NO172802C - Analogifremgangsmaate for fremstilling av terapeutisk aktive tienopyraner - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive tienopyraner

Info

Publication number
NO172802C
NO172802C NO893775A NO893775A NO172802C NO 172802 C NO172802 C NO 172802C NO 893775 A NO893775 A NO 893775A NO 893775 A NO893775 A NO 893775A NO 172802 C NO172802 C NO 172802C
Authority
NO
Norway
Prior art keywords
tienopyranes
preparation
therapeutic active
analogy procedure
analogy
Prior art date
Application number
NO893775A
Other languages
English (en)
Norwegian (no)
Other versions
NO893775D0 (no
NO172802B (no
NO893775L (no
Inventor
Jeffery B Press
Pauline Sanfilippo
James J Mcnally
Robert Falotico
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/249,043 external-priority patent/US4992435A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of NO893775D0 publication Critical patent/NO893775D0/no
Publication of NO893775L publication Critical patent/NO893775L/no
Publication of NO172802B publication Critical patent/NO172802B/no
Publication of NO172802C publication Critical patent/NO172802C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
NO893775A 1988-09-23 1989-09-22 Analogifremgangsmaate for fremstilling av terapeutisk aktive tienopyraner NO172802C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/249,043 US4992435A (en) 1988-09-23 1988-09-23 Substituted thienopyrans as antihypertensive agents
US40162889A 1989-09-06 1989-09-06

Publications (4)

Publication Number Publication Date
NO893775D0 NO893775D0 (no) 1989-09-22
NO893775L NO893775L (no) 1990-03-26
NO172802B NO172802B (no) 1993-06-01
NO172802C true NO172802C (no) 1993-09-08

Family

ID=26939780

Family Applications (1)

Application Number Title Priority Date Filing Date
NO893775A NO172802C (no) 1988-09-23 1989-09-22 Analogifremgangsmaate for fremstilling av terapeutisk aktive tienopyraner

Country Status (19)

Country Link
US (2) US5284857A (fr)
EP (1) EP0360621B1 (fr)
JP (1) JPH02174781A (fr)
KR (1) KR920008824B1 (fr)
CN (1) CN1032210C (fr)
AU (1) AU619896B2 (fr)
CA (1) CA1338419C (fr)
DE (1) DE68912476T2 (fr)
DK (1) DK469189A (fr)
ES (1) ES2062027T3 (fr)
FI (1) FI894491A (fr)
HU (1) HUT54162A (fr)
IE (1) IE63301B1 (fr)
IL (1) IL91709A (fr)
MY (1) MY129947A (fr)
NO (1) NO172802C (fr)
NZ (1) NZ230711A (fr)
PH (2) PH30818A (fr)
PT (1) PT91787B (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE63935B1 (en) * 1989-06-27 1995-06-28 Chem Pharm Forsch Gmbh Novel thienopyran derivatives a process for their preparation and their use
DE3925719A1 (de) * 1989-08-03 1991-02-07 Bayer Ag Substituierte thienopyranone, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung von parasiten
NZ240933A (en) * 1990-12-21 1993-05-26 Ortho Pharma Corp Preparing enantiomerically pure thienopyran derivatives
GB9225860D0 (en) * 1992-12-11 1993-02-03 Smithkline Beecham Plc Novel treatment
GB9411635D0 (en) 1994-06-10 1994-08-03 Smithkline Beecham Plc Novel treatment
DE19706892A1 (de) * 1997-02-21 1998-08-27 Hoechst Ag Sulfonamid-substituierte Thiophene, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
EP0895994A3 (fr) * 1997-08-05 1999-12-15 Hoechst Marion Roussel Deutschland GmbH Dérivés de pyranopyridine substitués par un sulfonamide, procédé pour leur préparation, leur utilisation comme médicaments ou diagnostics et médicament les contenant
GB9909792D0 (en) * 1998-12-04 1999-06-23 Cambridge Bioclinical Limited Potassium channel activators and their use
AU6019900A (en) * 1999-11-24 2001-06-04 Sumika Fine Chemicals Co., Ltd. Anhydrous mirtazapine crystals and process for producing the same
WO2016209996A1 (fr) * 2015-06-23 2016-12-29 University Of Oregon Hétérocycles contenant du phosphore et procédé de production et d'utilisation

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8308063D0 (en) * 1983-03-24 1983-05-05 Beecham Group Plc Active compounds
DE3479726D1 (de) * 1983-05-18 1989-10-19 Beecham Group Plc Benzopyran derivatives.
EP0139992B1 (fr) * 1983-09-01 1988-12-28 Beecham Group Plc Dérivés du chromanol
GB8324547D0 (en) * 1983-09-14 1983-10-19 Beecham Group Plc Compounds
US4824968A (en) * 1984-12-12 1989-04-25 Merck & Co., Inc. Substituted aromatic sulfonamides as antiglaucoma agents
US4797413A (en) * 1986-05-14 1989-01-10 Merck & Co., Inc. Thieno thiopyran sulfonamide derivatives, pharmaceutical compositions and use
DE3682331D1 (de) * 1985-06-08 1991-12-12 Beecham Group Plc Pyrano(3,2-c)pyridinderivate, verfahren und zwischenprodukte zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen.
GB8515207D0 (en) * 1985-06-15 1985-07-17 Boots Co Plc Therapeutic agents
GB8613786D0 (en) * 1986-06-06 1986-07-09 Beecham Group Plc Active compounds
GB8627698D0 (en) * 1986-11-20 1986-12-17 Boots Co Plc Therapeutic agents
US5030736A (en) * 1988-09-23 1991-07-09 Ortho Pharmaceutical Corporation Substituted thienopyrans
US4992465A (en) * 1988-09-27 1991-02-12 Ciba-Geigy Corporation 3-amino-dihydro-(1)-benzopyrans
IE63935B1 (en) * 1989-06-27 1995-06-28 Chem Pharm Forsch Gmbh Novel thienopyran derivatives a process for their preparation and their use
US5120757A (en) * 1989-07-31 1992-06-09 Merck & Co., Inc. Substituted aromatic sulfonamides as antiglaucoma agents
DE3925719A1 (de) * 1989-08-03 1991-02-07 Bayer Ag Substituierte thienopyranone, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung von parasiten

Also Published As

Publication number Publication date
CN1042152A (zh) 1990-05-16
US5284857A (en) 1994-02-08
KR920008824B1 (ko) 1992-10-09
JPH02174781A (ja) 1990-07-06
IE893045L (en) 1990-03-23
IL91709A0 (en) 1990-06-10
IL91709A (en) 1994-07-31
PH30818A (en) 1997-10-17
PT91787A (pt) 1990-03-30
EP0360621B1 (fr) 1994-01-19
DE68912476D1 (de) 1994-03-03
DE68912476T2 (de) 1994-05-19
NO893775D0 (no) 1989-09-22
EP0360621A1 (fr) 1990-03-28
DK469189A (da) 1990-03-24
HUT54162A (en) 1991-01-28
ES2062027T3 (es) 1994-12-16
NZ230711A (en) 1990-10-26
NO172802B (no) 1993-06-01
PT91787B (pt) 1995-05-31
IE63301B1 (en) 1995-04-05
DK469189D0 (da) 1989-09-22
US5378713A (en) 1995-01-03
FI894491A (fi) 1990-03-24
AU619896B2 (en) 1992-02-06
FI894491A0 (fi) 1989-09-22
KR900004745A (ko) 1990-04-12
CN1032210C (zh) 1996-07-03
MY129947A (en) 2007-05-31
NO893775L (no) 1990-03-26
AU4170889A (en) 1990-03-29
CA1338419C (fr) 1996-06-25
PH30773A (en) 1997-10-17

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