NL193818B - Farmaceutisch vast preparaat voor vertraagde en beheerste afgifte van een therapeutisch werkzame polypeptide verbinding. - Google Patents

Farmaceutisch vast preparaat voor vertraagde en beheerste afgifte van een therapeutisch werkzame polypeptide verbinding.

Info

Publication number
NL193818B
NL193818B NL8802323A NL8802323A NL193818B NL 193818 B NL193818 B NL 193818B NL 8802323 A NL8802323 A NL 8802323A NL 8802323 A NL8802323 A NL 8802323A NL 193818 B NL193818 B NL 193818B
Authority
NL
Netherlands
Prior art keywords
delayed
controlled release
therapeutically active
solid preparation
active polypeptide
Prior art date
Application number
NL8802323A
Other languages
English (en)
Other versions
NL193818C (nl
NL8802323A (nl
Original Assignee
Debiopharm Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Debiopharm Sa filed Critical Debiopharm Sa
Publication of NL8802323A publication Critical patent/NL8802323A/nl
Publication of NL193818B publication Critical patent/NL193818B/nl
Application granted granted Critical
Publication of NL193818C publication Critical patent/NL193818C/nl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
NL8802323A 1987-09-21 1988-09-20 Farmaceutisch vast preparaat voor vertraagde en beheerste afgifte van een therapeutisch werkzame polypeptide verbinding. NL193818C (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8722134 1987-09-21
GB8722134A GB2209937B (en) 1987-09-21 1987-09-21 Water insoluble polypeptides

Publications (3)

Publication Number Publication Date
NL8802323A NL8802323A (nl) 1989-04-17
NL193818B true NL193818B (nl) 2000-08-01
NL193818C NL193818C (nl) 2000-12-04

Family

ID=10624108

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8802323A NL193818C (nl) 1987-09-21 1988-09-20 Farmaceutisch vast preparaat voor vertraagde en beheerste afgifte van een therapeutisch werkzame polypeptide verbinding.

Country Status (23)

Country Link
US (2) US5192741A (nl)
JP (1) JPH0713023B2 (nl)
AT (1) AT397035B (nl)
AU (1) AU611944B2 (nl)
BE (1) BE1001685A5 (nl)
CA (1) CA1326438C (nl)
CH (1) CH675968A5 (nl)
DE (2) DE122004000023I2 (nl)
DK (1) DK175311B1 (nl)
ES (1) ES2009346A6 (nl)
FI (1) FI96919C (nl)
FR (1) FR2620621B1 (nl)
GB (1) GB2209937B (nl)
GR (1) GR1002244B (nl)
IE (1) IE60608B1 (nl)
IL (1) IL87790A (nl)
IT (1) IT1225148B (nl)
LU (1) LU87340A1 (nl)
NL (1) NL193818C (nl)
NO (2) NO178604C (nl)
PT (1) PT88557B (nl)
SE (1) SE503406C2 (nl)
ZA (1) ZA886827B (nl)

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SE8803321L (sv) 1989-03-22
IL87790A (en) 1992-05-25
AU611944B2 (en) 1991-06-27
SE503406C2 (sv) 1996-06-10
IT1225148B (it) 1990-11-02
NO884154L (no) 1989-03-22
CH675968A5 (nl) 1990-11-30
DK175311B1 (da) 2004-08-16
PT88557A (pt) 1988-10-01
JPH01121222A (ja) 1989-05-12
IE882727L (en) 1989-03-21
NL193818C (nl) 2000-12-04
PT88557B (pt) 1992-11-30
ATA223488A (de) 1993-06-15
BE1001685A5 (fr) 1990-02-06
GB2209937A (en) 1989-06-01
CA1326438C (en) 1994-01-25
DE3822459C2 (de) 1994-07-07
JPH0713023B2 (ja) 1995-02-15
NO2005012I2 (no) 2008-12-01
NO884154D0 (no) 1988-09-19
ES2009346A6 (es) 1989-09-16
NL8802323A (nl) 1989-04-17
AT397035B (de) 1994-01-25
GR880100619A (el) 1989-06-22
IE60608B1 (en) 1994-07-27
GB2209937B (en) 1991-07-03
LU87340A1 (fr) 1989-04-06
SE8803321D0 (sv) 1988-09-20
FR2620621B1 (fr) 1993-02-19
AU2232688A (en) 1989-03-23
NO178604B (no) 1996-01-22
US5192741A (en) 1993-03-09
DE3822459A1 (de) 1989-03-30
IL87790A0 (en) 1989-03-31
DK518988A (da) 1989-03-22
ZA886827B (en) 1989-05-30
FI884297A0 (fi) 1988-09-19
IT8805213A0 (it) 1988-09-20
US5776885A (en) 1998-07-07
FR2620621A1 (fr) 1989-03-24
FI884297A (fi) 1989-03-22
DE122004000023I2 (de) 2009-05-07
GR1002244B (en) 1996-04-22
GB8722134D0 (en) 1987-10-28
FI96919B (fi) 1996-06-14
DK518988D0 (da) 1988-09-16
NO178604C (no) 1996-05-02
FI96919C (fi) 1996-09-25

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