MX9203787A - Composicion farmaceutica que contiene un portador farmaceuticamente adecuado y el compuesto que contiene la estructura (7 alfa, 17 alfa)-17-hidroxi-7-metil-19-nor-17-pregn-5(10)-en 20-in-3-ona. - Google Patents

Composicion farmaceutica que contiene un portador farmaceuticamente adecuado y el compuesto que contiene la estructura (7 alfa, 17 alfa)-17-hidroxi-7-metil-19-nor-17-pregn-5(10)-en 20-in-3-ona.

Info

Publication number
MX9203787A
MX9203787A MX9203787A MX9203787A MX9203787A MX 9203787 A MX9203787 A MX 9203787A MX 9203787 A MX9203787 A MX 9203787A MX 9203787 A MX9203787 A MX 9203787A MX 9203787 A MX9203787 A MX 9203787A
Authority
MX
Mexico
Prior art keywords
alpha
pregn
methyl
pharmaceutical composition
hidroxi
Prior art date
Application number
MX9203787A
Other languages
English (en)
Inventor
Gerard Arnoud Jozef Maria Sas
Emili Martin Van Doornum
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=19854317&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX9203787(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of MX9203787A publication Critical patent/MX9203787A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
MX9203787A 1989-03-18 1992-06-29 Composicion farmaceutica que contiene un portador farmaceuticamente adecuado y el compuesto que contiene la estructura (7 alfa, 17 alfa)-17-hidroxi-7-metil-19-nor-17-pregn-5(10)-en 20-in-3-ona. MX9203787A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
NL8900673 1989-03-18

Publications (1)

Publication Number Publication Date
MX9203787A true MX9203787A (es) 1992-07-01

Family

ID=19854317

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9203787A MX9203787A (es) 1989-03-18 1992-06-29 Composicion farmaceutica que contiene un portador farmaceuticamente adecuado y el compuesto que contiene la estructura (7 alfa, 17 alfa)-17-hidroxi-7-metil-19-nor-17-pregn-5(10)-en 20-in-3-ona.

Country Status (17)

Country Link
US (1) US5037817A (es)
EP (1) EP0389035B1 (es)
JP (2) JP3139709B2 (es)
KR (1) KR0183401B1 (es)
AT (1) ATE98490T1 (es)
AU (1) AU625083B2 (es)
CA (1) CA2011452C (es)
DE (1) DE69005165T2 (es)
DK (1) DK0389035T3 (es)
ES (1) ES2062292T3 (es)
FI (1) FI94865C (es)
HK (1) HK1002019A1 (es)
IE (1) IE63051B1 (es)
MX (1) MX9203787A (es)
NZ (1) NZ232946A (es)
PT (1) PT93488B (es)
ZA (1) ZA901674B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE180669T1 (de) * 1993-03-05 1999-06-15 Akzo Nobel Nv Verwendung von pregnanderivaten zur behandlung von tumoren
US6242434B1 (en) * 1997-08-08 2001-06-05 Bone Care International, Inc. 24-hydroxyvitamin D, analogs and uses thereof
IL123984A (en) * 1997-04-22 2004-09-27 Akzo Nobel Nv Pharmacological dosage units containing tibolone and carrier pharmacy are acceptable
PL197870B1 (pl) * 1998-10-16 2008-05-30 Organon Nv Kompozycja o wysokiej czystości zawierająca (7α, 17α)-17-hydroksy-7-metylo-19-nor-17-pregn-5-(10)-en-20-yn-3-on, sposób wytwarzania tej kompozycji i farmaceutyczna jednostka dawkowania
US7045513B1 (en) 1999-03-18 2006-05-16 Genelabs Technologies, Inc. DHEA composition and method
AU779138B2 (en) * 1999-03-18 2005-01-06 Genelabs Technologies, Inc. DHEA composition and method
TWI265167B (en) * 1999-11-29 2006-11-01 Akzo Nobel Nv 3-methylene steroid derivatives
US20040229854A1 (en) * 2000-11-28 2004-11-18 Pieter Haan De Immediate release dosage form for HRT
ATE364619T1 (de) * 2001-10-18 2007-07-15 Norton Healthcare Ltd Tibolonformulierungen
GB0125061D0 (en) * 2001-10-18 2001-12-12 Norton Healthcare Ltd Pharmaceutical composition
CN1620298A (zh) * 2002-01-22 2005-05-25 阿克佐诺贝尔公司 替勃龙用于治疗与施用阻止内源性***合成的药物有关的疾病
GB0304927D0 (en) 2003-03-04 2003-04-09 Resolution Chemicals Ltd Process for the production of tibolone
CN1324041C (zh) * 2003-04-01 2007-07-04 上海迪赛诺医药科技开发有限公司 替勃龙晶型i的制备方法
PL1499278T3 (pl) * 2003-05-23 2005-09-30 Msd Oss Bv Farmaceutyczna postać użytkowa o natychmiastowym uwalnianiu zawierająca polimorficzny tibolon
EP1883648A1 (en) * 2005-05-23 2008-02-06 Newchem S.p.A. Process for the preparation of pure crystalline tibolone
EP1821571A1 (en) * 2006-02-15 2007-08-22 Oticon A/S Loop antenna for in the ear audio device
ITMI20130120A1 (it) * 2013-01-25 2014-07-26 Ind Chimica Srl Processo per la preparazione in forma cristallina di tibolone, (7alfa,17alfa)-17-idrossi-7-metil-19-norpregn-5(10)-en-20-in-3-one
US10736907B2 (en) 2016-05-04 2020-08-11 Novalon S.A. Use of sugar-alcohols in tibolone compositions

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE665514A (es) * 1964-06-16
US4933168A (en) * 1975-05-27 1990-06-12 Syntex Pharmaceuticals International Limited Stable, crystalline flunisolide
US4273710A (en) * 1979-05-21 1981-06-16 Syntex Corporation Process for preparing flunisolide
US4447426A (en) * 1982-01-18 1984-05-08 E. R. Squibb & Sons, Inc. Steroid monohydrates, formulations containing same and method
US4391755A (en) * 1982-01-18 1983-07-05 E. R. Squibb & Sons, Inc. Steroid monohydrates, formulations containing same and method
US4701450A (en) * 1984-03-21 1987-10-20 Akzo N.V. Steroids for use as immunomodulators

Also Published As

Publication number Publication date
HK1002019A1 (en) 1998-07-24
JPH0347195A (ja) 1991-02-28
US5037817A (en) 1991-08-06
AU625083B2 (en) 1992-07-02
ATE98490T1 (de) 1994-01-15
FI901328A0 (fi) 1990-03-16
IE63051B1 (en) 1995-03-22
DE69005165T2 (de) 1994-05-05
ES2062292T3 (es) 1994-12-16
CA2011452C (en) 1999-05-25
DE69005165D1 (de) 1994-01-27
EP0389035B1 (en) 1993-12-15
JP3139709B2 (ja) 2001-03-05
KR900013950A (ko) 1990-10-22
IE900709L (en) 1990-09-18
DK0389035T3 (da) 1994-02-14
FI94865B (fi) 1995-07-31
PT93488B (pt) 1996-02-29
FI94865C (fi) 1995-11-10
ZA901674B (en) 1990-12-28
PT93488A (pt) 1990-11-07
CA2011452A1 (en) 1990-09-18
KR0183401B1 (ko) 1999-05-01
AU5139490A (en) 1990-09-20
EP0389035A1 (en) 1990-09-26
JP2001139473A (ja) 2001-05-22
NZ232946A (en) 1991-08-27

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