SK284103B6 - 3-Substituované deriváty 3H-2,3-benzodiazepínu, spôsob ich výroby, ich použitie v liečivách a farmaceutický prostriedok tieto látky obsahujúci - Google Patents

3-Substituované deriváty 3H-2,3-benzodiazepínu, spôsob ich výroby, ich použitie v liečivách a farmaceutický prostriedok tieto látky obsahujúci Download PDF

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Publication number
SK284103B6
SK284103B6 SK135-97A SK13597A SK284103B6 SK 284103 B6 SK284103 B6 SK 284103B6 SK 13597 A SK13597 A SK 13597A SK 284103 B6 SK284103 B6 SK 284103B6
Authority
SK
Slovakia
Prior art keywords
carbon atoms
group
optionally substituted
alkanoyl
alkyl
Prior art date
Application number
SK135-97A
Other languages
English (en)
Slovak (sk)
Other versions
SK13597A3 (en
Inventor
Tam�S H�Mori
Istv�N Tarnawa
S�Ndor S�Lyom
P�L Berzsenyi
Erzs�Bet Birk�S Falgin�
Ferenc Andr�Si
Istv�N Ling
Tibor Hask
G�Bor Kapus
Emese Csuzdi
M�Rta Sz�Ll�Sy
Franciska Erd� Vid�N�
Antal Simay
G�Bor Z�Lyomi
Original Assignee
Schering Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Aktiengesellschaft filed Critical Schering Aktiengesellschaft
Publication of SK13597A3 publication Critical patent/SK13597A3/sk
Publication of SK284103B6 publication Critical patent/SK284103B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A61P39/02—Antidotes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
SK135-97A 1994-08-01 1995-07-28 3-Substituované deriváty 3H-2,3-benzodiazepínu, spôsob ich výroby, ich použitie v liečivách a farmaceutický prostriedok tieto látky obsahujúci SK284103B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4428835A DE4428835A1 (de) 1994-08-01 1994-08-01 Neue 3-substituierte 3H-2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel
PCT/DE1995/001029 WO1996004283A1 (de) 1994-08-01 1995-07-28 Neue 3-substituierte 3h-2,3-benzodiazepinderivate, deren herstellung und verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
SK13597A3 SK13597A3 (en) 1997-07-09
SK284103B6 true SK284103B6 (sk) 2004-09-08

Family

ID=6525693

Family Applications (1)

Application Number Title Priority Date Filing Date
SK135-97A SK284103B6 (sk) 1994-08-01 1995-07-28 3-Substituované deriváty 3H-2,3-benzodiazepínu, spôsob ich výroby, ich použitie v liečivách a farmaceutický prostriedok tieto látky obsahujúci

Country Status (21)

Country Link
US (1) US5756495A (fi)
EP (1) EP0775143B1 (fi)
JP (1) JPH10504543A (fi)
KR (1) KR100386709B1 (fi)
CN (1) CN1048728C (fi)
AT (1) ATE223415T1 (fi)
AU (1) AU693241B2 (fi)
CA (1) CA2195747C (fi)
CZ (1) CZ291276B6 (fi)
DE (2) DE4428835A1 (fi)
DK (1) DK0775143T3 (fi)
ES (1) ES2181787T3 (fi)
FI (1) FI113177B (fi)
HU (1) HU225500B1 (fi)
MX (1) MX9700813A (fi)
NO (1) NO319151B1 (fi)
NZ (1) NZ290777A (fi)
PT (1) PT775143E (fi)
RU (1) RU2146678C1 (fi)
SK (1) SK284103B6 (fi)
WO (1) WO1996004283A1 (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP9701325A1 (hu) 1997-07-31 2000-08-28 Gyógyszerkutató Intézet Kft. Új 2,3-benzodiazepin-származékok
BR9812119A (pt) * 1997-08-12 2004-06-22 Egyt Gyogyszervegyeszeti Gyar Derivados de 1,3-dioxolo/4, 5-h//2,3/benzodiazepina, processo para a preparação dos mesmos e composição farmacêutica
UA67749C2 (uk) 1997-08-12 2004-07-15 Егіш Дьйодьсердьяр Рт. Похідна 8-заміщеного-9н-1,3-діоксол/4,5-h//2,3/бензодіазепіну з властивостями амра/каїнатного антагоніста, спосіб одержання похідних, фармацевтична композиція (варіанти), спосіб її одержання та спосіб лікування
HU227128B1 (en) * 1999-07-07 2010-07-28 Egyt Gyogyszervegyeszeti Gyar New 2,3-benzodiazepine derivatives
NO320473B1 (no) * 2002-09-09 2005-12-12 Norsk Hydro As Anordning ved separator for separasjon av flerfasefluid.
US6858605B2 (en) * 2003-02-04 2005-02-22 Ivax Drug Research Institute, Ltd. Substituted 2,3-benzodiazepine derivatives
GB0405034D0 (en) * 2004-03-05 2004-04-07 Novartis Ag Organic compounds
RS51822B (en) * 2005-04-04 2012-02-29 Eisai R. &D. Management Co. Ltd. DIHYDROPYRIDINE COMPOUNDS FOR TREATMENT OF NEURODEGENERATIVE DISEASES AND Dementia
KR101476591B1 (ko) * 2005-09-09 2014-12-24 노파르티스 아게 자가면역성 질환의 치료
WO2015121268A1 (de) * 2014-02-14 2015-08-20 Bayer Pharma Aktiengesellschaft 1-phenyl-3h-2,3-benzodiazepine und ihre verwendung als bromodomänen-inhibitoren

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU219778B (hu) * 1990-12-21 2001-07-30 Gyógyszerkutató Intézet Közös Vállalat Eljárás N-acil-2,3-benzodiazepin-származékok, savaddíciós sóik és az ezeket tartalmazó gyógyászati készítmények előállítására, valamint a vegyületek egy csoportja, és az ezeket tartalmazó gyógyászati készítmények

Also Published As

Publication number Publication date
EP0775143A1 (de) 1997-05-28
DK0775143T3 (da) 2002-12-02
MX9700813A (es) 1997-05-31
WO1996004283A1 (de) 1996-02-15
NO970435L (no) 1997-01-31
US5756495A (en) 1998-05-26
AU693241B2 (en) 1998-06-25
RU2146678C1 (ru) 2000-03-20
ATE223415T1 (de) 2002-09-15
FI113177B (fi) 2004-03-15
JPH10504543A (ja) 1998-05-06
SK13597A3 (en) 1997-07-09
ES2181787T3 (es) 2003-03-01
CA2195747C (en) 2006-01-24
NO319151B1 (no) 2005-06-27
DE59510364D1 (de) 2002-10-10
CN1048728C (zh) 2000-01-26
CZ291276B6 (cs) 2003-01-15
NZ290777A (en) 1998-07-28
FI970434A (fi) 1997-01-31
HUT76801A (en) 1997-11-28
NO970435D0 (no) 1997-01-31
CN1155285A (zh) 1997-07-23
HU225500B1 (en) 2007-01-29
DE4428835A1 (de) 1996-02-08
PT775143E (pt) 2003-01-31
CZ15997A3 (en) 1997-06-11
KR100386709B1 (ko) 2003-08-19
FI970434A0 (fi) 1997-01-31
CA2195747A1 (en) 1996-02-15
EP0775143B1 (de) 2002-09-04
AU3160995A (en) 1996-03-04

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