PL1778686T3 - Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38 - Google Patents

Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38

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Publication number
PL1778686T3
PL1778686T3 PL05772546T PL05772546T PL1778686T3 PL 1778686 T3 PL1778686 T3 PL 1778686T3 PL 05772546 T PL05772546 T PL 05772546T PL 05772546 T PL05772546 T PL 05772546T PL 1778686 T3 PL1778686 T3 PL 1778686T3
Authority
PL
Poland
Prior art keywords
kinase inhibitors
map kinase
triazolopyridinylsulfanyl
derivatives
triazolopyridinylsulfanyl derivatives
Prior art date
Application number
PL05772546T
Other languages
English (en)
Inventor
John Paul Mathias
David Simon Millan
Russell Andrew Lewthwaite
Christopher Phillips
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0418015A external-priority patent/GB0418015D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of PL1778686T3 publication Critical patent/PL1778686T3/pl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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PL05772546T 2004-08-12 2005-08-09 Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38 PL1778686T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0418015A GB0418015D0 (en) 2004-08-12 2004-08-12 New compounds
US69155905P 2005-06-17 2005-06-17
EP05772546A EP1778686B9 (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors
PCT/IB2005/002574 WO2006018718A2 (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors

Publications (1)

Publication Number Publication Date
PL1778686T3 true PL1778686T3 (pl) 2009-04-30

Family

ID=35783420

Family Applications (1)

Application Number Title Priority Date Filing Date
PL05772546T PL1778686T3 (pl) 2004-08-12 2005-08-09 Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38

Country Status (35)

Country Link
US (2) US7511057B2 (pl)
EP (1) EP1778686B9 (pl)
JP (1) JP4084836B2 (pl)
AP (1) AP2326A (pl)
AR (1) AR050692A1 (pl)
AT (1) ATE412652T1 (pl)
AU (1) AU2005273612B2 (pl)
BR (1) BRPI0514255A (pl)
CA (1) CA2576297C (pl)
CR (1) CR8918A (pl)
CU (1) CU23497A3 (pl)
CY (1) CY1108788T1 (pl)
DE (1) DE602005010714D1 (pl)
DK (1) DK1778686T3 (pl)
EA (1) EA012119B1 (pl)
EC (1) ECSP077232A (pl)
ES (1) ES2314690T3 (pl)
GE (1) GEP20104973B (pl)
GT (1) GT200500218A (pl)
HK (1) HK1105536A1 (pl)
HN (1) HN2005000418A (pl)
HR (1) HRP20080608T3 (pl)
IL (1) IL181047A (pl)
MA (1) MA28798B1 (pl)
MX (1) MX2007001759A (pl)
MY (1) MY140021A (pl)
NL (1) NL1029726C2 (pl)
NO (1) NO339320B1 (pl)
NZ (1) NZ552868A (pl)
PL (1) PL1778686T3 (pl)
PT (1) PT1778686E (pl)
SI (1) SI1778686T1 (pl)
SV (1) SV2006002193A (pl)
TN (1) TNSN07050A1 (pl)
WO (1) WO2006018718A2 (pl)

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US7572807B2 (en) * 2005-06-09 2009-08-11 Bristol-Myers Squibb Company Heteroaryl 11-beta-hydroxysteroid dehydrogenase type I inhibitors
CA2642209A1 (en) * 2006-02-09 2007-08-16 Pfizer Limited Triazolopyridine compounds
JP5244369B2 (ja) * 2006-11-10 2013-07-24 富士フイルム株式会社 ５−アミノピラゾール誘導体の製造方法、アゾ色素
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
US8119658B2 (en) 2007-10-01 2012-02-21 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
SI2303267T1 (sl) * 2008-02-04 2013-09-30 Pfizer Limited Polimorfna oblika derivata (1,2,4)triazolo(4,3-a)piridina za zdravljenje vnetnih bolezni
US8498729B2 (en) 2008-08-29 2013-07-30 Smp Logic Systems Llc Manufacturing execution system for use in manufacturing baby formula
US20110166059A1 (en) * 2008-09-12 2011-07-07 Dorothee Viemann Means and methods for evaluating a therapy with a p38 map kinase inhibitor
EP2398798A1 (en) 2009-02-17 2011-12-28 CHIESI FARMACEUTICI S.p.A. Triazolopyridine derivatives as p38 map kinase inhibitors
GB0905955D0 (en) 2009-04-06 2009-05-20 Respivert Ltd Novel compounds
MX2011012961A (es) 2009-06-05 2012-01-30 Cephalon Inc Preparacion y usos de derivados de 1,2,4-triazolo[1,5a]-piridina.
GB201005589D0 (en) 2010-04-01 2010-05-19 Respivert Ltd Novel compounds
EP2556068B1 (en) 2010-04-08 2019-01-23 Respivert Limited P38 map kinase inhibitors
WO2011158044A2 (en) 2010-06-17 2011-12-22 Respivert Limited Respiratory formulations and compounds for use therein
ES2671748T3 (es) * 2011-07-21 2018-06-08 Tolero Pharmaceuticals, Inc. Inhibidores heterocíclicos de proteína quinasas
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