fr) * | 1994-06-01 | 1995-12-07 | Yamanouchi Pharmaceutical Co. Ltd. | Derive de l'oxadiazole et composition medicinale a base de ce dernier |
-
1996
- 1996-02-15 TW TW085101860A patent/TW360653B/zh not_active IP Right Cessation
- 1996-02-21 EA EA199700205A patent/EA001084B1/ru not_active IP Right Cessation
- 1996-02-21 AT AT96903000T patent/ATE384716T1/de not_active IP Right Cessation
- 1996-02-21 ES ES96903000T patent/ES2301166T3/es not_active Expired - Lifetime
- 1996-02-21 KR KR1019970705701A patent/KR100443554B1/ko not_active IP Right Cessation
- 1996-02-21 CA CA002212893A patent/CA2212893C/en not_active Expired - Lifetime
- 1996-02-21 US US08/894,340 patent/US5854261A/en not_active Expired - Lifetime
- 1996-02-21 PL PL96322019A patent/PL183712B1/pl not_active IP Right Cessation
- 1996-02-21 AU AU47188/96A patent/AU702932B2/en not_active Ceased
- 1996-02-21 CZ CZ19972723A patent/CZ286992B6/cs not_active IP Right Cessation
- 1996-02-21 CN CN96192300A patent/CN1092656C/zh not_active Expired - Fee Related
- 1996-02-21 WO PCT/EP1996/000784 patent/WO1996026937A1/en active IP Right Grant
- 1996-02-21 BR BR9607316A patent/BR9607316A/pt not_active Application Discontinuation
- 1996-02-21 JP JP52601096A patent/JP3980056B2/ja not_active Expired - Lifetime
- 1996-02-21 EP EP96903000A patent/EP0812321B1/en not_active Expired - Lifetime
- 1996-02-21 TR TR97/00876T patent/TR199700876T1/xx unknown
- 1996-02-21 NZ NZ301699A patent/NZ301699A/en not_active IP Right Cessation
- 1996-02-21 DE DE69637412T patent/DE69637412T2/de not_active Expired - Lifetime
- 1996-02-21 HU HU9702395A patent/HUP9702395A3/hu unknown
- 1996-02-29 MY MYPI96000748A patent/MY113584A/en unknown
- 1996-02-29 IL IL11731596A patent/IL117315A/xx not_active IP Right Cessation
- 1996-02-29 AR ARP960101592A patent/AR003932A1/es unknown
- 1996-02-29 ZA ZA9601652A patent/ZA961652B/xx unknown
-
1997
- 1997-08-19 NO NO973808A patent/NO309425B1/no not_active IP Right Cessation
- 1997-08-29 FI FI973562A patent/FI973562A0/fi not_active Application Discontinuation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL116917A (en) | Piperidine derivatives and pharmaceutical compositions containing them | |
IL111002A0 (en) | Piperidine derivatives, their preparation and pharmaceutical compositions containing them | |
IL104445A0 (en) | Piperidine derivatives,their preparation and pharmaceutical compositions containing them | |
IL116851A (en) | 3-arylidene-2-oxindole derivatives and pharmaceutical compositions containing them | |
HUP9701281A2 (en) | Piperidine derivatives as neurokinin antagonists and pharmaceutical compositions containing them | |
IL117860A0 (en) | Substituted 1-phenyl-3-pyrazolecarboxamides their preparation and pharmaceutical compositions containing them | |
IL119995A0 (en) | Pyrido-fused thienyl - and furanyl-oxazolidinones their preparation and pharmaceutical compositions containing them | |
IL116486A0 (en) | Novel piperidine derivatives processes for their preparation and pharmaceutical compositions containing them | |
IL116957A0 (en) | Substituted heterocyclic compounds their preparation and pharmaceutical compositions containing them | |
HUP0003362A2 (en) | Piperidine derivatives and pharmaceutical compositions containing them | |
IL122618A0 (en) | Substituted imidazolylacetonitrile compounds their preparation and pharmaceutical compositions containing them | |
IL122293A0 (en) | Substituted 4-phenylaminothiazoles their preparation and pharmaceutical compositions containing them | |
IL119559A0 (en) | Purin -6- one derivatives their preparation and pharmaceutical compositions containing them | |
IL115905A0 (en) | Sordarin derivatives their preparation and pharmaceutical compositions containing them | |
IL118768A0 (en) | Diphenylmethylene piperidine derivatives and pharmaceutical compositions containing them | |
IL118410A0 (en) | Substituted camptothecin derivatives their preparation and pharmaceutical compositions containing them | |
IL117554A0 (en) | Imidazoquinazolines their preparation and pharmaceutical compositions containing them | |
IL122705A (en) | 2-(4-Susbstituted)-benzylamino-2-methyl-propanamide derivatives their preparation and pharmaceutical compositions containing them | |
IL117817A0 (en) | N-subsituted azaheterocyclic compounds their preparation and pharmaceutical compositions containing them | |
IL116930A (en) | 4-(1H-indol-1-YL)-1-piperidinyl derivatives their preparation and pharmaceutical compositions containing them | |
NZ234124A (en) | Piperidine derivatives and pharmaceutical compositions | |
IL109751A0 (en) | Piperidine derivatives, their preparation and pharmaceutical compositions containing them | |
ZA948689B (en) | New taxicin derivatives their preparation and pharmaceutical compositions containing them | |
IL118672A (en) | Benzisothiazolyl-substituted aminomethylchromans their preparation and pharmaceutical compositions containing them | |
IL119371A0 (en) | Sulfonylaminopyrimidines their preparation and pharmaceutical compositions containing them |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
KB | Patent renewed | ||
MM9K | Patent not in force due to non-payment of renewal fees |