NO20082209L - Homo- og heterocykliske forbindelser anvendbare som CETP-inhibitorer - Google Patents

Homo- og heterocykliske forbindelser anvendbare som CETP-inhibitorer

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Publication number
NO20082209L
NO20082209L NO20082209A NO20082209A NO20082209L NO 20082209 L NO20082209 L NO 20082209L NO 20082209 A NO20082209 A NO 20082209A NO 20082209 A NO20082209 A NO 20082209A NO 20082209 L NO20082209 L NO 20082209L
Authority
NO
Norway
Prior art keywords
homo
heterocyclic compounds
compounds useful
cetp inhibitors
cetp
Prior art date
Application number
NO20082209A
Other languages
English (en)
Inventor
Wu Yang
Mark E Salvati
Heather Finlay
Bang-Chi Chen
Lalgudi S Harikrishnan
Ji Jiang
James A Johnson
Muthoni G Kamau
Michael R Lawrence
Jianqing Li
John Lloyd
Michael M Miller
Zulan Pi
Jennifer X Qiao
Richard RAMPULLA
Tammy C Wang
Yufeng Wang
Jacques Y Roberge
Original Assignee
Bristol Myers Squibb Co
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Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37733576&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20082209(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20082209L publication Critical patent/NO20082209L/no

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    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D333/70—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Abstract

Forbindelser med formel Ia og Ib: Ia Ib hvor A, B, C og R1 er som beskrevet her.
NO20082209A 2005-11-23 2008-05-14 Homo- og heterocykliske forbindelser anvendbare som CETP-inhibitorer NO20082209L (no)

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US11/558,979 US7790770B2 (en) 2005-11-23 2006-11-13 Heterocyclic CETP inhibitors
PCT/US2006/060958 WO2007062308A2 (en) 2005-11-23 2006-11-16 Homo- and heterocyclic compounds suitable as cetp inhibitors

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