SU695558A3 - Способ получени производных 5-ароил1,2-дигидро-3н-пиррол(1,2-а)-пиррол-1карбоновой кислоты или их солей - Google Patents

Способ получени производных 5-ароил1,2-дигидро-3н-пиррол(1,2-а)-пиррол-1карбоновой кислоты или их солей

Info

Publication number: SU695558A3
Authority: SU; USSR - Soviet Union
Prior art keywords: pyrrole; dihydro; carboxylate; methyl; carboxylic acid
Prior art date: 1976-07-14

Application number

SU772501050A

Other languages

English (en)

Russian (ru)

Inventor

М.Маковски Джозеф

Ф.Клюге Артур

Original Assignee

Синтекс (Ю.С.А.) Инк (Фирма)

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1977-07-13

Publication date

1979-10-30

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SU695558(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1977-02-23 Priority claimed from US05/771,286 external-priority patent/US4089969A/en

1977-07-13 Application filed by Синтекс (Ю.С.А.) Инк (Фирма) filed Critical Синтекс (Ю.С.А.) Инк (Фирма)

1979-10-30 Application granted granted Critical

1979-10-30 Publication of SU695558A3 publication Critical patent/SU695558A3/ru

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Rheumatology (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)

SU772501050A 1976-07-14 1977-07-13 Способ получени производных 5-ароил1,2-дигидро-3н-пиррол(1,2-а)-пиррол-1карбоновой кислоты или их солей SU695558A3 (ru)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70490976A	1976-07-14	1976-07-14
US05/771,286 US4089969A (en)	1976-07-14	1977-02-23	5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (1)

Publication Number	Publication Date
SU695558A3 true SU695558A3 (ru)	1979-10-30

Family

ID=27107410

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SU772501050A SU695558A3 (ru)	1976-07-14	1977-07-13	Способ получени производных 5-ароил1,2-дигидро-3н-пиррол(1,2-а)-пиррол-1карбоновой кислоты или их солей

Country Status (27)

Country	Link
JP (1)	JPS539788A (xx)
AR (1)	AR224997A1 (xx)
CA (1)	CA1102809A (xx)
CH (3)	CH641458A5 (xx)
CS (1)	CS204954B2 (xx)
DE (2)	DE2731678A1 (xx)
DK (1)	DK151886C (xx)
ES (2)	ES460706A1 (xx)
FI (1)	FI63406C (xx)
FR (2)	FR2358406A1 (xx)
GB (1)	GB1554075A (xx)
GR (1)	GR61111B (xx)
HK (1)	HK15981A (xx)
HU (1)	HU174224B (xx)
IE (1)	IE45253B1 (xx)
IL (2)	IL52493A (xx)
IT (1)	IT1117313B (xx)
MX (1)	MX163202B (xx)
MY (1)	MY8100357A (xx)
NL (2)	NL186318C (xx)
NO (1)	NO147564C (xx)
NZ (1)	NZ184610A (xx)
PL (4)	PL124444B1 (xx)
PT (1)	PT66780B (xx)
SE (1)	SE434643B (xx)
SU (1)	SU695558A3 (xx)
YU (1)	YU40816B (xx)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4140698A (en) *	1977-07-25	1979-02-20	Syntex (Usa) Inc.	1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) *	1979-03-19	1980-09-25	Sohachi Takeuchi	Manufacturing method of tubular vessel
US4344943A (en) *	1980-06-09	1982-08-17	Syntex (U.S.A.) Inc.	6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) *	1980-11-21	1982-10-12	Syntex (U.S.A.) Inc.	Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
JPS5910589A (ja) *	1982-06-10	1984-01-20	メルク　エンド　カムパニー　インコーポレーテツド	抗炎症剤および鎮痛剤として新規な５−（ピロ−ル−２−オイル）−１，２−ジヒドロ−３Ｈ−ピロロ〔１，２−ａ〕ピロ−ル誘導体
US4511724A (en) *	1982-06-10	1985-04-16	Merck & Co., Inc.	5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
US4874871A (en) *	1987-03-25	1989-10-17	Syntex (U.S.A.) Inc.	Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (ja) *	1987-09-10	1995-05-01	久光製薬株式会社	新規な３−アロイル−６，７−ジヒドロ−５Ｈ−ピロロ〔１，２−ｃ〕イミダゾール−７−カルボン酸誘導体
JP2649168B2 (ja) *	1988-02-25	1997-09-03	久光製薬株式会社	新規な５，６−ジフェニル−１，２−ジヒドロ−３Ｈ−ピロロ［１，２−ａ］ピロール−１−カルボン酸誘導体
IT1250691B (it) *	1991-07-22	1995-04-21	Giancarlo Santus	Composizioni terapeutiche per somministrazione intranasale comprendenti ketorolac.
DK0612521T3 (da) *	1991-11-11	2000-01-17	Hisamitsu Pharmaceutical Co	Keterolacholdigt varmt omslag
DE4300697C1 (de) *	1993-01-13	1994-05-19	Roemmers Sa	Keterolac-Derivat mit wesentlich geringerer gastrointestinaler Reizung und Ulzeration
US5622948A (en) *	1994-12-01	1997-04-22	Syntex (U.S.A.) Inc.	Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (ja) *	2007-02-27	2008-09-11	Okamura Corp	商品陳列棚における照明装置

1977
- 1977-05-17 JP JP5697777A patent/JPS539788A/ja active Granted
- 1977-07-07 DK DK307577A patent/DK151886C/da active
- 1977-07-07 AR AR268356A patent/AR224997A1/es active
- 1977-07-07 GR GR53907A patent/GR61111B/el unknown
- 1977-07-08 IL IL52493A patent/IL52493A/xx unknown
- 1977-07-08 NL NLAANVRAGE7707651,A patent/NL186318C/xx not_active IP Right Cessation
- 1977-07-08 CH CH850077A patent/CH641458A5/de not_active IP Right Cessation
- 1977-07-08 PT PT66780A patent/PT66780B/pt unknown
- 1977-07-08 IE IE1423/77A patent/IE45253B1/en not_active IP Right Cessation
- 1977-07-11 NZ NZ184610A patent/NZ184610A/xx unknown
- 1977-07-11 YU YU1721/77A patent/YU40816B/xx unknown
- 1977-07-11 FR FR7721356A patent/FR2358406A1/fr active Granted
- 1977-07-11 FI FI772153A patent/FI63406C/fi not_active IP Right Cessation
- 1977-07-11 GB GB28919/77A patent/GB1554075A/en not_active Expired
- 1977-07-12 CS CS774646A patent/CS204954B2/cs unknown
- 1977-07-12 CA CA282,599A patent/CA1102809A/en not_active Expired
- 1977-07-13 IT IT68630/77A patent/IT1117313B/it active Protection Beyond IP Right Term
- 1977-07-13 PL PL1977227290A patent/PL124444B1/pl unknown
- 1977-07-13 ES ES460706A patent/ES460706A1/es not_active Expired
- 1977-07-13 PL PL1977227291A patent/PL124445B1/pl unknown
- 1977-07-13 DE DE19772731678 patent/DE2731678A1/de active Granted
- 1977-07-13 SE SE7708141A patent/SE434643B/xx not_active IP Right Cessation
- 1977-07-13 NO NO772494A patent/NO147564C/no unknown
- 1977-07-13 SU SU772501050A patent/SU695558A3/ru active
- 1977-07-13 DE DE2760330A patent/DE2760330C2/de not_active Expired
- 1977-07-13 PL PL1977227289A patent/PL124711B1/pl unknown
- 1977-07-13 PL PL1977199603A patent/PL109390B1/pl unknown
- 1977-07-14 HU HU77SI1582A patent/HU174224B/hu unknown
- 1977-12-20 FR FR7738508A patent/FR2375234A1/fr active Granted
1978
- 1978-05-24 ES ES470214A patent/ES470214A1/es not_active Expired
1979
- 1979-11-22 IL IL58779A patent/IL58779A0/xx unknown
1981
- 1981-04-23 HK HK159/81A patent/HK15981A/xx unknown
- 1981-12-30 MY MY357/81A patent/MY8100357A/xx unknown
1984
- 1984-02-22 CH CH86684A patent/CH646973A5/de not_active IP Right Cessation
- 1984-02-22 CH CH86584A patent/CH646972A5/de not_active IP Right Cessation
1991
- 1991-07-05 MX MX9100104A patent/MX163202B/es unknown
1993
- 1993-03-23 NL NL930021C patent/NL930021I2/nl unknown

Also Published As

Publication number	Publication date
NO772494L (no)	1978-01-17
AU513384B2 (en)	1980-11-27
IL52493A (en)	1982-02-28
DE2731678C2 (xx)	1989-06-08
DK151886C (da)	1988-06-06
NZ184610A (en)	1979-03-28
NL186318C (nl)	1990-11-01
MY8100357A (en)	1981-12-31
GR61111B (en)	1978-09-12
ES470214A1 (es)	1979-09-16
FI63406B (fi)	1983-02-28
NL7707651A (nl)	1978-01-17
PL124444B1 (en)	1983-01-31
MX163202B (es)	1992-02-20
AR224997A1 (es)	1982-02-15
JPS539788A (en)	1978-01-28
IE45253B1 (en)	1982-07-14
DE2760330C2 (xx)	1989-06-15
IL52493A0 (en)	1977-10-31
JPS6254109B2 (xx)	1987-11-13
GB1554075A (en)	1979-10-17
CH641458A5 (en)	1984-02-29
NO147564C (no)	1983-05-18
NO147564B (no)	1983-01-24
HU174224B (hu)	1979-11-28
PL124711B1 (en)	1983-02-28
YU172177A (en)	1983-09-30
DK151886B (da)	1988-01-11
CH646973A5 (en)	1984-12-28
CA1102809A (en)	1981-06-09
AU2697577A (en)	1979-01-18
FI63406C (fi)	1983-06-10
FR2358406B1 (xx)	1981-04-17
YU40816B (en)	1986-06-30
SE434643B (sv)	1984-08-06
CH646972A5 (en)	1984-12-28
FR2358406A1 (fr)	1978-02-10
FI772153A (xx)	1978-01-15
CS204954B2 (en)	1981-04-30
PT66780A (fr)	1977-08-01
HK15981A (en)	1981-05-01
PL124445B1 (en)	1983-01-31
PT66780B (fr)	1978-12-18
DE2731678A1 (de)	1978-03-16
FR2375234B1 (xx)	1980-11-07
DK307577A (da)	1978-01-15
NL930021I2 (nl)	1997-03-03
NL186318B (nl)	1990-06-01
ES460706A1 (es)	1978-12-01
IL58779A0 (en)	1980-02-29
NL930021I1 (nl)	1993-05-03
FR2375234A1 (fr)	1978-07-21
IT1117313B (it)	1986-02-17
SE7708141L (sv)	1978-01-15
PL199603A1 (pl)	1978-04-24
PL109390B1 (en)	1980-05-31
IE45253L (en)	1978-01-14

Publication	Publication Date	Title
SU695558A3 (ru)	1979-10-30	Способ получени производных 5-ароил1,2-дигидро-3н-пиррол(1,2-а)-пиррол-1карбоновой кислоты или их солей
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EP0053021B1 (en)	1985-05-02	Process for 5-aroylation of 1,2-dihydro-3h-pyrrolo(1,2-a)pyrrole-1-carboxylic esters and nitriles
EP0454121B1 (en)	1996-11-13	Azatetracyclic compounds
JPH07500349A (ja)	1995-01-12	キノリン抗生物質の合成における中間体の製造
JPH08319290A (ja)	1996-12-03	イミダゾール誘導体
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EP0019788A2 (en)	1980-12-10	Novel process for the manufacture of thiophene derivatives suited for the manufacture of biotin, process for the manufacture of biotin and novel intermediates in this process
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