NO327983B1 - Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade - Google Patents
Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade Download PDFInfo
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- NO327983B1 NO327983B1 NO20000786A NO20000786A NO327983B1 NO 327983 B1 NO327983 B1 NO 327983B1 NO 20000786 A NO20000786 A NO 20000786A NO 20000786 A NO20000786 A NO 20000786A NO 327983 B1 NO327983 B1 NO 327983B1
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- gabapentin
- treatment
- gaba
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Addiction (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Psychiatry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
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US5675397P | 1997-08-20 | 1997-08-20 | |
US7479498P | 1998-02-16 | 1998-02-16 | |
US8293698P | 1998-04-24 | 1998-04-24 | |
PCT/US1998/017082 WO1999008671A1 (en) | 1997-08-20 | 1998-08-18 | Gaba analogs to prevent and treat gastrointestinal damage |
Publications (3)
Publication Number | Publication Date |
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NO20000786D0 NO20000786D0 (no) | 2000-02-17 |
NO20000786L NO20000786L (no) | 2000-02-17 |
NO327983B1 true NO327983B1 (no) | 2009-11-02 |
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NO20000786A NO327983B1 (no) | 1997-08-20 | 2000-02-17 | Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade |
Country Status (25)
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US (2) | US6242488B1 (is) |
EP (1) | EP1009399B1 (is) |
JP (1) | JP4681116B2 (is) |
KR (2) | KR100609359B1 (is) |
AT (1) | ATE461698T1 (is) |
AU (2) | AU8668598A (is) |
BR (1) | BR9812133A (is) |
CA (1) | CA2297163C (is) |
CO (1) | CO4960645A1 (is) |
CY (1) | CY1109981T1 (is) |
DE (1) | DE69841574D1 (is) |
DK (1) | DK1009399T3 (is) |
ES (1) | ES2341154T3 (is) |
HU (1) | HUP0004551A3 (is) |
IL (1) | IL134164A (is) |
IS (1) | IS2749B (is) |
MY (1) | MY155223A (is) |
NO (1) | NO327983B1 (is) |
NZ (1) | NZ502729A (is) |
PE (1) | PE107299A1 (is) |
PL (1) | PL194125B1 (is) |
PT (1) | PT1009399E (is) |
TW (2) | TW570794B (is) |
UY (1) | UY25148A1 (is) |
WO (2) | WO1999008670A1 (is) |
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EP1031350A1 (en) * | 1999-02-23 | 2000-08-30 | Warner-Lambert Company | Use of a gabapentin-analog for the manufacture of a medicament for preventing and treating visceral pain |
US6451857B1 (en) | 1999-03-10 | 2002-09-17 | Warner-Lambert Company | Analgesic compositions comprising anti-epileptic compounds and methods of using same |
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WO2000061188A1 (en) * | 1999-04-09 | 2000-10-19 | Euro-Celtique S.A. | Sodium channel blocker compositions and the use thereof |
EP1840117A1 (en) * | 1999-06-10 | 2007-10-03 | Warner-Lambert Company LLC | Mono- and disubstituted 3-propyl gamma-aminobutyric acids |
PT1202725E (pt) | 1999-07-22 | 2007-07-11 | Universuty Of Rochester | Método para tratar sintomas de alteração hormonal, incluindo afrontamentos. |
FR2801217B1 (fr) * | 1999-11-24 | 2002-12-06 | Aventis Pharma Sa | Association de riluzole et de gabapentine et son utilisation comme medicament |
JP2003533223A (ja) * | 2000-05-16 | 2003-11-11 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | α2δ2カルシウムチャネルサブユニットの発現細胞株 |
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US7186855B2 (en) | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
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JP2005501013A (ja) | 2001-06-11 | 2005-01-13 | ゼノポート,インコーポレイテッド | Gaba類似体の全身濃度が持続するアミノ酸コンジュゲート |
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AU2002333374B2 (en) | 2001-09-03 | 2007-03-22 | Newron Pharmaceuticals S.P.A. | Pharmaceutical composition comprising gabapentin or an analogue thereof and an (alpha)- aminoamide and its analgesic use |
TWI312285B (en) | 2001-10-25 | 2009-07-21 | Depomed Inc | Methods of treatment using a gastric retained gabapentin dosage |
US20060159743A1 (en) * | 2001-10-25 | 2006-07-20 | Depomed, Inc. | Methods of treating non-nociceptive pain states with gastric retentive gabapentin |
US7612112B2 (en) | 2001-10-25 | 2009-11-03 | Depomed, Inc. | Methods of treatment using a gastric retained gabapentin dosage |
US20070184104A1 (en) * | 2001-10-25 | 2007-08-09 | Depomed, Inc. | Gastric retentive gabapentin dosage forms and methods for using same |
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- 1998-07-29 AU AU86685/98A patent/AU8668598A/en not_active Withdrawn
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- 1998-08-18 HU HU0004551A patent/HUP0004551A3/hu unknown
- 1998-08-18 PL PL98338705A patent/PL194125B1/pl not_active IP Right Cessation
- 1998-08-18 ES ES98945758T patent/ES2341154T3/es not_active Expired - Lifetime
- 1998-08-18 DE DE69841574T patent/DE69841574D1/de not_active Expired - Lifetime
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- 1998-08-18 BR BR9812133-2A patent/BR9812133A/pt not_active Application Discontinuation
- 1998-08-18 KR KR1020057022543A patent/KR20050116168A/ko not_active Application Discontinuation
- 1998-08-18 AU AU92930/98A patent/AU9293098A/en not_active Abandoned
- 1998-08-18 DK DK98945758.5T patent/DK1009399T3/da active
- 1998-08-18 JP JP2000509411A patent/JP4681116B2/ja not_active Expired - Fee Related
- 1998-08-18 CA CA002297163A patent/CA2297163C/en not_active Expired - Lifetime
- 1998-08-18 WO PCT/US1998/017082 patent/WO1999008671A1/en active IP Right Grant
- 1998-08-18 EP EP98945758A patent/EP1009399B1/en not_active Expired - Lifetime
- 1998-08-18 AT AT98945758T patent/ATE461698T1/de active
- 1998-08-18 IL IL13416498A patent/IL134164A/xx not_active IP Right Cessation
- 1998-08-18 TW TW092130045A patent/TWI251485B/zh not_active IP Right Cessation
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- 1998-08-20 UY UY25148A patent/UY25148A1/es unknown
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