RS50720B - 3,11 b-cis-dihidrotetrabenazin za lečenje proliferativne bolesti ili inflamacije - Google Patents

3,11 b-cis-dihidrotetrabenazin za lečenje proliferativne bolesti ili inflamacije

Info

Publication number
RS50720B
RS50720B RSP-2009/0015A RSP20090015A RS50720B RS 50720 B RS50720 B RS 50720B RS P20090015 A RSP20090015 A RS P20090015A RS 50720 B RS50720 B RS 50720B
Authority
RS
Serbia
Prior art keywords
treatment
dihydrotetrabenzine
cis
inflammation
proliferative disease
Prior art date
Application number
RSP-2009/0015A
Other languages
English (en)
Inventor
Jean Elisabeth Yarrow
Andrew John Duffield
Original Assignee
Biovail Laboratories International (Barbados) Srl.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biovail Laboratories International (Barbados) Srl. filed Critical Biovail Laboratories International (Barbados) Srl.
Publication of RS50720B publication Critical patent/RS50720B/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Jedinjenje 3,1 lb-m-dihidrotetrabenazina formule (Ia):ili njegove farmaceutski prihvatljive soli, za profilaksu ili lečenje inflamatorne bolesti.Prijava sadrži još 9 patentnih zahteva.
RSP-2009/0015A 2005-08-05 2006-08-04 3,11 b-cis-dihidrotetrabenazin za lečenje proliferativne bolesti ili inflamacije RS50720B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0516168.2A GB0516168D0 (en) 2005-08-05 2005-08-05 Pharmaceutical compounds
PCT/GB2006/002909 WO2007017643A1 (en) 2005-08-05 2006-08-04 3 , llB-CIS-DIHYDROTETRABENAZINE FOR THE TREATMENT OF A PROLIFERATIVE DISEASE OR AN INFLAMMATION

Publications (1)

Publication Number Publication Date
RS50720B true RS50720B (sr) 2010-08-31

Family

ID=34984180

Family Applications (1)

Application Number Title Priority Date Filing Date
RSP-2009/0015A RS50720B (sr) 2005-08-05 2006-08-04 3,11 b-cis-dihidrotetrabenazin za lečenje proliferativne bolesti ili inflamacije

Country Status (24)

Country Link
US (1) US20090275605A1 (sr)
EP (2) EP1861100B1 (sr)
JP (1) JP2009503045A (sr)
KR (1) KR20080033501A (sr)
CN (1) CN101321528B (sr)
AT (1) ATE412414T1 (sr)
AU (1) AU2006277836B8 (sr)
CA (1) CA2620952A1 (sr)
CY (1) CY1108729T1 (sr)
DE (1) DE602006003415D1 (sr)
DK (1) DK1861100T3 (sr)
ES (1) ES2317564T3 (sr)
GB (1) GB0516168D0 (sr)
HK (1) HK1111084A1 (sr)
HR (1) HRP20090017T3 (sr)
MX (1) MX2008001546A (sr)
NZ (1) NZ566010A (sr)
PL (1) PL1861100T3 (sr)
PT (1) PT1861100E (sr)
RS (1) RS50720B (sr)
RU (1) RU2409364C2 (sr)
SI (1) SI1861100T1 (sr)
WO (1) WO2007017643A1 (sr)
ZA (2) ZA200801170B (sr)

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GB2410947B (en) * 2004-02-11 2008-09-17 Cambridge Lab Ltd Pharmaceutical compounds
GB0514501D0 (en) * 2005-07-14 2005-08-24 Cambridge Lab Ireland Ltd Pharmaceutical compounds
CA2668689C (en) 2006-11-08 2015-12-29 Neurocrine Biosciences Inc. Substituted 3-isobutyl-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2h-pyrido[2,1-a]isoquinolin-2-ol compounds and methods relating thereto
GB0721669D0 (en) * 2007-11-02 2007-12-12 Cambridge Lab Ireland Ltd Pharmaceutical compounds
GB0810857D0 (en) * 2008-06-13 2008-07-23 Cambridge Lab Ireland Ltd Pharmaceutical compounds
GB2462611A (en) * 2008-08-12 2010-02-17 Cambridge Lab Pharmaceutical composition comprising tetrabenazine
US20110053866A1 (en) * 2008-08-12 2011-03-03 Biovail Laboratories International (Barbados) S.R.L. Pharmaceutical compositions
GB2463451A (en) * 2008-09-08 2010-03-17 Cambridge Lab 3, 11b cis-dihydrotetrabenazine compounds for use in the treatment of dementia
GB2463283A (en) * 2008-09-08 2010-03-10 Cambridge Lab 3,11b-cis-dihydrotetrabenazine for use in treating asthma
GB2463452A (en) * 2008-09-08 2010-03-17 Cambridge Lab Desmethyl derivatives of tetrabenazine and pharmaceutical compositions thereof
US20120003330A1 (en) 2010-06-01 2012-01-05 Auspex Pharmaceuticals, Inc. Benzoquinolone inhibitors of vmat2
CN102285984B (zh) * 2010-11-25 2012-10-10 江苏威凯尔医药科技有限公司 (2R,3R,11bR)-二氢丁苯那嗪及相关化合物的制备方法
AU2015209330A1 (en) 2014-01-27 2016-07-28 Auspex Pharmaceuticals, Inc. Benzoquinoline inhibitors of vesicular monoamine transporter 2
MA41177A (fr) * 2014-12-15 2017-10-24 Esteve Labor Dr Utilisation de ligands des récepteurs sigma dans l'arthrose
US10550120B2 (en) 2016-03-25 2020-02-04 Tohoku University Indole alkaloid compound having immune checkpoint inhibitory action
CN109283279B (zh) * 2017-07-21 2019-11-01 南京正大天晴制药有限公司 通过高效液相色谱法分离测定雷替曲塞及其对映异构体的方法
CN109283263B (zh) * 2017-07-21 2019-06-25 南京正大天晴制药有限公司 用于雷替曲塞合成质量控制的检测分析方法

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GB0514501D0 (en) * 2005-07-14 2005-08-24 Cambridge Lab Ireland Ltd Pharmaceutical compounds
GB0810857D0 (en) * 2008-06-13 2008-07-23 Cambridge Lab Ireland Ltd Pharmaceutical compounds
US20110053866A1 (en) * 2008-08-12 2011-03-03 Biovail Laboratories International (Barbados) S.R.L. Pharmaceutical compositions
GB2462611A (en) * 2008-08-12 2010-02-17 Cambridge Lab Pharmaceutical composition comprising tetrabenazine
GB2463452A (en) * 2008-09-08 2010-03-17 Cambridge Lab Desmethyl derivatives of tetrabenazine and pharmaceutical compositions thereof
GB2463283A (en) * 2008-09-08 2010-03-10 Cambridge Lab 3,11b-cis-dihydrotetrabenazine for use in treating asthma
GB2463451A (en) * 2008-09-08 2010-03-17 Cambridge Lab 3, 11b cis-dihydrotetrabenazine compounds for use in the treatment of dementia

Also Published As

Publication number Publication date
EP1964565A1 (en) 2008-09-03
MX2008001546A (es) 2008-04-04
PT1861100E (pt) 2008-12-26
SI1861100T1 (sl) 2009-04-30
DK1861100T3 (da) 2008-12-15
HK1111084A1 (en) 2008-08-01
ZA200801171B (en) 2009-08-26
WO2007017643A1 (en) 2007-02-15
NZ566010A (en) 2010-05-28
EP1861100B1 (en) 2008-10-29
CA2620952A1 (en) 2007-02-15
ZA200801170B (en) 2009-12-30
CN101321528B (zh) 2011-05-25
AU2006277836B8 (en) 2011-12-08
AU2006277836B2 (en) 2011-11-10
ATE412414T1 (de) 2008-11-15
ES2317564T3 (es) 2009-04-16
JP2009503045A (ja) 2009-01-29
DE602006003415D1 (de) 2008-12-11
HRP20090017T3 (en) 2009-03-31
PL1861100T3 (pl) 2009-06-30
CY1108729T1 (el) 2014-04-09
CN101321528A (zh) 2008-12-10
EP1861100A1 (en) 2007-12-05
RU2008108516A (ru) 2009-09-10
GB0516168D0 (en) 2005-09-14
US20090275605A1 (en) 2009-11-05
RU2409364C2 (ru) 2011-01-20
KR20080033501A (ko) 2008-04-16
AU2006277836A1 (en) 2007-02-15

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