NO324595B1 - Tartratsalt av tiazolidindionderivat, fremgangsmate for fremstilling derav, anvendelse derav og farmasoytisk preparat omfattende saltet - Google Patents

Tartratsalt av tiazolidindionderivat, fremgangsmate for fremstilling derav, anvendelse derav og farmasoytisk preparat omfattende saltet Download PDF

Info

Publication number: NO324595B1
Authority: NO; Norway
Prior art keywords: tartrate; solvate; salt; methyl; thiazolidine
Prior art date: 2000-08-04

Application number

NO20030507A

Other languages

English (en)

Norwegian (no)

Other versions

NO20030507D0 (no

NO20030507L (no

Inventor

Bernadette Marie Choudary

Andrew Simon Craig

Tim Chien Ting Ho

Donald Colin Mackenzie

Deirdre O'keeffe

Original Assignee

Smithkline Beecham Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-04

Filing date

2003-01-31

Publication date

2007-11-26

2003-01-31 Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc

2003-01-31 Publication of NO20030507D0 publication Critical patent/NO20030507D0/no

2003-03-26 Publication of NO20030507L publication Critical patent/NO20030507L/no

2007-11-26 Publication of NO324595B1 publication Critical patent/NO324595B1/no

Links

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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Diabetes (AREA)
General Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Hematology (AREA)
Obesity (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Cosmetics (AREA)

NO20030507A 2000-08-04 2003-01-31 Tartratsalt av tiazolidindionderivat, fremgangsmate for fremstilling derav, anvendelse derav og farmasoytisk preparat omfattende saltet NO324595B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0019228.6A GB0019228D0 (en)	2000-08-04	2000-08-04	Novel pharmaceutical
PCT/GB2001/003515 WO2002012234A1 (en)	2000-08-04	2001-08-03	Tartrate salts of thiazolidinedione derivative

Publications (3)

Publication Number	Publication Date
NO20030507D0 NO20030507D0 (no)	2003-01-31
NO20030507L NO20030507L (no)	2003-03-26
NO324595B1 true NO324595B1 (no)	2007-11-26

Family

ID=9897030

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20030507A NO324595B1 (no)	2000-08-04	2003-01-31	Tartratsalt av tiazolidindionderivat, fremgangsmate for fremstilling derav, anvendelse derav og farmasoytisk preparat omfattende saltet

Country Status (36)

Country	Link
US (1)	US20040048899A1 (es)
EP (1)	EP1305312B1 (es)
JP (1)	JP2004505972A (es)
KR (1)	KR100755173B1 (es)
CN (1)	CN1458931A (es)
AP (1)	AP1814A (es)
AT (1)	ATE393153T1 (es)
AU (1)	AU2001276509A1 (es)
BG (1)	BG107606A (es)
BR (1)	BR0112981A (es)
CA (1)	CA2417829A1 (es)
CZ (1)	CZ2003316A3 (es)
DE (1)	DE60133746T2 (es)
DK (1)	DK1305312T3 (es)
DZ (1)	DZ3467A1 (es)
EA (1)	EA004764B1 (es)
EC (1)	ECSP034469A (es)
ES (1)	ES2302506T3 (es)
GB (1)	GB0019228D0 (es)
HK (1)	HK1057359A1 (es)
HR (1)	HRP20030070A2 (es)
HU (1)	HUP0300777A3 (es)
IL (2)	IL154278A0 (es)
MA (1)	MA25898A1 (es)
MX (1)	MXPA03001087A (es)
NO (1)	NO324595B1 (es)
NZ (1)	NZ524032A (es)
OA (1)	OA12352A (es)
PL (1)	PL360703A1 (es)
PT (1)	PT1305312E (es)
SI (1)	SI1305312T1 (es)
SK (1)	SK1442003A3 (es)
UA (1)	UA76721C2 (es)
WO (1)	WO2002012234A1 (es)
YU (1)	YU16303A (es)
ZA (1)	ZA200300963B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
USRE39384E1 (en)	1993-09-01	2006-11-07	Smithkline Beecham P.L.C.	Substituted thiazolidinedione derivatives
AR047530A1 (es) *	2004-02-04	2006-01-25	Novartis Ag	Formas de sal de 4-(4-metilpiperazin-1-ilmetil)-n-(4-metil-3-(4-piridin-3-il)pirimidin-2-ilamino)fenil)-benzamida
CN1984903A (zh) *	2004-06-30	2007-06-20	伊莱利利公司	1－(吲哚－6－羰基－d－苯基甘氨酰基)－4－(1－甲基哌啶－4－基)哌嗪d－酒石酸盐
US7435741B2 (en)	2006-05-09	2008-10-14	Teva Pharmaceutical Industries, Ltd.	2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
GB0616574D0 (en) *	2006-08-21	2006-09-27	Glaxo Group Ltd	Compounds
DE102009053562A1 (de)	2009-11-18	2011-05-19	Alfred E. Tiefenbacher (Gmbh & Co. Kg)	Rosiglitazonsuccinat enthaltende pharmazeutische Zusammensetzung
CN102532122B (zh) *	2010-12-29	2015-12-02	开封制药(集团)有限公司	酒石酸罗格列酮的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6288095B1 (en) *	1987-09-04	2001-09-11	Beecham Group P.L.C.	Compounds
ES2137915T3 (es) *	1987-09-04	2000-01-01	Beecham Group Plc	Derivados de tiazolidindiona sustituida.
GB9218830D0 (en) *	1992-09-05	1992-10-21	Smithkline Beecham Plc	Novel compounds
US5741803A (en) *	1992-09-05	1998-04-21	Smithkline Beecham Plc	Substituted thiazolidinedionle derivatives

2000
- 2000-08-04 GB GBGB0019228.6A patent/GB0019228D0/en not_active Ceased
2001
- 2001-03-08 UA UA2003020940A patent/UA76721C2/uk unknown
- 2001-08-03 CZ CZ2003316A patent/CZ2003316A3/cs unknown
- 2001-08-03 DK DK01954162T patent/DK1305312T3/da active
- 2001-08-03 EA EA200300234A patent/EA004764B1/ru not_active IP Right Cessation
- 2001-08-03 US US10/343,866 patent/US20040048899A1/en not_active Abandoned
- 2001-08-03 WO PCT/GB2001/003515 patent/WO2002012234A1/en active IP Right Grant
- 2001-08-03 CN CN01815685A patent/CN1458931A/zh active Pending
- 2001-08-03 SK SK144-2003A patent/SK1442003A3/sk unknown
- 2001-08-03 EP EP01954162A patent/EP1305312B1/en not_active Expired - Lifetime
- 2001-08-03 KR KR1020037001606A patent/KR100755173B1/ko not_active IP Right Cessation
- 2001-08-03 BR BR0112981-3A patent/BR0112981A/pt not_active IP Right Cessation
- 2001-08-03 AT AT01954162T patent/ATE393153T1/de not_active IP Right Cessation
- 2001-08-03 PT PT01954162T patent/PT1305312E/pt unknown
- 2001-08-03 PL PL36070301A patent/PL360703A1/xx not_active Application Discontinuation
- 2001-08-03 OA OA1200300026A patent/OA12352A/en unknown
- 2001-08-03 DZ DZ013467A patent/DZ3467A1/fr active
- 2001-08-03 MX MXPA03001087A patent/MXPA03001087A/es active IP Right Grant
- 2001-08-03 AU AU2001276509A patent/AU2001276509A1/en not_active Abandoned
- 2001-08-03 ES ES01954162T patent/ES2302506T3/es not_active Expired - Lifetime
- 2001-08-03 HU HU0300777A patent/HUP0300777A3/hu unknown
- 2001-08-03 YU YU16303A patent/YU16303A/sh unknown
- 2001-08-03 AP APAP/P/2003/002738A patent/AP1814A/en active
- 2001-08-03 CA CA002417829A patent/CA2417829A1/en not_active Abandoned
- 2001-08-03 DE DE60133746T patent/DE60133746T2/de not_active Expired - Fee Related
- 2001-08-03 SI SI200130830T patent/SI1305312T1/sl unknown
- 2001-08-03 NZ NZ524032A patent/NZ524032A/en unknown
- 2001-08-03 IL IL15427801A patent/IL154278A0/xx active IP Right Grant
- 2001-08-03 JP JP2002518209A patent/JP2004505972A/ja not_active Withdrawn
2003
- 2003-01-31 NO NO20030507A patent/NO324595B1/no not_active IP Right Cessation
- 2003-02-03 MA MA27021A patent/MA25898A1/fr unknown
- 2003-02-03 HR HR20030070A patent/HRP20030070A2/hr not_active Application Discontinuation
- 2003-02-03 IL IL154278A patent/IL154278A/en not_active IP Right Cessation
- 2003-02-04 EC EC2003004469A patent/ECSP034469A/es unknown
- 2003-02-28 BG BG107606A patent/BG107606A/bg unknown
- 2003-03-04 ZA ZA200300963A patent/ZA200300963B/en unknown
- 2003-10-24 HK HK03107710.1A patent/HK1057359A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
DE60133746T2 (de)	2009-05-14
EA004764B1 (ru)	2004-08-26
YU16303A (sh)	2006-01-16
MXPA03001087A (es)	2003-05-27
AU2001276509A1 (en)	2002-02-18
WO2002012234A1 (en)	2002-02-14
SK1442003A3 (en)	2004-05-04
PL360703A1 (en)	2004-09-20
KR100755173B1 (ko)	2007-09-03
GB0019228D0 (en)	2000-09-27
CZ2003316A3 (en)	2004-03-17
NO20030507D0 (no)	2003-01-31
BG107606A (bg)	2003-09-30
ZA200300963B (en)	2004-04-19
ES2302506T3 (es)	2008-07-16
HUP0300777A2 (hu)	2003-11-28
DE60133746D1 (de)	2008-06-05
HK1057359A1 (en)	2004-04-02
CA2417829A1 (en)	2002-02-14
PT1305312E (pt)	2008-06-19
EA200300234A1 (ru)	2003-06-26
IL154278A0 (en)	2003-09-17
NO20030507L (no)	2003-03-26
ATE393153T1 (de)	2008-05-15
US20040048899A1 (en)	2004-03-11
BR0112981A (pt)	2003-08-26
OA12352A (en)	2006-05-16
SI1305312T1 (sl)	2008-08-31
EP1305312A1 (en)	2003-05-02
NZ524032A (en)	2004-07-30
DK1305312T3 (da)	2008-07-28
AP2003002738A0 (en)	2003-03-31
UA76721C2 (uk)	2006-09-15
MA25898A1 (fr)	2003-10-01
HRP20030070A2 (en)	2005-02-28
EP1305312B1 (en)	2008-04-23
KR20030022357A (ko)	2003-03-15
IL154278A (en)	2009-02-11
JP2004505972A (ja)	2004-02-26
HUP0300777A3 (en)	2005-04-28
ECSP034469A (es)	2003-06-25
DZ3467A1 (fr)	2002-02-14
CN1458931A (zh)	2003-11-26
AP1814A (en)	2008-01-04

Legal Events

Date	Code	Title	Description
2010-03-22	MM1K	Lapsed by not paying the annual fees

Publication	Publication Date	Title
US7291740B2 (en)	2007-11-06	5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione Mesylate salt
NO324595B1 (no)	2007-11-26	Tartratsalt av tiazolidindionderivat, fremgangsmate for fremstilling derav, anvendelse derav og farmasoytisk preparat omfattende saltet
NO324020B1 (no)	2007-07-30	Hydrokloridsalt av 5-[4-[2-(N-metyl-N (2-pyridyl)amino)etoksy]benzyl]tiazolidin-2,4-dion, farmasoytisk sammensetning som innbefatter dette samt fremgangsmate for fremstilling og anvendelse derav
EP1305311B1 (en)	2008-01-16	Tartrate salt of thiazolidinedione derivative
US20040014791A1 (en)	2004-01-22	Thiazolidinedione derivative and its use as antidiabetic
KR20040062965A (ko)	2004-07-09	로시글리타존 에디실레이트 및 항당뇨제로서의 그의 용도
NO324598B1 (no)	2007-11-26	Tartratsalter av tiazolidindionderivat, fremgangsmate for fremstilling drav, anvendelse derav samt farmasoytisk preparat inneholdende saltet
EP1325000B1 (en)	2007-07-25	A thiazolidinedione derivative and its use as antidiabetic
WO2002012233A1 (en)	2002-02-14	Tartrate salts of thiazolidinedione derivative
US20040102485A1 (en)	2004-05-27	Tartrate salt of thiazolidinedione derivative
WO2003050112A1 (en)	2003-06-19	Toluenesulfonate hydrates of a thiazolidinedione derivative