NO20030382L - Nye indolderivater og deres anvendelse som medikamenter - Google Patents

Nye indolderivater og deres anvendelse som medikamenter

Info

Publication number
NO20030382L
NO20030382L NO20030382A NO20030382A NO20030382L NO 20030382 L NO20030382 L NO 20030382L NO 20030382 A NO20030382 A NO 20030382A NO 20030382 A NO20030382 A NO 20030382A NO 20030382 L NO20030382 L NO 20030382L
Authority
NO
Norway
Prior art keywords
drugs
indole derivatives
new indole
new
derivatives
Prior art date
Application number
NO20030382A
Other languages
English (en)
Other versions
NO20030382D0 (no
NO324594B1 (no
Inventor
Peter Emig
Gerald Bacher
Dietmar Reichert
Silke Baasner
Beate Aue
Bernd Nickel
Eckhard Guenther
Original Assignee
Zentaris Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Ag filed Critical Zentaris Ag
Publication of NO20030382D0 publication Critical patent/NO20030382D0/no
Publication of NO20030382L publication Critical patent/NO20030382L/no
Publication of NO324594B1 publication Critical patent/NO324594B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
NO20030382A 2000-07-28 2003-01-24 Nye indolderivater, fremgangsmate for fremstilling derav og deres anvendelse og medikamenter inneholdende derivatene. NO324594B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10037310A DE10037310A1 (de) 2000-07-28 2000-07-28 Neue Indolderivate und deren Verwendung als Arzneimittel
PCT/EP2001/008644 WO2002010152A2 (de) 2000-07-28 2001-07-26 Neue indolderivate und deren verwendung als arzneimittel

Publications (3)

Publication Number Publication Date
NO20030382D0 NO20030382D0 (no) 2003-01-24
NO20030382L true NO20030382L (no) 2003-02-20
NO324594B1 NO324594B1 (no) 2007-11-26

Family

ID=7650860

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20030382A NO324594B1 (no) 2000-07-28 2003-01-24 Nye indolderivater, fremgangsmate for fremstilling derav og deres anvendelse og medikamenter inneholdende derivatene.

Country Status (31)

Country Link
US (3) US7365081B2 (no)
EP (3) EP1309585B1 (no)
JP (1) JP5113973B2 (no)
KR (1) KR100810453B1 (no)
CN (1) CN1215066C (no)
AR (1) AR055209A1 (no)
AT (1) ATE392420T1 (no)
AU (2) AU2001289758B2 (no)
BG (1) BG66457B1 (no)
BR (1) BR0112807A (no)
CA (3) CA2704693A1 (no)
CY (1) CY1108770T1 (no)
CZ (1) CZ304197B6 (no)
DE (2) DE10037310A1 (no)
DK (1) DK1309585T3 (no)
ES (1) ES2303532T3 (no)
HK (1) HK1058201A1 (no)
HU (1) HU229254B1 (no)
IL (2) IL153930A0 (no)
MX (1) MXPA03000644A (no)
NO (1) NO324594B1 (no)
NZ (1) NZ524404A (no)
PL (1) PL208673B1 (no)
PT (1) PT1309585E (no)
RU (1) RU2270196C9 (no)
SI (1) SI1309585T1 (no)
SK (1) SK288085B6 (no)
TW (1) TWI291955B (no)
UA (1) UA80670C2 (no)
WO (1) WO2002010152A2 (no)
ZA (1) ZA200300584B (no)

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US7205299B2 (en) * 2003-06-05 2007-04-17 Zentaris Gmbh Indole derivatives having an apoptosis-inducing effect
EP1484329A1 (de) * 2003-06-06 2004-12-08 Zentaris GmbH Indolderivate mit Apoptose induzierender Wirkung
CN1816543B (zh) * 2003-06-05 2011-01-19 赞塔里斯有限公司 具有细胞凋亡诱导效应的吲哚衍生物
US7211588B2 (en) * 2003-07-25 2007-05-01 Zentaris Gmbh N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation
US20050124623A1 (en) 2003-11-26 2005-06-09 Bender John A. Diazaindole-dicarbonyl-piperazinyl antiviral agents
US20060100432A1 (en) 2004-11-09 2006-05-11 Matiskella John D Crystalline materials of 1-(4-benzoyl-piperazin-1-yl)-2-[4-methoxy-7-(3-methyl-[1,2,4]triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-ethane-1,2-dione
GB2431927B (en) 2005-11-04 2010-03-17 Amira Pharmaceuticals Inc 5-Lipoxygenase-activating protein (FLAP) inhibitors
US7977359B2 (en) 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
US7851476B2 (en) 2005-12-14 2010-12-14 Bristol-Myers Squibb Company Crystalline forms of 1-benzoyl-4-[2-[4-methoxy-7-(3-methyl-1H-1,2,4-triazol-1-YL)-1-[(phosphonooxy)methyl]-1H-pyrrolo[2,3-C]pyridin-3-YL]-1,2-dioxoethyl]-piperazine
US7807671B2 (en) 2006-04-25 2010-10-05 Bristol-Myers Squibb Company Diketo-piperazine and piperidine derivatives as antiviral agents
NZ596024A (en) 2006-08-07 2013-07-26 Ironwood Pharmaceuticals Inc Indole compounds
BRPI0912267A2 (pt) 2008-05-23 2015-10-13 Amira Pharmaceuticals Inc sal farmaceuticamente aceitável, composição farmacêutica, artigo de fabricação, métodos para tratar asma, rinite alérgica, doença, lesões gástricas e dor, métodos para prevenir broncoconstrição e rinite alérgica, uso de um sal farmaceuticamente aceitável, e, processo para a preparação de um sal farmaceuticamente aceitável.
AR084433A1 (es) 2010-12-22 2013-05-15 Ironwood Pharmaceuticals Inc Inhibidores de la faah y composiciones farmaceuticas que los contienen

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US6204261B1 (en) 1995-12-20 2001-03-20 Vertex Pharmaceuticals Incorporated Inhibitors of interleukin-1β Converting enzyme inhibitors
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US5192770A (en) 1990-12-07 1993-03-09 Syntex (U.S.A.) Inc. Serotonergic alpha-oxoacetamides
US5480883A (en) * 1991-05-10 1996-01-02 Rhone-Poulenc Rorer Pharmaceuticals Inc. Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase
US5965582A (en) * 1994-08-03 1999-10-12 Asta Medica Aktiengesellschaft N-benzylindole and benzopyrazole derivatives with anti-asthmatic, anti-allergic, anti-inflammatory and immunemodulating effect
US5732113A (en) 1996-06-20 1998-03-24 Stanford University Timing and frequency synchronization of OFDM signals
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Also Published As

Publication number Publication date
PL361356A1 (en) 2004-10-04
CA2354210C (en) 2010-09-14
US20080153875A1 (en) 2008-06-26
CN1447805A (zh) 2003-10-08
US20030100597A1 (en) 2003-05-29
US7989453B2 (en) 2011-08-02
BR0112807A (pt) 2003-07-01
BG66457B1 (bg) 2014-10-31
DE10037310A1 (de) 2002-02-07
US8008324B2 (en) 2011-08-30
DK1309585T3 (da) 2008-06-23
UA80670C2 (en) 2007-10-25
AU2001289758B2 (en) 2006-07-06
IL153930A (en) 2008-11-03
EP1939195A1 (de) 2008-07-02
CA2704693A1 (en) 2002-01-28
CZ304197B6 (cs) 2013-12-27
US7365081B2 (en) 2008-04-29
NO20030382D0 (no) 2003-01-24
IL153930A0 (en) 2003-07-31
SI1309585T1 (sl) 2008-08-31
RU2270196C2 (ru) 2006-02-20
PT1309585E (pt) 2008-06-09
EP2163552A1 (de) 2010-03-17
HUP0300677A2 (hu) 2003-11-28
HK1058201A1 (en) 2004-05-07
AU8975801A (en) 2002-02-13
DE50113867D1 (de) 2008-05-29
EP1309585B1 (de) 2008-04-16
SK288085B6 (sk) 2013-06-03
US20080108819A1 (en) 2008-05-08
KR100810453B1 (ko) 2008-03-07
CY1108770T1 (el) 2014-04-09
WO2002010152A2 (de) 2002-02-07
TWI291955B (en) 2008-01-01
ZA200300584B (en) 2003-07-18
ATE392420T1 (de) 2008-05-15
EP1309585A2 (de) 2003-05-14
KR20030017658A (ko) 2003-03-03
NZ524404A (en) 2004-08-27
NO324594B1 (no) 2007-11-26
SK2222003A3 (en) 2004-04-06
JP2004505075A (ja) 2004-02-19
AR055209A1 (es) 2007-08-15
RU2270196C9 (ru) 2007-11-27
CZ2003500A3 (cs) 2004-03-17
WO2002010152A3 (de) 2002-08-01
MXPA03000644A (es) 2003-06-06
CN1215066C (zh) 2005-08-17
PL208673B1 (pl) 2011-05-31
CA2704691A1 (en) 2002-01-28
CA2354210A1 (en) 2002-01-28
HU229254B1 (en) 2013-10-28
JP5113973B2 (ja) 2013-01-09
BG107560A (bg) 2003-10-31
ES2303532T3 (es) 2008-08-16

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