MXPA03010596A - Preparaciones granuladas de gaboxadol. - Google Patents
Preparaciones granuladas de gaboxadol.Info
- Publication number
- MXPA03010596A MXPA03010596A MXPA03010596A MXPA03010596A MXPA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A MX PA03010596 A MXPA03010596 A MX PA03010596A
- Authority
- MX
- Mexico
- Prior art keywords
- gaboxadol
- granular preparations
- preparation
- granular
- dosage forms
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Inorganic Chemistry (AREA)
- Anesthesiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
La presente invencion se relaciona con un producto granulado que contiene gaboxadol como sal de adicion de acido, con un proceso de granulacion en fusion para la preparacion del mismo y con formas de dosificacion unitaria farmaceuticas macizas preparadas con dicha preparacion granulada de gaboxadol.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200100817 | 2001-05-21 | ||
| PCT/DK2002/000332 WO2002094225A1 (en) | 2001-05-21 | 2002-05-17 | Granular preparations of gaboxadol |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03010596A true MXPA03010596A (es) | 2004-03-09 |
Family
ID=8160520
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03010596A MXPA03010596A (es) | 2001-05-21 | 2002-05-17 | Preparaciones granuladas de gaboxadol. |
Country Status (26)
| Country | Link |
|---|---|
| US (1) | US20040157876A1 (es) |
| EP (1) | EP1389091A1 (es) |
| JP (1) | JP2004530695A (es) |
| KR (1) | KR20030097890A (es) |
| CN (1) | CN1511026A (es) |
| AR (1) | AR033896A1 (es) |
| AU (1) | AU2002338855B2 (es) |
| BG (1) | BG108441A (es) |
| BR (1) | BR0209834A (es) |
| CA (1) | CA2447603A1 (es) |
| CZ (1) | CZ20033269A3 (es) |
| EA (2) | EA009731B1 (es) |
| HR (1) | HRP20030950A2 (es) |
| HU (1) | HUP0400051A2 (es) |
| IL (1) | IL158733A0 (es) |
| IS (1) | IS7020A (es) |
| ME (1) | MEP6308A (es) |
| MX (1) | MXPA03010596A (es) |
| NO (1) | NO20035146L (es) |
| NZ (1) | NZ547636A (es) |
| PL (1) | PL366541A1 (es) |
| SK (1) | SK15542003A3 (es) |
| UA (1) | UA80092C2 (es) |
| WO (1) | WO2002094225A1 (es) |
| YU (1) | YU92103A (es) |
| ZA (1) | ZA200308594B (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001022941A1 (en) * | 1999-09-28 | 2001-04-05 | H. Lundbeck A/S | Melt granulated composition and modified release dosage form prepared from said composition |
| PT1641456E (pt) | 2003-06-25 | 2010-06-01 | Lundbeck & Co As H | Gaboxadol para o tratamento de depressão e outros distúrbios afectivos |
| TW200528098A (en) * | 2003-12-18 | 2005-09-01 | Lundbeck & Co As H | Treatment of insomnia in human patients |
| GB0402118D0 (en) | 2004-01-30 | 2004-03-03 | Merck Sharp & Dohme | Polymorphic forms of a GABAA agonist |
| WO2006083682A2 (en) | 2005-01-28 | 2006-08-10 | H.Lundbeck A/S | Polymorphic forms of a gabaa agonist |
| EP1906953A4 (en) * | 2005-04-29 | 2009-05-20 | Lundbeck & Co As H | FORMS OF ACID SALTS AND BASIC SALTS OF GABOXADOL |
| EP2374459A1 (en) * | 2008-05-30 | 2011-10-12 | Psychogenics Inc. | Treatment for neurological and mental disorders |
| CA2732636A1 (en) * | 2008-09-01 | 2009-05-07 | H. Lundbeck A/S | Pharmaceutical composition comprising gaboxadol and an inhibitor of pat1 or oat |
| EP4035683A1 (en) * | 2011-12-12 | 2022-08-03 | Adare Pharmaceuticals USA, Inc. | Sustained release particle formulations |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4315934A (en) * | 1979-09-24 | 1982-02-16 | Sandoz Ltd. | Organic compounds |
| DE19525598C2 (de) * | 1995-07-13 | 1997-09-25 | Max Planck Gesellschaft | Schlafmittel |
| US6649186B1 (en) * | 1996-09-20 | 2003-11-18 | Ethypharm | Effervescent granules and methods for their preparation |
| WO2001022941A1 (en) * | 1999-09-28 | 2001-04-05 | H. Lundbeck A/S | Melt granulated composition and modified release dosage form prepared from said composition |
| US6375982B1 (en) * | 2000-07-05 | 2002-04-23 | Capricorn Pharma, Inc. | Rapid-melt semi-solid compositions, methods of making same and method of using same |
-
2002
- 2002-05-17 WO PCT/DK2002/000332 patent/WO2002094225A1/en active Application Filing
- 2002-05-17 PL PL02366541A patent/PL366541A1/xx not_active Application Discontinuation
- 2002-05-17 HU HU0400051A patent/HUP0400051A2/hu unknown
- 2002-05-17 AR ARP020101839A patent/AR033896A1/es unknown
- 2002-05-17 CZ CZ20033269A patent/CZ20033269A3/cs unknown
- 2002-05-17 CN CNA028104587A patent/CN1511026A/zh active Pending
- 2002-05-17 NZ NZ547636A patent/NZ547636A/en unknown
- 2002-05-17 SK SK1554-2003A patent/SK15542003A3/sk not_active Application Discontinuation
- 2002-05-17 US US10/478,983 patent/US20040157876A1/en not_active Abandoned
- 2002-05-17 ME MEP-63/08A patent/MEP6308A/xx unknown
- 2002-05-17 CA CA002447603A patent/CA2447603A1/en not_active Abandoned
- 2002-05-17 YU YU92103A patent/YU92103A/sh unknown
- 2002-05-17 MX MXPA03010596A patent/MXPA03010596A/es not_active Application Discontinuation
- 2002-05-17 AU AU2002338855A patent/AU2002338855B2/en not_active Ceased
- 2002-05-17 KR KR10-2003-7015136A patent/KR20030097890A/ko not_active Application Discontinuation
- 2002-05-17 EP EP02742834A patent/EP1389091A1/en not_active Ceased
- 2002-05-17 EA EA200301282A patent/EA009731B1/ru not_active IP Right Cessation
- 2002-05-17 JP JP2002590944A patent/JP2004530695A/ja active Pending
- 2002-05-17 BR BR0209834-2A patent/BR0209834A/pt not_active IP Right Cessation
- 2002-05-17 EA EA200700703A patent/EA200700703A1/ru unknown
- 2002-05-17 IL IL15873302A patent/IL158733A0/xx unknown
- 2002-05-17 UA UA20031110120A patent/UA80092C2/uk unknown
-
2003
- 2003-11-04 ZA ZA200308594A patent/ZA200308594B/en unknown
- 2003-11-10 IS IS7020A patent/IS7020A/is unknown
- 2003-11-19 NO NO20035146A patent/NO20035146L/no not_active Application Discontinuation
- 2003-11-21 HR HR20030950A patent/HRP20030950A2/hr not_active Application Discontinuation
- 2003-12-12 BG BG108441A patent/BG108441A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1389091A1 (en) | 2004-02-18 |
| PL366541A1 (en) | 2005-02-07 |
| IS7020A (is) | 2003-11-10 |
| UA80092C2 (en) | 2007-08-27 |
| AR033896A1 (es) | 2004-01-07 |
| SK15542003A3 (sk) | 2004-05-04 |
| IL158733A0 (en) | 2004-05-12 |
| AU2002338855B2 (en) | 2007-08-16 |
| JP2004530695A (ja) | 2004-10-07 |
| KR20030097890A (ko) | 2003-12-31 |
| WO2002094225A1 (en) | 2002-11-28 |
| CN1511026A (zh) | 2004-07-07 |
| CZ20033269A3 (en) | 2004-03-17 |
| NZ547636A (en) | 2008-03-28 |
| ZA200308594B (en) | 2004-11-04 |
| EA200700703A1 (ru) | 2007-08-31 |
| HUP0400051A2 (hu) | 2004-04-28 |
| BR0209834A (pt) | 2004-06-15 |
| EA200301282A1 (ru) | 2004-04-29 |
| NO20035146D0 (no) | 2003-11-19 |
| YU92103A (sh) | 2006-05-25 |
| NO20035146L (no) | 2003-11-19 |
| US20040157876A1 (en) | 2004-08-12 |
| EA009731B1 (ru) | 2008-02-28 |
| MEP6308A (xx) | 2010-02-10 |
| CA2447603A1 (en) | 2002-11-28 |
| HRP20030950A2 (en) | 2005-08-31 |
| BG108441A (en) | 2005-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |