SV2005002047A - " compuestos de heteroaril- y fenilsulfamoilo sustituidos " ref. pc25391a - Google Patents

" compuestos de heteroaril- y fenilsulfamoilo sustituidos " ref. pc25391a

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Publication number
SV2005002047A
SV2005002047A SV2005002047A SV2005002047A SV2005002047A SV 2005002047 A SV2005002047 A SV 2005002047A SV 2005002047 A SV2005002047 A SV 2005002047A SV 2005002047 A SV2005002047 A SV 2005002047A SV 2005002047 A SV2005002047 A SV 2005002047A
Authority
SV
El Salvador
Prior art keywords
compounds
heteroaril
cholesterol
pc25391a
fenilsulfamoil
Prior art date
Application number
SV2005002047A
Other languages
English (en)
Inventor
Ernest Seiichi Hamanaka
Jr Marcus Eugene Kehrli
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34960729&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2005002047(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SV2005002047A publication Critical patent/SV2005002047A/es

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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P13/00—Drugs for disorders of the urinary system
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    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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    • C07C323/46—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having at least one of the nitrogen atoms, not being part of nitro or nitroso groups, further bound to other hetero atoms
    • C07C323/49—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having at least one of the nitrogen atoms, not being part of nitro or nitroso groups, further bound to other hetero atoms to sulfur atoms
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
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    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

SE REFIERE A COMPUESTOS HETEROARIL- Y FENILSULFAMOILO SUSTITUIDOS A COMPOSICIONES FARMACEUTICAS QUE CONTIENEN TALES COMPUESTOS Y AL USO DE TALES COMPUESTOS COMO AGONISTAS DEL RECEPTOR ACTIVADOR DEL PROLIFERADOR DE PEROXISOMA (PPAR). LOS ACTIVADORES DE PPAR ALFA, COMPOSICIONES FARMACEUTICAS QUE CONTIENEN DICHOS COMPUESTOS Y EL USO DE DICHOS COMPUESTOS PARA ELEVAR CIERTOS NIVELES DE LIPIDOS EN PLASMA, INCLUYENDO EL COLESTEROL DE LIPOPROTEINAS DE ALTA DENSIDAD Y PARA DISMINUIR OTROS CIERTOS NIVELES DE LIPIDOS EN PLASMA, TALES COMO COLESTEROL-LDL Y TRIGLICERIDOS Y POR CONSIGUIENTE PARA TRATAR ENFERMEDADES QUE SE AGRAVAN POR BAJOS NIVELES DE COLESTEROL-HDL Y/O ALTOS NIVELES DE COLESTEROL-LDL Y TRIGLICERIDOS, TALES COMO ATEROSCLEROSIS Y ENFERMEDADES CARDIOVASCULARES, EN MAMIFEROS, INCLUYENDO SERES HUMANOS. LOS COMPUESTOS TAMBIEN SON UTILES PARA EL TRATAMIENTO DEL BALANCE ENERGETICO NEGATI VO (NEB) Y ENFERMEDADES ASOCIADAS EN RUMIANTES
SV2005002047A 2004-03-10 2005-03-10 " compuestos de heteroaril- y fenilsulfamoilo sustituidos " ref. pc25391a SV2005002047A (es)

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US11/012,139 US7262318B2 (en) 2004-03-10 2004-12-16 Substituted heteroaryl- and phenylsulfamoyl compounds

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KR20070001173A (ko) 2007-01-03
MA28461B1 (fr) 2007-03-01
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US7262318B2 (en) 2007-08-28
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AP2006003714A0 (en) 2006-08-31
DOP2005000034A (es) 2005-12-15
NL1028519C2 (nl) 2006-06-22
CA2559035A1 (en) 2005-10-06
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EA200601442A1 (ru) 2007-02-27
NO20064615L (no) 2006-12-07
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