NO327983B1 - Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade - Google Patents

Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade Download PDF

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Publication number
NO327983B1
NO327983B1 NO20000786A NO20000786A NO327983B1 NO 327983 B1 NO327983 B1 NO 327983B1 NO 20000786 A NO20000786 A NO 20000786A NO 20000786 A NO20000786 A NO 20000786A NO 327983 B1 NO327983 B1 NO 327983B1
Authority
NO
Norway
Prior art keywords
gabapentin
treatment
gaba
drug
ethanol
Prior art date
Application number
NO20000786A
Other languages
English (en)
Norwegian (no)
Other versions
NO20000786D0 (no
NO20000786L (no
Inventor
Jr Charles Price Taylor
Antonio Guglietta
Jiayuan Ren
William Patrick Watson
Laurent Diop
Maria Chovet
Lionel Bueno
Hillary J Little
Michael Francis Rafferty
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27369092&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO327983(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of NO20000786D0 publication Critical patent/NO20000786D0/no
Publication of NO20000786L publication Critical patent/NO20000786L/no
Publication of NO327983B1 publication Critical patent/NO327983B1/no

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/405Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32Alcohol-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Addiction (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
NO20000786A 1997-08-20 2000-02-17 Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade NO327983B1 (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US5675397P 1997-08-20 1997-08-20
US7479498P 1998-02-16 1998-02-16
US8293698P 1998-04-24 1998-04-24
PCT/US1998/017082 WO1999008671A1 (en) 1997-08-20 1998-08-18 Gaba analogs to prevent and treat gastrointestinal damage

Publications (3)

Publication Number Publication Date
NO20000786D0 NO20000786D0 (no) 2000-02-17
NO20000786L NO20000786L (no) 2000-02-17
NO327983B1 true NO327983B1 (no) 2009-11-02

Family

ID=27369092

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20000786A NO327983B1 (no) 1997-08-20 2000-02-17 Anvendelse av GABA analoger og et ikke-steroidalt anti-inflammatorisk legemiddel for fremstilling av et medikament for forebyggelse og behandling av gastrointestinal skade

Country Status (25)

Country Link
US (2) US6242488B1 (is)
EP (1) EP1009399B1 (is)
JP (1) JP4681116B2 (is)
KR (2) KR100609359B1 (is)
AT (1) ATE461698T1 (is)
AU (2) AU8668598A (is)
BR (1) BR9812133A (is)
CA (1) CA2297163C (is)
CO (1) CO4960645A1 (is)
CY (1) CY1109981T1 (is)
DE (1) DE69841574D1 (is)
DK (1) DK1009399T3 (is)
ES (1) ES2341154T3 (is)
HU (1) HUP0004551A3 (is)
IL (1) IL134164A (is)
IS (1) IS2749B (is)
MY (1) MY155223A (is)
NO (1) NO327983B1 (is)
NZ (1) NZ502729A (is)
PE (1) PE107299A1 (is)
PL (1) PL194125B1 (is)
PT (1) PT1009399E (is)
TW (2) TW570794B (is)
UY (1) UY25148A1 (is)
WO (2) WO1999008670A1 (is)

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Publication number Publication date
CO4960645A1 (es) 2000-09-25
TWI251485B (en) 2006-03-21
TW570794B (en) 2004-01-11
WO1999008670A1 (en) 1999-02-25
IL134164A (en) 2005-05-17
EP1009399A1 (en) 2000-06-21
TW200412938A (en) 2004-08-01
KR20010023084A (ko) 2001-03-26
WO1999008671A1 (en) 1999-02-25
PL194125B1 (pl) 2007-04-30
CA2297163C (en) 2001-11-20
EP1009399B1 (en) 2010-03-24
AU8668598A (en) 1999-03-08
UY25148A1 (es) 1999-01-26
DE69841574D1 (de) 2010-05-06
AU9293098A (en) 1999-03-08
IS2749B (is) 2011-08-15
ATE461698T1 (de) 2010-04-15
KR20050116168A (ko) 2005-12-09
HUP0004551A3 (en) 2002-11-28
KR100609359B1 (ko) 2006-08-04
NO20000786D0 (no) 2000-02-17
NO20000786L (no) 2000-02-17
US6426368B2 (en) 2002-07-30
US20010014698A1 (en) 2001-08-16
PT1009399E (pt) 2010-05-21
DK1009399T3 (da) 2010-05-31
CA2297163A1 (en) 1999-02-25
PE107299A1 (es) 1999-12-19
ES2341154T3 (es) 2010-06-15
JP2001515033A (ja) 2001-09-18
BR9812133A (pt) 2000-07-18
HUP0004551A2 (hu) 2001-05-28
IS5361A (is) 2000-01-25
IL134164A0 (en) 2001-04-30
PL338705A1 (en) 2000-11-20
MY155223A (en) 2015-09-30
US6242488B1 (en) 2001-06-05
CY1109981T1 (el) 2014-09-10
JP4681116B2 (ja) 2011-05-11
NZ502729A (en) 2002-10-25

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