SK281752B6 - Spôsob prípravy 3-{2-[4-(6-fluórbenzo[d]izoxazol-3-yl)piperidin- 1-yl]etyl}-2-metyl-6,7,8,9-tetrahydro-4h- pyridol[1,2-a]pyrimidin-4-ónu a medziprodukty tohto spôsobu - Google Patents

Spôsob prípravy 3-{2-[4-(6-fluórbenzo[d]izoxazol-3-yl)piperidin- 1-yl]etyl}-2-metyl-6,7,8,9-tetrahydro-4h- pyridol[1,2-a]pyrimidin-4-ónu a medziprodukty tohto spôsobu Download PDF

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Publication number
SK281752B6
SK281752B6 SK156-95A SK15695A SK281752B6 SK 281752 B6 SK281752 B6 SK 281752B6 SK 15695 A SK15695 A SK 15695A SK 281752 B6 SK281752 B6 SK 281752B6
Authority
SK
Slovakia
Prior art keywords
formula
tetrahydro
pyrimidin
methyl
pyrido
Prior art date
Application number
SK156-95A
Other languages
English (en)
Slovak (sk)
Other versions
SK15695A3 (en
Inventor
Barjoan Pere Dalmases
Olondriz Francisco Marquillas
Clotet Joan Huguet
Rovira Ana Bosch
Castillo Nieto Juan Carlos Del
Ges José María Caldero
Original Assignee
Vita-Invest, S. A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita-Invest, S. A. filed Critical Vita-Invest, S. A.
Publication of SK15695A3 publication Critical patent/SK15695A3/sk
Publication of SK281752B6 publication Critical patent/SK281752B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SK156-95A 1994-02-11 1995-02-07 Spôsob prípravy 3-{2-[4-(6-fluórbenzo[d]izoxazol-3-yl)piperidin- 1-yl]etyl}-2-metyl-6,7,8,9-tetrahydro-4h- pyridol[1,2-a]pyrimidin-4-ónu a medziprodukty tohto spôsobu SK281752B6 (sk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09400252A ES2074966B1 (es) 1994-02-11 1994-02-11 Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona.

Publications (2)

Publication Number Publication Date
SK15695A3 SK15695A3 (en) 1995-10-11
SK281752B6 true SK281752B6 (sk) 2001-07-10

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
SK156-95A SK281752B6 (sk) 1994-02-11 1995-02-07 Spôsob prípravy 3-{2-[4-(6-fluórbenzo[d]izoxazol-3-yl)piperidin- 1-yl]etyl}-2-metyl-6,7,8,9-tetrahydro-4h- pyridol[1,2-a]pyrimidin-4-ónu a medziprodukty tohto spôsobu

Country Status (14)

Country Link
KR (1) KR100221108B1 (is)
AT (1) AT405401B (is)
CZ (1) CZ286398B6 (is)
EG (1) EG20877A (is)
ES (1) ES2074966B1 (is)
FI (1) FI110000B (is)
GR (1) GR1002344B (is)
HU (1) HU222110B1 (is)
IS (1) IS1766B (is)
NO (1) NO306022B1 (is)
PL (1) PL181420B1 (is)
PT (1) PT101654B (is)
RU (1) RU2123004C1 (is)
SK (1) SK281752B6 (is)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (es) * 1995-04-12 1998-04-01 Ferrer Int Nuevo compuesto derivado del cromeno.
ES2144355B1 (es) * 1997-12-30 2001-01-01 Ferrer Int Compuestos derivados del cromeno.
ATE264329T1 (de) * 2000-05-05 2004-04-15 Rpg Life Sciences Ltd Verfahren zur herstellung von antipsychotischem 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-
PT1783118E (pt) 2000-08-14 2008-08-19 Teva Pharma Preparação de risperidona
KR20040034996A (ko) 2002-10-18 2004-04-29 한미약품 주식회사 리스페리돈의 개선된 제조방법
EP1560814A1 (en) 2002-11-13 2005-08-10 Synthon B.V. Process for making risperidone and intermediates therefor
DK2154138T3 (en) * 2007-04-19 2015-11-02 Youxin Li Novel compounds for the treatment of psychotic disorders, methods of preparation and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
AT405401B (de) 1999-08-25
NO950501L (no) 1995-08-14
HU222110B1 (hu) 2003-04-28
CZ286398B6 (en) 2000-04-12
NO306022B1 (no) 1999-09-06
SK15695A3 (en) 1995-10-11
ES2074966B1 (es) 1996-06-16
PT101654B (pt) 2002-01-30
ES2074966A1 (es) 1995-09-16
EG20877A (en) 2000-05-31
FI950579A0 (fi) 1995-02-10
KR100221108B1 (ko) 1999-09-15
PL307200A1 (en) 1995-08-21
RU2123004C1 (ru) 1998-12-10
HUT70169A (en) 1995-09-28
RU95101859A (ru) 1997-03-20
IS4259A (is) 1995-08-12
HU9500418D0 (en) 1995-03-28
CZ32995A3 (en) 1995-09-13
NO950501D0 (no) 1995-02-09
FI950579A (fi) 1995-08-12
KR950032196A (ko) 1995-12-20
FI110000B (fi) 2002-11-15
GR1002344B (el) 1996-05-24
PL181420B1 (pl) 2001-07-31
ATA24995A (de) 1998-12-15
PT101654A (pt) 1995-09-12
IS1766B (is) 2001-03-15

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Legal Events

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MM4A Patent lapsed due to non-payment of maintenance fees

Effective date: 20110207