SV2001000338A - Las 5- alquilpirido [2,3-d] pirimidinas son inhibidoras de la cinasas de tirosina y que dependen de la ciclina - Google Patents

Las 5- alquilpirido [2,3-d] pirimidinas son inhibidoras de la cinasas de tirosina y que dependen de la ciclina

Info

Publication number
SV2001000338A
SV2001000338A SV2001000338A SV2001000338A SV2001000338A SV 2001000338 A SV2001000338 A SV 2001000338A SV 2001000338 A SV2001000338 A SV 2001000338A SV 2001000338 A SV2001000338 A SV 2001000338A SV 2001000338 A SV2001000338 A SV 2001000338A
Authority
SV
El Salvador
Prior art keywords
depend
pyrimidines
inhibitors
alkylpiride
cyclone
Prior art date
Application number
SV2001000338A
Other languages
English (en)
Inventor
Richard John Booth
Ellen Myra Dobrusin
Peter Laurence Toogood
Scott Norman Vanderwel
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of SV2001000338A publication Critical patent/SV2001000338A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

ESTA INVENCIÓN SE REFIERE A 5-ALQUILPIRIDOPIRIMIDINAS COMO INHIBIDORES DE LAS CINASAS QUE DEPENDEN DE LA CICLINA, EN PARTICULAR DE LA CINASAS 4 QUE DEPENDEN DE LA CICLINA. LOS COMPUESTOS DE LA INVENCION SON UTILES PARA EL TRATAMIENTO DE LA INFLAMACION, LAS ENFERMEDADES PROLIFERATIVAS DE LAS CELULAS COMO EL CANCER Y LA RESTENOSIS, Y LAS ENFERMEDADES NEURODEGENERATIVAS, COMO LA ENFERMEDAD DE ALZHEIMER.
SV2001000338A 2000-03-06 2001-03-05 Las 5- alquilpirido [2,3-d] pirimidinas son inhibidoras de la cinasas de tirosina y que dependen de la ciclina SV2001000338A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18712400P 2000-03-06 2000-03-06

Publications (1)

Publication Number Publication Date
SV2001000338A true SV2001000338A (es) 2001-11-30

Family

ID=22687699

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2001000338A SV2001000338A (es) 2000-03-06 2001-03-05 Las 5- alquilpirido [2,3-d] pirimidinas son inhibidoras de la cinasas de tirosina y que dependen de la ciclina

Country Status (36)

Country Link
EP (1) EP1268476A1 (es)
JP (1) JP2003528101A (es)
KR (1) KR20020075805A (es)
CN (1) CN1422268A (es)
AP (1) AP2002002643A0 (es)
AR (1) AR034119A1 (es)
AU (1) AU2001233028A1 (es)
BG (1) BG107161A (es)
BR (1) BR0109056A (es)
CA (1) CA2401368A1 (es)
CO (1) CO5280200A1 (es)
CR (1) CR6736A (es)
CZ (1) CZ20022929A3 (es)
DZ (1) DZ3308A1 (es)
EA (1) EA200200802A1 (es)
EE (1) EE200200506A (es)
GT (1) GT200100037A (es)
HN (1) HN2001000040A (es)
HR (1) HRP20020798A2 (es)
HU (1) HUP0300136A2 (es)
IL (1) IL151480A0 (es)
IS (1) IS6524A (es)
MA (1) MA26881A1 (es)
MX (1) MXPA02008535A (es)
NO (1) NO20024235L (es)
NZ (1) NZ520962A (es)
OA (1) OA12227A (es)
PA (1) PA8513201A1 (es)
PE (1) PE20011177A1 (es)
PL (1) PL358271A1 (es)
SK (1) SK12472002A3 (es)
SV (1) SV2001000338A (es)
TN (1) TNSN01036A1 (es)
WO (1) WO2001070741A1 (es)
YU (1) YU66502A (es)
ZA (1) ZA200207110B (es)

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Also Published As

Publication number Publication date
PA8513201A1 (es) 2003-06-30
AU2001233028A1 (en) 2001-10-03
BG107161A (en) 2003-06-30
NZ520962A (en) 2003-09-26
WO2001070741A1 (en) 2001-09-27
CZ20022929A3 (cs) 2003-02-12
IS6524A (is) 2002-08-23
CN1422268A (zh) 2003-06-04
AP2002002643A0 (en) 2002-12-31
MA26881A1 (fr) 2004-12-20
HN2001000040A (es) 2001-09-06
TNSN01036A1 (en) 2005-11-10
SK12472002A3 (sk) 2003-04-01
NO20024235D0 (no) 2002-09-05
NO20024235L (no) 2002-11-05
MXPA02008535A (es) 2002-12-13
HUP0300136A2 (en) 2003-05-28
GT200100037A (es) 2002-03-04
PL358271A1 (en) 2004-08-09
YU66502A (sh) 2005-09-19
IL151480A0 (en) 2003-04-10
BR0109056A (pt) 2003-06-03
KR20020075805A (ko) 2002-10-05
CO5280200A1 (es) 2003-05-30
EA200200802A1 (ru) 2003-02-27
EP1268476A1 (en) 2003-01-02
EE200200506A (et) 2004-02-16
DZ3308A1 (fr) 2001-09-27
OA12227A (en) 2004-03-18
ZA200207110B (en) 2003-12-04
PE20011177A1 (es) 2001-11-23
CA2401368A1 (en) 2001-09-27
CR6736A (es) 2004-03-10
AR034119A1 (es) 2004-02-04
HRP20020798A2 (en) 2004-02-29
JP2003528101A (ja) 2003-09-24

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